Assay ID | Title | Year | Journal | Article |
AID512345 | Inhibition of His-tagged human LCK expressed in Sf9 cells at 1 uM | 2000 | The Biochemical journal, Oct-01, Volume: 351, Issue:Pt 1
| Specificity and mechanism of action of some commonly used protein kinase inhibitors. |
AID512338 | Inhibition of His-tagged human SGK expressed in Sf9 cells at 1 uM | 2000 | The Biochemical journal, Oct-01, Volume: 351, Issue:Pt 1
| Specificity and mechanism of action of some commonly used protein kinase inhibitors. |
AID512334 | Inhibition of bovine heart PKA at 1 uM | 2000 | The Biochemical journal, Oct-01, Volume: 351, Issue:Pt 1
| Specificity and mechanism of action of some commonly used protein kinase inhibitors. |
AID512344 | Inhibition of PHK from rabbit skeletal muscle at 1 uM | 2000 | The Biochemical journal, Oct-01, Volume: 351, Issue:Pt 1
| Specificity and mechanism of action of some commonly used protein kinase inhibitors. |
AID512339 | Inhibition of His-tagged human S6K1 expressed in Escherichia coli at 1 uM | 2000 | The Biochemical journal, Oct-01, Volume: 351, Issue:Pt 1
| Specificity and mechanism of action of some commonly used protein kinase inhibitors. |
AID512342 | Inhibition of rat liver AMPK at 1 uM | 2000 | The Biochemical journal, Oct-01, Volume: 351, Issue:Pt 1
| Specificity and mechanism of action of some commonly used protein kinase inhibitors. |
AID512340 | Inhibition of His-tagged human GSK3b expressed in Sf21 cells at 1 uM | 2000 | The Biochemical journal, Oct-01, Volume: 351, Issue:Pt 1
| Specificity and mechanism of action of some commonly used protein kinase inhibitors. |
AID512343 | Inhibition of His-tagged human CK2 expressed in Sf9 cells at 1 uM | 2000 | The Biochemical journal, Oct-01, Volume: 351, Issue:Pt 1
| Specificity and mechanism of action of some commonly used protein kinase inhibitors. |
AID409445 | Inhibition of Ca(2+))/phosphatidylserine/diacylglycerol-dependent aph8 phosphorylation in Streptomyces coelicolor cell lysate assessed as [32Pi] incorporation into aph8 at 500 nM by microplate scintillation counter relative to control | 2008 | Journal of medicinal chemistry, Dec-25, Volume: 51, Issue:24
| Search for inhibitors of bacterial and human protein kinases among derivatives of diazepines[1,4] annelated with maleimide and indole cycles. |
AID512327 | Inhibition of His-tagged human SAPK2b/p38b2 expressed in Escherichia coli at 1 uM | 2000 | The Biochemical journal, Oct-01, Volume: 351, Issue:Pt 1
| Specificity and mechanism of action of some commonly used protein kinase inhibitors. |
AID274367 | Inhibition of human recombinant SIRT2 | 2006 | Journal of medicinal chemistry, Dec-14, Volume: 49, Issue:25
| Adenosine mimetics as inhibitors of NAD+-dependent histone deacetylases, from kinase to sirtuin inhibition. |
AID512332 | Inhibition of His-tagged human MSK1 expressed in Sf9 cells at 1 uM | 2000 | The Biochemical journal, Oct-01, Volume: 351, Issue:Pt 1
| Specificity and mechanism of action of some commonly used protein kinase inhibitors. |
AID512323 | Inhibition of rabbit MKK1 expressed in Escherichia coli at 1 uM | 2000 | The Biochemical journal, Oct-01, Volume: 351, Issue:Pt 1
| Specificity and mechanism of action of some commonly used protein kinase inhibitors. |
AID512331 | Inhibition of His-tagged human MAPKAPK2 expressed in Escherichia coli at 1 uM | 2000 | The Biochemical journal, Oct-01, Volume: 351, Issue:Pt 1
| Specificity and mechanism of action of some commonly used protein kinase inhibitors. |
AID274372 | Inhibition of human recombinant SIRT2 by fluorescent deacetylase assay | 2006 | Journal of medicinal chemistry, Dec-14, Volume: 49, Issue:25
| Adenosine mimetics as inhibitors of NAD+-dependent histone deacetylases, from kinase to sirtuin inhibition. |
AID274371 | Inhibition of human SIRT1 by radioactive deacetylase assay | 2006 | Journal of medicinal chemistry, Dec-14, Volume: 49, Issue:25
| Adenosine mimetics as inhibitors of NAD+-dependent histone deacetylases, from kinase to sirtuin inhibition. |
AID512324 | Inhibition of His-tagged human MAPK2/ERK2 expressed in Escherichia coli at 1 uM | 2000 | The Biochemical journal, Oct-01, Volume: 351, Issue:Pt 1
| Specificity and mechanism of action of some commonly used protein kinase inhibitors. |
AID409446 | Inhibition of aph8-induced kanamycin phosphorylation in Streptomyces coelicolor cell lysate assessed as [32Pi] incorporation into kanamycin at 10 uM by microplate scintillation counter relative to control | 2008 | Journal of medicinal chemistry, Dec-25, Volume: 51, Issue:24
