| Assay ID | Title | Year | Journal | Article |
|---|
| AID1322289 | Inhibition of human APN at <2 mM using AMC-labeled substrate preincubated for 30 mins followed by substrate addition by spectrofluorimetric method | 2016 | Bioorganic & medicinal chemistry letters, 11-01, Volume: 26, Issue:21
| Identification of methionine aminopeptidase 2 as a molecular target of the organoselenium drug ebselen and its derivatives/analogues: Synthesis, inhibitory activity and molecular modeling study. |
| AID1632339 | Steady state inhibition of Sporosarcina pasteurii CCM 2056 urease using urea as substrate assessed as inhibition constant for final enzyme conformation-inhibitor complex by measuring ammonia levels after 120 mins by phenol-hypochlorite method | 2016 | Journal of medicinal chemistry, 09-08, Volume: 59, Issue:17
| 1,2-Benzisoselenazol-3(2H)-one Derivatives As a New Class of Bacterial Urease Inhibitors. |
| AID1632340 | Competitive reversible inhibition of recombinant Helicobacter pylori urease infected in transformed Escherichia coli rosetta DE3 after 120 mins by Lineweaver-Burk plot analysis | 2016 | Journal of medicinal chemistry, 09-08, Volume: 59, Issue:17
| 1,2-Benzisoselenazol-3(2H)-one Derivatives As a New Class of Bacterial Urease Inhibitors. |
| AID1632343 | Inhibition of recombinant Helicobacter pylori urease expressed in Escherichia coli rosetta DE3 using urea as substrate assessed as transformed cell urea splitting activity preincubated for 2 hrs followed by substrate addition measured after 2 hrs by Berth | 2016 | Journal of medicinal chemistry, 09-08, Volume: 59, Issue:17
| 1,2-Benzisoselenazol-3(2H)-one Derivatives As a New Class of Bacterial Urease Inhibitors. |
| AID274136 | Inhibition of gamma radiation-induced lipid peroxidation in liposomes at 200 uM | 2006 | Bioorganic & medicinal chemistry letters, Oct-15, Volume: 16, Issue:20
| Horseradish peroxidase inhibition and antioxidant activity of ebselen and related organoselenium compounds. |
| AID1632344 | Inhibition of urease in Helicobacter pylori J99 in Brucella broth using urea as substrate after 2 hrs by Berthelot assay | 2016 | Journal of medicinal chemistry, 09-08, Volume: 59, Issue:17
| 1,2-Benzisoselenazol-3(2H)-one Derivatives As a New Class of Bacterial Urease Inhibitors. |
| AID274138 | Effect on gamma irradiation-induced TBARS formation in liposomes at 50 uM | 2006 | Bioorganic & medicinal chemistry letters, Oct-15, Volume: 16, Issue:20
| Horseradish peroxidase inhibition and antioxidant activity of ebselen and related organoselenium compounds. |
| AID1632338 | Reversible inhibition of Sporosarcina pasteurii CCM 2056 urease using urea as substrate assessed as ammonia levels after 120 mins by fast dilution assay | 2016 | Journal of medicinal chemistry, 09-08, Volume: 59, Issue:17
| 1,2-Benzisoselenazol-3(2H)-one Derivatives As a New Class of Bacterial Urease Inhibitors. |
| AID1632342 | Inhibition of recombinant Helicobacter pylori urease expressed in Escherichia coli rosetta DE3 using urea as substrate assessed as transformed cell urea splitting activity after 2 hrs by Berthelot assay | 2016 | Journal of medicinal chemistry, 09-08, Volume: 59, Issue:17
| 1,2-Benzisoselenazol-3(2H)-one Derivatives As a New Class of Bacterial Urease Inhibitors. |
| AID274137 | Inhibition of horseradish peroxidase by spectrophotometric method | 2006 | Bioorganic & medicinal chemistry letters, Oct-15, Volume: 16, Issue:20
| Horseradish peroxidase inhibition and antioxidant activity of ebselen and related organoselenium compounds. |
| AID1632345 | Inhibition of urease in Helicobacter pylori J99 in Brucella broth using urea as substrate preincubated for 2 hrs followed by substrate addition measured after 2 hrs by Berthelot assay | 2016 | Journal of medicinal chemistry, 09-08, Volume: 59, Issue:17
| 1,2-Benzisoselenazol-3(2H)-one Derivatives As a New Class of Bacterial Urease Inhibitors. |
| AID1322290 | Inhibition of pig APN at <2 mM using AMC-labeled substrate preincubated for 30 mins followed by substrate addition by spectrofluorimetric method | 2016 | Bioorganic & medicinal chemistry letters, 11-01, Volume: 26, Issue:21
| Identification of methionine aminopeptidase 2 as a molecular target of the organoselenium drug ebselen and its derivatives/analogues: Synthesis, inhibitory activity and molecular modeling study. |
| AID274141 | Antioxidant activity assessed by singlet oxygen quenching ability at 1mM | 2006 | Bioorganic & medicinal chemistry letters, Oct-15, Volume: 16, Issue:20
| Horseradish peroxidase inhibition and antioxidant activity of ebselen and related organoselenium compounds. |
| AID1632337 | Competitive inhibition of Sporosarcina pasteurii CCM 2056 urease using urea as substrate assessed as ammonia levels after 120 mins by Lineweaver-Burk plot analysis | 2016 | Journal of medicinal chemistry, 09-08, Volume: 59, Issue:17
| 1,2-Benzisoselenazol-3(2H)-one Derivatives As a New Class of Bacterial Urease Inhibitors. |
| AID1322288 | Non-covalent/mixed type inhibition of recombinant human MetAP2 using Met-AMC as substrate preincubated for 30 mins followed by substrate addition by spectrofluorimetric method | 2016 | Bioorganic & medicinal chemistry letters, 11-01, Volume: 26, Issue:21
| Identification of methionine aminopeptidase 2 as a molecular target of the organoselenium drug ebselen and its derivatives/analogues: Synthesis, inhibitory activity and molecular modeling study. |
| AID1632341 | Inhibition of recombinant Helicobacter pylori urease expressed in Escherichia coli rosetta DE3 after 120 mins by Berthelot colorimetric analysis | 2016 | Journal of medicinal chemistry, 09-08, Volume: 59, Issue:17
| 1,2-Benzisoselenazol-3(2H)-one Derivatives As a New Class of Bacterial Urease Inhibitors. |
| AID1322291 | Inhibition of pig LAP at <2 mM using AMC-labeled substrate preincubated for 30 mins followed by substrate addition by spectrofluorimetric method | 2016 | Bioorganic & medicinal chemistry letters, 11-01, Volume: 26, Issue:21
| Identification of methionine aminopeptidase 2 as a molecular target of the organoselenium drug ebselen and its derivatives/analogues: Synthesis, inhibitory activity and molecular modeling study. |
| [information is prepared from bioassay data collected from National Library of Medicine (NLM), extracted Dec-2023] |