Page last updated: 2024-08-01 07:22:59

N3-(2,4-dimethylphenyl)-N1-phenylpyrazole-1,3-dicarboxamide

Description

N3-(2,4-dimethylphenyl)-N1-phenylpyrazole-1,3-dicarboxamide : no description available [CHeBI]

Cross-References

ID SourceID
PubMed CID5219026
CHEMBL ID1372995
CHEBI ID109747

Synonyms (17)

Synonym
3-n-(2,4-dimethylphenyl)-1-n-phenylpyrazole-1,3-dicarboxamide
EU-0074550
MLS000723892
smr000305487
n~3~-(2,4-dimethylphenyl)-n~1~-phenyl-1h-pyrazole-1,3-dicarboxamide
BIM-0045688.P001
CBMICRO_045502 ,
OPREA1_462680
CHEBI:109747
STK996920
AKOS001643597
HMS2662H11
CHEMBL1372995
n3-(2,4-dimethylphenyl)-n1-phenylpyrazole-1,3-dicarboxamide
Q27189029
SR-01000459276-1
sr-01000459276

Drug Classes (1)

ClassDescription
aromatic amideAn amide in which the amide linkage is bonded directly to an aromatic system.

Protein Targets (7)

Potency Measurements

ProteinTaxonomyMeasurementAverage (mM)Bioassay(s)
Chain A, MAJOR APURINIC/APYRIMIDINIC ENDONUCLEASEHomo sapiens (human)Potency56.2341AID2517
LuciferasePhotinus pyralis (common eastern firefly)Potency30.1313AID588342
BRCA1Homo sapiens (human)Potency35.4813AID624202
ATAD5 protein, partialHomo sapiens (human)Potency29.0810AID504467
aldehyde dehydrogenase 1 family, member A1Homo sapiens (human)Potency3.1623AID1030
euchromatic histone-lysine N-methyltransferase 2Homo sapiens (human)Potency28.1838AID504332
nuclear factor erythroid 2-related factor 2 isoform 2Homo sapiens (human)Potency23.1093AID504444

Bioassays (8)

