| Assay ID | Title | Year | Journal | Article |
|---|
| AID25302 | Apparent rate of cyclization (kobsd) value at pH 7.00(in 0.1 M acetate). | 1983 | Journal of medicinal chemistry, Oct, Volume: 26, Issue:10
| Aporphines. 50. Kinetics of solvolysis of N-(2-chloroethyl)norapomorphine, an irreversible dopamine receptor antagonist. |
| AID26677 | Half-life period at pH 6.50(in 0.1 M acetate). | 1983 | Journal of medicinal chemistry, Oct, Volume: 26, Issue:10
| Aporphines. 50. Kinetics of solvolysis of N-(2-chloroethyl)norapomorphine, an irreversible dopamine receptor antagonist. |
| AID62574 | Compound was evaluated at 100 uM concentration to displace [3H]spiperone and result indicates the percent displacement. | 1984 | Journal of medicinal chemistry, Jun, Volume: 27, Issue:6
| Aporphines. 58. N-(2-chloroethyl) [8,9-2H]norapomorphine, an irreversible ligand for dopamine receptors: synthesis and application. |
| AID26675 | Half-life period at pH 6.00(in 0.1 M acetate). | 1983 | Journal of medicinal chemistry, Oct, Volume: 26, Issue:10
| Aporphines. 50. Kinetics of solvolysis of N-(2-chloroethyl)norapomorphine, an irreversible dopamine receptor antagonist. |
| AID26676 | Half-life period at pH 6.25(in 0.1 M acetate). | 1983 | Journal of medicinal chemistry, Oct, Volume: 26, Issue:10
| Aporphines. 50. Kinetics of solvolysis of N-(2-chloroethyl)norapomorphine, an irreversible dopamine receptor antagonist. |
| AID25503 | Apparent rate of cyclization (kobsd) value at pH 7.50(in 0.1 M acetate). | 1983 | Journal of medicinal chemistry, Oct, Volume: 26, Issue:10
| Aporphines. 50. Kinetics of solvolysis of N-(2-chloroethyl)norapomorphine, an irreversible dopamine receptor antagonist. |
| AID25299 | Apparent rate of cyclization (kobsd) value at pH 6.25(in 0.1 M phosphate). | 1983 | Journal of medicinal chemistry, Oct, Volume: 26, Issue:10
| Aporphines. 50. Kinetics of solvolysis of N-(2-chloroethyl)norapomorphine, an irreversible dopamine receptor antagonist. |
| AID26673 | Half-life period at pH 5.60(in 0.1 M acetate). | 1983 | Journal of medicinal chemistry, Oct, Volume: 26, Issue:10
| Aporphines. 50. Kinetics of solvolysis of N-(2-chloroethyl)norapomorphine, an irreversible dopamine receptor antagonist. |
| AID34461 | Dopamine sensitive adenylate cyclase activity (stimulation) in homogenates of rat brain striatal tissue was assessed at 50 uM of compound; Inhibitis the cyclase activity | 1981 | Journal of medicinal chemistry, Dec, Volume: 24, Issue:12
| Aporphines, 36. Dopamine receptor interactions of trihydroxyaporphines. Synthesis, radioreceptor binding, and striatal adenylate cyclase stimulation of 2,10,11-trihydroxyaporphines in comparison with other hydroxylated aporphines. |
| AID26679 | Half-life period at pH 7.00(in 0.1 M acetate). | 1983 | Journal of medicinal chemistry, Oct, Volume: 26, Issue:10
| Aporphines. 50. Kinetics of solvolysis of N-(2-chloroethyl)norapomorphine, an irreversible dopamine receptor antagonist. |
| AID25298 | Apparent rate of cyclization (kobsd) value at pH 6.00(in 0.1 M phosphate). | 1983 | Journal of medicinal chemistry, Oct, Volume: 26, Issue:10
| Aporphines. 50. Kinetics of solvolysis of N-(2-chloroethyl)norapomorphine, an irreversible dopamine receptor antagonist. |
| AID25504 | Apparent rate of cyclization (kobsd) value at pH 8.00(in 0.1 M acetate). | 1983 | Journal of medicinal chemistry, Oct, Volume: 26, Issue:10
| Aporphines. 50. Kinetics of solvolysis of N-(2-chloroethyl)norapomorphine, an irreversible dopamine receptor antagonist. |
| AID26683 | Half-life period at pH 8.00(in 0.1 M acetate). | 1983 | Journal of medicinal chemistry, Oct, Volume: 26, Issue:10
