Assay ID | Title | Year | Journal | Article |
AID1347153 | Confirmatory screen GU AMC qHTS for Zika virus inhibitors | 2020 | Proceedings of the National Academy of Sciences of the United States of America, 12-08, Volume: 117, Issue:49
| Therapeutic candidates for the Zika virus identified by a high-throughput screen for Zika protease inhibitors. |
AID1347057 | CD47-SIRPalpha protein protein interaction - LANCE assay qHTS validation | 2019 | PloS one, , Volume: 14, Issue:7
| Quantitative high-throughput screening assays for the discovery and development of SIRPα-CD47 interaction inhibitors. |
AID1347169 | Tertiary RLuc qRT-PCR qHTS assay for Zika virus inhibitors | 2020 | Proceedings of the National Academy of Sciences of the United States of America, 12-08, Volume: 117, Issue:49
| Therapeutic candidates for the Zika virus identified by a high-throughput screen for Zika protease inhibitors. |
AID1347059 | CD47-SIRPalpha protein protein interaction - Alpha assay qHTS validation | 2019 | PloS one, , Volume: 14, Issue:7
| Quantitative high-throughput screening assays for the discovery and development of SIRPα-CD47 interaction inhibitors. |
AID1347152 | Confirmatory screen NINDS AMC qHTS for Zika virus inhibitors | 2020 | Proceedings of the National Academy of Sciences of the United States of America, 12-08, Volume: 117, Issue:49
| Therapeutic candidates for the Zika virus identified by a high-throughput screen for Zika protease inhibitors. |
AID1347168 | HepG2 cells viability qHTS for Zika virus inhibitors | 2020 | Proceedings of the National Academy of Sciences of the United States of America, 12-08, Volume: 117, Issue:49
| Therapeutic candidates for the Zika virus identified by a high-throughput screen for Zika protease inhibitors. |
AID1347405 | qHTS to identify inhibitors of the type 1 interferon - major histocompatibility complex class I in skeletal muscle: primary screen against the NCATS LOPAC collection | 2020 | ACS chemical biology, 07-17, Volume: 15, Issue:7
| High-Throughput Screening to Identify Inhibitors of the Type I Interferon-Major Histocompatibility Complex Class I Pathway in Skeletal Muscle. |
AID1347161 | Confirmatory screen NINDS Rhodamine qHTS for Zika virus inhibitors | 2020 | Proceedings of the National Academy of Sciences of the United States of America, 12-08, Volume: 117, Issue:49
| Therapeutic candidates for the Zika virus identified by a high-throughput screen for Zika protease inhibitors. |
AID1347167 | Vero cells viability qHTS for Zika virus inhibitors | 2020 | Proceedings of the National Academy of Sciences of the United States of America, 12-08, Volume: 117, Issue:49
| Therapeutic candidates for the Zika virus identified by a high-throughput screen for Zika protease inhibitors. |
AID1347410 | qHTS for inhibitors of adenylyl cyclases using a fission yeast platform: a pilot screen against the NCATS LOPAC library | 2019 | Cellular signalling, 08, Volume: 60 | A fission yeast platform for heterologous expression of mammalian adenylyl cyclases and high throughput screening. |
AID1347058 | CD47-SIRPalpha protein protein interaction - HTRF assay qHTS validation | 2019 | PloS one, , Volume: 14, Issue:7
| Quantitative high-throughput screening assays for the discovery and development of SIRPα-CD47 interaction inhibitors. |
AID1347151 | Optimization of GU AMC qHTS for Zika virus inhibitors: Unlinked NS2B-NS3 protease assay | 2020 | Proceedings of the National Academy of Sciences of the United States of America, 12-08, Volume: 117, Issue:49
| Therapeutic candidates for the Zika virus identified by a high-throughput screen for Zika protease inhibitors. |
AID1347149 | Furin counterscreen qHTS for Zika virus inhibitors | 2020 | Proceedings of the National Academy of Sciences of the United States of America, 12-08, Volume: 117, Issue:49
| Therapeutic candidates for the Zika virus identified by a high-throughput screen for Zika protease inhibitors. |
AID1347159 | Primary screen GU Rhodamine qHTS for Zika virus inhibitors: Unlinked NS2B-NS3 protease assay | 2020 | Proceedings of the National Academy of Sciences of the United States of America, 12-08, Volume: 117, Issue:49
| Therapeutic candidates for the Zika virus identified by a high-throughput screen for Zika protease inhibitors. |
AID1296008 | Cytotoxic Profiling of Annotated Libraries Using Quantitative High-Throughput Screening | 2020 | SLAS discovery : advancing life sciences R & D, 01, Volume: 25, Issue:1