Assay IDTitleYearJournalArticle
AID504812Inverse Agonists of the Thyroid Stimulating Hormone Receptor: HTS campaign2010Endocrinology, Jul, Volume: 151, Issue:7
ISSN: 1945-7170
A small molecule inverse agonist for the human thyroid-stimulating hormone receptor.
AID588501High-throughput multiplex microsphere screening for inhibitors of toxin protease, specifically Lethal Factor Protease, MLPCN compound set2010Current protocols in cytometry, Oct, Volume: Chapter 13ISSN: 1934-9300Microsphere-based flow cytometry protease assays for use in protease activity detection and high-throughput screening.
AID588501High-throughput multiplex microsphere screening for inhibitors of toxin protease, specifically Lethal Factor Protease, MLPCN compound set2006Cytometry. Part A : the journal of the International Society for Analytical Cytology, May, Volume: 69, Issue:5
ISSN: 1552-4922
Microsphere-based protease assays and screening application for lethal factor and factor Xa.
AID588501High-throughput multiplex microsphere screening for inhibitors of toxin protease, specifically Lethal Factor Protease, MLPCN compound set2010Assay and drug development technologies, Feb, Volume: 8, Issue:1
ISSN: 1557-8127
High-throughput multiplex flow cytometry screening for botulinum neurotoxin type a light chain protease inhibitors.
AID651635Viability Counterscreen for Primary qHTS for Inhibitors of ATXN expression2022The Journal of biological chemistry, 08, Volume: 298, Issue:8
ISSN: 1083-351X
AID588497High-throughput multiplex microsphere screening for inhibitors of toxin protease, specifically Botulinum neurotoxin light chain F protease, MLPCN compound set2010Current protocols in cytometry, Oct, Volume: Chapter 13ISSN: 1934-9300Microsphere-based flow cytometry protease assays for use in protease activity detection and high-throughput screening.
AID588497High-throughput multiplex microsphere screening for inhibitors of toxin protease, specifically Botulinum neurotoxin light chain F protease, MLPCN compound set2006Cytometry. Part A : the journal of the International Society for Analytical Cytology, May, Volume: 69, Issue:5
ISSN: 1552-4922
Microsphere-based protease assays and screening application for lethal factor and factor Xa.
AID588497High-throughput multiplex microsphere screening for inhibitors of toxin protease, specifically Botulinum neurotoxin light chain F protease, MLPCN compound set2010Assay and drug development technologies, Feb, Volume: 8, Issue:1
ISSN: 1557-8127
High-throughput multiplex flow cytometry screening for botulinum neurotoxin type a light chain protease inhibitors.
AID588499High-throughput multiplex microsphere screening for inhibitors of toxin protease, specifically Botulinum neurotoxin light chain A protease, MLPCN compound set2010Current protocols in cytometry, Oct, Volume: Chapter 13ISSN: 1934-9300Microsphere-based flow cytometry protease assays for use in protease activity detection and high-throughput screening.
AID588499High-throughput multiplex microsphere screening for inhibitors of toxin protease, specifically Botulinum neurotoxin light chain A protease, MLPCN compound set2006Cytometry. Part A : the journal of the International Society for Analytical Cytology, May, Volume: 69, Issue:5
ISSN: 1552-4922
Microsphere-based protease assays and screening application for lethal factor and factor Xa.
AID588499High-throughput multiplex microsphere screening for inhibitors of toxin protease, specifically Botulinum neurotoxin light chain A protease, MLPCN compound set2010Assay and drug development technologies, Feb, Volume: 8, Issue:1
ISSN: 1557-8127
High-throughput multiplex flow cytometry screening for botulinum neurotoxin type a light chain protease inhibitors.
AID1745845Primary qHTS for Inhibitors of ATXN expression2022The Journal of biological chemistry, 08, Volume: 298, Issue:8
ISSN: 1083-351X
AID504810Antagonists of the Thyroid Stimulating Hormone Receptor: HTS campaign2010Endocrinology, Jul, Volume: 151, Issue:7
ISSN: 1945-7170
A small molecule inverse agonist for the human thyroid-stimulating hormone receptor.
AID1794808Fluorescence-based screening to identify small molecule inhibitors of Plasmodium falciparum apicoplast DNA polymerase (Pf-apPOL).2014Journal of biomolecular screening, Jul, Volume: 19, Issue:6
ISSN: 1552-454X
A High-Throughput Assay to Identify Inhibitors of the Apicoplast DNA Polymerase from Plasmodium falciparum.
AID1794808Fluorescence-based screening to identify small molecule inhibitors of Plasmodium falciparum apicoplast DNA polymerase (Pf-apPOL).2022Journal of enzyme inhibition and medicinal chemistry, Dec, Volume: 37, Issue:1
ISSN: 1475-6374

Research

Studies (7)

TimeframeStudies, This Drug (%)All Drugs %
pre-19900 (0.00)18.7374
1990's0 (0.00)18.2507
2000's1 (14.29)29.6817
2010's4 (57.14)24.3611
2020's2 (28.57)2.80