| Aporphines. 50. Kinetics of solvolysis of N-(2-chloroethyl)norapomorphine, an irreversible dopamine receptor antagonist. |
| AID26682 | Half-life period at pH 7.50(in 0.1 M acetate). | 1983 | Journal of medicinal chemistry, Oct, Volume: 26, Issue:10
| Aporphines. 50. Kinetics of solvolysis of N-(2-chloroethyl)norapomorphine, an irreversible dopamine receptor antagonist. |
| AID25296 | Apparent rate of cyclization (kobsd) value at pH 5.60(in 0.1 M acetate). | 1983 | Journal of medicinal chemistry, Oct, Volume: 26, Issue:10
| Aporphines. 50. Kinetics of solvolysis of N-(2-chloroethyl)norapomorphine, an irreversible dopamine receptor antagonist. |
| AID62572 | Compound was evaluated for the competitive binding with [3H]spiperone binding to Canine striatal membranes. | 1984 | Journal of medicinal chemistry, Jun, Volume: 27, Issue:6
| Aporphines. 58. N-(2-chloroethyl) [8,9-2H]norapomorphine, an irreversible ligand for dopamine receptors: synthesis and application. |
| AID25301 | Apparent rate of cyclization (kobsd) value at pH 6.75(in 0.1 M phosphate). | 1983 | Journal of medicinal chemistry, Oct, Volume: 26, Issue:10
| Aporphines. 50. Kinetics of solvolysis of N-(2-chloroethyl)norapomorphine, an irreversible dopamine receptor antagonist. |
| AID26674 | Half-life period at pH 5.80(in 0.1 M acetate). | 1983 | Journal of medicinal chemistry, Oct, Volume: 26, Issue:10
| Aporphines. 50. Kinetics of solvolysis of N-(2-chloroethyl)norapomorphine, an irreversible dopamine receptor antagonist. |
| AID45982 | Inhibition of [3H]apomorphine binding to calf caudate membrane preparation (p4) | 1981 | Journal of medicinal chemistry, Dec, Volume: 24, Issue:12
| Aporphines, 36. Dopamine receptor interactions of trihydroxyaporphines. Synthesis, radioreceptor binding, and striatal adenylate cyclase stimulation of 2,10,11-trihydroxyaporphines in comparison with other hydroxylated aporphines. |
| AID45983 | Inhibition of [3H]spiroperidol binding to calf caudate membrane preparation (p4) | 1981 | Journal of medicinal chemistry, Dec, Volume: 24, Issue:12
| Aporphines, 36. Dopamine receptor interactions of trihydroxyaporphines. Synthesis, radioreceptor binding, and striatal adenylate cyclase stimulation of 2,10,11-trihydroxyaporphines in comparison with other hydroxylated aporphines. |
| AID25297 | Apparent rate of cyclization (kobsd) value at pH 5.80(in 0.1 M acetate). | 1983 | Journal of medicinal chemistry, Oct, Volume: 26, Issue:10
| Aporphines. 50. Kinetics of solvolysis of N-(2-chloroethyl)norapomorphine, an irreversible dopamine receptor antagonist. |
| AID26672 | Half-life period at pH 5.40(in 0.1 M acetate). | 1983 | Journal of medicinal chemistry, Oct, Volume: 26, Issue:10
| Aporphines. 50. Kinetics of solvolysis of N-(2-chloroethyl)norapomorphine, an irreversible dopamine receptor antagonist. |
| AID25300 | Apparent rate of cyclization (kobsd) value at pH 6.50(in 0.1 M phosphate). | 1983 | Journal of medicinal chemistry, Oct, Volume: 26, Issue:10
| Aporphines. 50. Kinetics of solvolysis of N-(2-chloroethyl)norapomorphine, an irreversible dopamine receptor antagonist. |
| AID25295 | Apparent rate of cyclization (kobsd) value at pH 5.40(in 0.1 M acetate). | 1983 | Journal of medicinal chemistry, Oct, Volume: 26, Issue:10
| Aporphines. 50. Kinetics of solvolysis of N-(2-chloroethyl)norapomorphine, an irreversible dopamine receptor antagonist. |
| AID26678 | Half-life period at pH 6.75(in 0.1 M acetate). | 1983 | Journal of medicinal chemistry, Oct, Volume: 26, Issue:10
| Aporphines. 50. Kinetics of solvolysis of N-(2-chloroethyl)norapomorphine, an irreversible dopamine receptor antagonist. |
| [information is prepared from bioassay data collected from National Library of Medicine (NLM), extracted Dec-2023] |