| Search for inhibitors of bacterial and human protein kinases among derivatives of diazepines[1,4] annelated with maleimide and indole cycles. |
AID512337 | Inhibition of human PKBalpha expressed in SF9 cells at 1 uM | 2000 | The Biochemical journal, Oct-01, Volume: 351, Issue:Pt 1
| Specificity and mechanism of action of some commonly used protein kinase inhibitors. |
AID512333 | Inhibition of His-tagged human PRAK expressed in Sf9 cells at 1 uM | 2000 | The Biochemical journal, Oct-01, Volume: 351, Issue:Pt 1
| Specificity and mechanism of action of some commonly used protein kinase inhibitors. |
AID512329 | Inhibition of His-tagged human SAPK4/p38delta expressed in Escherichia coli at 1 uM | 2000 | The Biochemical journal, Oct-01, Volume: 351, Issue:Pt 1
| Specificity and mechanism of action of some commonly used protein kinase inhibitors. |
AID274373 | Inhibition of human recombinant SIRT2 by radioactive deacetylase assay | 2006 | Journal of medicinal chemistry, Dec-14, Volume: 49, Issue:25
| Adenosine mimetics as inhibitors of NAD+-dependent histone deacetylases, from kinase to sirtuin inhibition. |
AID512325 | Inhibition of His-tagged human JNK1a1/SAPK1c expressed in Escherichia coli at 1 uM | 2000 | The Biochemical journal, Oct-01, Volume: 351, Issue:Pt 1
| Specificity and mechanism of action of some commonly used protein kinase inhibitors. |
AID274370 | Inhibition of human SIRT1 by fluorescent deacetylase assay | 2006 | Journal of medicinal chemistry, Dec-14, Volume: 49, Issue:25
| Adenosine mimetics as inhibitors of NAD+-dependent histone deacetylases, from kinase to sirtuin inhibition. |
AID512336 | Inhibition of His-tagged human PDK1 expressed in Sf21 cells at 1 uM | 2000 | The Biochemical journal, Oct-01, Volume: 351, Issue:Pt 1
| Specificity and mechanism of action of some commonly used protein kinase inhibitors. |
AID512326 | Inhibition of His-tagged human SAPK2a/p38 expressed in Escherichia coli at 1 uM | 2000 | The Biochemical journal, Oct-01, Volume: 351, Issue:Pt 1
| Specificity and mechanism of action of some commonly used protein kinase inhibitors. |
AID274366 | Inhibition of human SIRT1 | 2006 | Journal of medicinal chemistry, Dec-14, Volume: 49, Issue:25
| Adenosine mimetics as inhibitors of NAD+-dependent histone deacetylases, from kinase to sirtuin inhibition. |
AID512328 | Inhibition of His-tagged human SAPK3/p38gamma expressed in Escherichia coli at 1 uM | 2000 | The Biochemical journal, Oct-01, Volume: 351, Issue:Pt 1
| Specificity and mechanism of action of some commonly used protein kinase inhibitors. |
AID512335 | Inhibition of His-tagged human PKCalpha expressed in Escherichia coli at 1 uM | 2000 | The Biochemical journal, Oct-01, Volume: 351, Issue:Pt 1
| Specificity and mechanism of action of some commonly used protein kinase inhibitors. |
AID512346 | Inhibition of His-tagged human CHK1 expressed in Escherichia coli at 1 uM | 2000 | The Biochemical journal, Oct-01, Volume: 351, Issue:Pt 1
| Specificity and mechanism of action of some commonly used protein kinase inhibitors. |
AID512330 | Inhibition of MAPKAPK1b from rabbit skeletal muscle at 1 uM | 2000 | The Biochemical journal, Oct-01, Volume: 351, Issue:Pt 1
| Specificity and mechanism of action of some commonly used protein kinase inhibitors. |
AID165104 | Inhibition of rat brain protein kinase C (PKC) with ATP and histone as substrates | 1992 | Journal of medicinal chemistry, Jan, Volume: 35, Issue:1
| Inhibitors of protein kinase C. 1. 2,3-Bisarylmaleimides. |
AID512341 | Inhibition of rat ROCK2 expressed in Sf9 cells at 1 uM | 2000 | The Biochemical journal, Oct-01, Volume: 351, Issue:Pt 1
| Specificity and mechanism of action of some commonly used protein kinase inhibitors. |
AID1795401 | PKC assay from Article 10.1021/jm00079a024: \\Inhibitors of protein kinase C. 1. 2,3-Bisarylmaleimides.\\ | 1992 | Journal of medicinal chemistry, Jan, Volume: 35, Issue:1
| Inhibitors of protein kinase C. 1. 2,3-Bisarylmaleimides. |
AID1795412 | PKC assay from Article : \\The bisindolylmaleimide GF 109203X is a potent and selective inhibitor of protein kinase C.\\ | 1991 | The Journal of biological chemistry, Aug-25, Volume: 266, Issue:24
| The bisindolylmaleimide GF 109203X is a potent and selective inhibitor of protein kinase C. |
[information is prepared from bioassay data collected from National Library of Medicine (NLM), extracted Dec-2023] |