Study Types

Publication TypeThis drug (%)All Drugs (%)
Trials0 (0.00%)5.53%
Reviews0 (0.00%)6.00%
Case Studies0 (0.00%)4.05%
Observational0 (0.00%)0.25%
Other7 (100.00%)84.16%
SubstanceStudiesClassesRolesFirst YearLast YearAverage AgeRelationship StrengthTrialspre-19901990's2000's2010'spost-2020
pk 11195aromatic amide;
isoquinolines;
monocarboxylic acid amide;
monochlorobenzenes
antineoplastic agent00low000000
acebutololaromatic amide;
ethanolamines;
ether;
monocarboxylic acid amide;
propanolamine;
secondary amino compound
anti-arrhythmia drug;
antihypertensive agent;
beta-adrenergic antagonist;
sympathomimetic agent
00low000000
acetochloraromatic amide;
monocarboxylic acid amide;
organochlorine compound
environmental contaminant;
herbicide;
xenobiotic
00low000000
alachloraromatic amide;
monocarboxylic acid amide;
organochlorine compound
environmental contaminant;
herbicide;
xenobiotic
00low000000
dan 2163aromatic amide;
aromatic amine;
benzamides;
pyrrolidines;
sulfone
environmental contaminant;
second generation antipsychotic;
xenobiotic
00low000000
arotinololaromatic amide;
thiophenes
00low000000
bupivacainearomatic amide;
piperidinecarboxamide;
tertiary amino compound
00low000000
glipizidearomatic amide;
monocarboxylic acid amide;
N-sulfonylurea;
pyrazines
EC 2.7.1.33 (pantothenate kinase) inhibitor;
hypoglycemic agent;
insulin secretagogue
00low000000
granisetronaromatic amide;
indazoles
00low000000
ly 278584aromatic amide;
indazoles
00low000000
metolachloraromatic amide;
benzenes;
ether;
organochlorine compound
00low000000
pyroxamidearomatic amide00low000000
n-phenylformamidearomatic amide;
formamides
00low000000
nithiamideacetamides;
aromatic amide
00low000000
furothiazolearomatic amide00low000000
iocetamic acidaromatic amide00low000000
benomylaromatic amide;
benzimidazole fungicide;
benzimidazoles;
benzimidazolylcarbamate fungicide;
carbamate ester
acaricide;
anthelminthic drug;
antifungal agrochemical;
microtubule-destabilising agent;
tubulin modulator
00low000000
butachloraromatic amide;
organochlorine compound;
tertiary carboxamide
environmental contaminant;
herbicide;
xenobiotic
00low000000
ribavirin1-ribosyltriazole;
aromatic amide;
monocarboxylic acid amide;
primary carboxamide
anticoronaviral agent;
antiinfective agent;
antimetabolite;
antiviral agent;
EC 2.7.7.49 (RNA-directed DNA polymerase) inhibitor
00low000000
iopronic acidaromatic amide00low000000
furalaxylalanine derivative;
aromatic amide;
carboxamide;
furans;
methyl ester
00low000000
closantelaromatic amide;
monocarboxylic acid amide;
monochlorobenzenes;
nitrile;
organoiodine compound;
phenols
00low000000
metalaxylalanine derivative;
aromatic amide;
carboxamide;
ether;
methyl ester
00low000000
metazachloraromatic amide;
organochlorine compound;
pyrazoles
environmental contaminant;
herbicide;
xenobiotic
00low000000
benalaxylalanine derivative;
aromatic amide;
carboxamide;
methyl ester
00low000000
oxadixylanilide fungicide;
aromatic amide;
carbohydrazide;
ether;
oxazolidinone
agrochemical00low000000
ranolazinearomatic amide;