| Cytotoxic Profiling of Annotated and Diverse Chemical Libraries Using Quantitative High-Throughput Screening. |
AID1347160 | Primary screen NINDS Rhodamine qHTS for Zika virus inhibitors | 2020 | Proceedings of the National Academy of Sciences of the United States of America, 12-08, Volume: 117, Issue:49
| Therapeutic candidates for the Zika virus identified by a high-throughput screen for Zika protease inhibitors. |
AID1346986 | P-glycoprotein substrates identified in KB-3-1 adenocarcinoma cell line, qHTS therapeutic library screen | 2019 | Molecular pharmacology, 11, Volume: 96, Issue:5
| A High-Throughput Screen of a Library of Therapeutics Identifies Cytotoxic Substrates of P-glycoprotein. |
AID1346987 | P-glycoprotein substrates identified in KB-8-5-11 adenocarcinoma cell line, qHTS therapeutic library screen | 2019 | Molecular pharmacology, 11, Volume: 96, Issue:5
| A High-Throughput Screen of a Library of Therapeutics Identifies Cytotoxic Substrates of P-glycoprotein. |
AID146736 | Binding affinity for human Neuropeptide Y4 receptor; No affinity | 2002 | Bioorganic & medicinal chemistry letters, Feb-11, Volume: 12, Issue:3
| Dihydropyridine neuropeptide Y Y(1) receptor antagonists. |
AID174813 | Ability to decrease spontaneous nocturnal food intake at 10 mg/kg (ip) in rats | 2002 | Bioorganic & medicinal chemistry letters, Feb-11, Volume: 12, Issue:3
| Dihydropyridine neuropeptide Y Y(1) receptor antagonists. |
AID146767 | Binding affinity for human Neuropeptide Y5 receptor; No affinity | 2002 | Bioorganic & medicinal chemistry letters, Feb-11, Volume: 12, Issue:3
| Dihydropyridine neuropeptide Y Y(1) receptor antagonists. |
AID669655 | Competitive displacement of [125I]peptideYY from NPY1 receptor in human SK-N-MC cells at 50 nM by equilibrium binding assay | 2012 | ACS medicinal chemistry letters, Mar-08, Volume: 3, Issue:3
| Discovery of a Novel Class of Bicyclo[3.1.0]hexanylpiperazines as Noncompetitive Neuropeptide Y Y1 Antagonists. |
AID146581 | Inhibition of binding of [125I]PYY radioligand to human neuropeptide Y1 receptor in SK-N-MC cell membrane | 2002 | Bioorganic & medicinal chemistry letters, Feb-11, Volume: 12, Issue:3
| Dihydropyridine neuropeptide Y Y(1) receptor antagonists. |
AID174814 | Ability to decrease spontaneous nocturnal food intake at 20 mg/kg (ip) in rats | 2002 | Bioorganic & medicinal chemistry letters, Feb-11, Volume: 12, Issue:3
| Dihydropyridine neuropeptide Y Y(1) receptor antagonists. |
AID174816 | Ability to inhibit food consumption increased by 10 ug icv infusion of NPY followed by compound administered at 30 mg/kg (ip) in satiated rats | 2002 | Bioorganic & medicinal chemistry letters, Feb-11, Volume: 12, Issue:3
| Dihydropyridine neuropeptide Y Y(1) receptor antagonists. |
AID146439 | Binding affinity against Neuropeptide Y receptor type 1 using I-PYY as a radioligand in human neuroblastoma SK-N-MC cells | 2002 | Bioorganic & medicinal chemistry letters, Feb-11, Volume: 12, Issue:3
| Novel dihydropyrazine analogues as NPY antagonists. |
AID174815 | Ability to inhibit food consumption increased by 10 ug icv infusion of NPY followed by compound administered at 10 mg/kg (ip) in satiated rats | 2002 | Bioorganic & medicinal chemistry letters, Feb-11, Volume: 12, Issue:3
| Dihydropyridine neuropeptide Y Y(1) receptor antagonists. |
AID146576 | Ability to inhibit human Neuropeptide Y1 receptor evaluated via forskolin-stimulated c-AMP accumulation in chinese hamster (CHO) cells | 2002 | Bioorganic & medicinal chemistry letters, Feb-11, Volume: 12, Issue:3
| Dihydropyridine neuropeptide Y Y(1) receptor antagonists. |
AID146603 | Binding affinity for human Neuropeptide Y2 receptor; No affinity | 2002 | Bioorganic & medicinal chemistry letters, Feb-11, Volume: 12, Issue:3
| Dihydropyridine neuropeptide Y Y(1) receptor antagonists. |
AID1794808 | Fluorescence-based screening to identify small molecule inhibitors of Plasmodium falciparum apicoplast DNA polymerase (Pf-apPOL). | 2014 | Journal of biomolecular screening, Jul, Volume: 19, Issue:6
| A High-Throughput Assay to Identify Inhibitors of the Apicoplast DNA Polymerase from Plasmodium falciparum. |
AID1794808 | Fluorescence-based screening to identify small molecule inhibitors of Plasmodium falciparum apicoplast DNA polymerase (Pf-apPOL). | | | |
[information is prepared from bioassay data collected from National Library of Medicine (NLM), extracted Dec-2023] |