Assay ID | Title | Year | Journal | Article |
AID1581820 | Inhibition of ERAP1 in human HeLa cells stably expressing H-2 Kb infected with vaccinia virus containing ss-LEQLE-SIINFEKL epitope assessed as suppression of ss-LEQLE-SIINFEKL binding to MHC1 H-2 Kb at cell surface by measuring reduction in 25D1 staining | 2020 | Journal of medicinal chemistry, 01-09, Volume: 63, Issue:1
| Discovery of Selective Inhibitors of Endoplasmic Reticulum Aminopeptidase 1. |
AID1581821 | Inhibition of TAP1/2 in human HeLa cells stably expressing H-2 Kb infected with vaccinia virus containing Ub-SIINFEKL epitope assessed as suppression of Ub-SIINFEKL binding to MHC1 H-2 Kb at cell surface by measuring reduction in 25D1 staining at 50 uM me | 2020 | Journal of medicinal chemistry, 01-09, Volume: 63, Issue:1
| Discovery of Selective Inhibitors of Endoplasmic Reticulum Aminopeptidase 1. |
AID35689 | Inhibition of partially purified soluble aminopeptidase from rat brain | 1988 | Journal of medicinal chemistry, Nov, Volume: 31, Issue:11
| Design of novel inhibitors of aminopeptidases. Synthesis of peptide-derived diamino thiols and sulfur replacement analogues of bestatin. |
AID38370 | Inhibition of pig kidney Aminopeptidase N | 1999 | Bioorganic & medicinal chemistry letters, Jun-07, Volume: 9, Issue:11
| Design of the first highly potent and selective aminopeptidase N (EC 3.4.11.2) inhibitor. |
[information is prepared from bioassay data collected from National Library of Medicine (NLM), extracted Dec-2023] |