monocarboxylic acid amide;
monomethoxybenzene;
N-alkylpiperazine;
secondary alcohol
00low000000
atorvastatinaromatic amide;
dihydroxy monocarboxylic acid;
monofluorobenzenes;
pyrroles;
statin (synthetic)
environmental contaminant;
xenobiotic
00low000000
1,2,4-triazole-3-carboxamidearomatic amide;
monocarboxylic acid amide;
primary carboxamide;
triazoles
drug metabolite;
human urinary metabolite
00low000000
isonixinaromatic amide00low000000
thifluzamide1,3-thiazoles;
anilide fungicide;
aromatic amide;
aromatic ether;
dibromobenzene;
organofluorine compound
antifungal agrochemical;
EC 1.3.5.1 [succinate dehydrogenase (quinone)] inhibitor
00low000000
foe 5043aromatic amide;
monofluorobenzenes;
thiadiazoles
environmental contaminant;
herbicide;
xenobiotic
00low000000
5-acetylamino-6-amino-3-methyluracilaromatic amide00low000000
dimethenamidaromatic amide;
ether;
organochlorine compound;
thiophenes
00low000000
ribavirin 5'-diphosphate1-ribosyltriazole;
aromatic amide;
monocarboxylic acid amide;
primary carboxamide;
ribose monophosphate
antiviral agent;
drug metabolite;
EC 1.1.1.205 (IMP dehydrogenase) inhibitor;
human blood serum metabolite
00low000000
phenazine-1-carboxamidearomatic amide;
monocarboxylic acid amide;
phenazines
00low000000
ribavirin 5'-triphosphate1-ribosyltriazole;
aromatic amide;
monocarboxylic acid amide;
primary carboxamide;
ribose triphosphate
antiviral agent;
drug metabolite;
EC 2.7.7.48 (RNA-directed RNA polymerase) inhibitor;
eukaryotic initiation factor 4F inhibitor;
human blood serum metabolite
00low000000
ribavirin 5'-diphosphate1-ribosyltriazole;
aromatic amide;
monocarboxylic acid amide;
primary carboxamide;
ribose diphosphate
antiviral agent;
drug metabolite
00low000000
rufinamidearomatic amide;
heteroarene
00low000000
cyclazosinaromatic amide;
aromatic ether;
furans;
monocarboxylic acid amide;
quinazolines;
quinoxaline derivative
adenosine A2A receptor antagonist00low000000
yh 439aromatic amide;
isopropyl ester;
secondary carboxamide
00low000000
allantoxanamidearomatic amide;
heteroarene
00low000000
fr 122047aromatic amide;
thiazoles
00low000000
dabigatran etexilatearomatic amide;
benzimidazoles;
beta-alanine derivative;
carboxamidine;
carboxylic ester;
pyridines
anticoagulant;
EC 3.4.21.5 (thrombin) inhibitor;
prodrug
00low000000
n-(2,3-dichloro-4-hydroxyphenyl)-1-methylcyclohexanecarboxamideanilide fungicide;
aromatic amide;
dichlorobenzene;
monocarboxylic acid amide;
phenols
antifungal agrochemical;
EC 1.14.13.72 (methylsterol monooxygenase) inhibitor;
sterol biosynthesis inhibitor
00low000000
dabigatranaromatic amide;
benzimidazoles;
beta-alanine derivative;
carboxamidine;
pyridines
anticoagulant;
EC 1.10.99.2 [ribosyldihydronicotinamide dehydrogenase (quinone)] inhibitor;
EC 3.4.21.5 (thrombin) inhibitor
00low000000
4-amino-N-(4-methoxyphenyl)-2-(methylthio)-5-thiazolecarboxamidearomatic amide00low000000
N-(2,6-dibromo-4-methylphenyl)-3-(2,6-dichlorophenyl)-5-methyl-4-isoxazolecarboxamidearomatic amide00low000000
N-(2-phenylphenyl)-2-pyrazinecarboxamidearomatic amide00low000000
y 27632aromatic amide00low000000
2-chloro-N-(5-methyl-3-isoxazolyl)acetamidearomatic amide00low000000
N-[3,5-dimethyl-1-(1-oxopropyl)-4-pyrazolyl]propanamidearomatic amide00low000000
N-(3,5-dimethoxyphenyl)-2-thiophenecarboxamidearomatic amide00low000000
N-[1-[(2-bromophenyl)methyl]-2-oxo-3-pyridinyl]butanamidearomatic amide00low000000
4-amino-3-[(cyclohexylamino)-oxomethyl]-5-isothiazolecarboxylic acid ethyl esteraromatic amide;
thiazoles
00low000000
2-[[2-[[4-(2-furanylmethyl)-5-(phenylmethyl)-1,2,4-triazol-3-yl]thio]-1-oxoethyl]amino]-5,6-dihydro-4H-cyclopenta[b]thiophene-3-carboxamidearomatic amide;
thiophenes
00low000000
2-[2-[[2-[(5-cyclopropyl-4-methyl-1,2,4-triazol-3-yl)thio]-1-oxoethyl]amino]-4-thiazolyl]acetic acid ethyl esteraromatic amide00low000000
N-[3-[[2-furanyl(oxo)methyl]amino]phenyl]-1-isoquinolinecarboxamidearomatic amide;
furans
00low000000
N-[2,5-diethoxy-4-[[2-(3-methoxyphenyl)-1-oxoethyl]amino]phenyl]-2-furancarboxamidearomatic amide;
furans
00low000000
5-(4-fluorophenyl)-N-[2-(1-piperidinyl)phenyl]-4-oxazolecarboxamidearomatic amide00low000000
2-[[4-(2-furanylmethyl)-5-methyl-1,2,4-triazol-3-yl]thio]-N-(4-methyl-2-thiazolyl)acetamidearomatic amide00low000000
5-methyl-N-[4-(4-morpholinyl)phenyl]-2-pyrazinecarboxamidearomatic amide00low000000
N-[4-[oxo-(2-pyridinylamino)methyl]phenyl]-2-furancarboxamidearomatic amide;
furans
00low000000
N-[2,5-dimethoxy-4-[[oxo(thiophen-2-yl)methyl]amino]phenyl]-2-furancarboxamidearomatic amide;
furans
00low000000
2-methoxy-N-(5-thiophen-2-yl-1,3,4-thiadiazol-2-yl)acetamidearomatic amide00low000000
N-(5-methyl-1,3,4-thiadiazol-2-yl)-N-phenyl-2-pyrazinecarboxamidearomatic amide00low000000
2-[[(4-methyl-5-thieno[3,2-b]pyrrolyl)-oxomethyl]amino]benzoic acid methyl esteraromatic amide00low000000
N-[2-methoxy-4-[(2-methyl-1-oxopropyl)amino]phenyl]-2-furancarboxamidearomatic amide;
furans
00low000000
4,5-dimethyl-2-[[oxo(thiophen-2-yl)methyl]amino]-3-thiophenecarboxylic acid ethyl esteraromatic amide;
thiophenes
00low000000
N-[2-methyl-5-(3-methyl-[1,2,4]triazolo[3,4-b][1,3,4]thiadiazol-6-yl)phenyl]-3-pyridinecarboxamidearomatic amide00low000000
N-[2-(cyclopentylamino)-2-oxoethyl]-N-(4-methoxyphenyl)-6-(1-piperidinyl)-3-pyridinecarboxamidearomatic amide00low000000
N-[2-methoxy-4-[[2-[(3-methyl-4-oxo-2-quinazolinyl)thio]-1-oxoethyl]amino]phenyl]-2-furancarboxamidearomatic amide;
furans
00low000000
N-propyl-N-(5-pyridin-4-yl-1,3,4-thiadiazol-2-yl)-2-thiophenecarboxamidearomatic amide;
thiophenes
00low000000
N-[2-[2-[2-(4-methoxyanilino)-2-oxoethyl]-5-tetrazolyl]phenyl]-2-furancarboxamidearomatic amide;
furans
00low000000
9-oxo-N-(3-pyridinylmethyl)-3,6-dihydro-2H-[1,4]dioxino[2,3-g]quinoline-8-carboxamidearomatic amide;
quinolines
00low000000
4-amino-N5-[1-(2-furanyl)-2-(3-methylbutylamino)-2-oxoethyl]-N5-(2-methoxyphenyl)isothiazole-3,5-dicarboxamidearomatic amide00low000000
N-[4-(4-acetyl-1-piperazinyl)phenyl]-2,3-dihydro-1,4-benzodioxin-6-carboxamidearomatic amide00low000000
N-[3-chloro-4-(4-morpholinyl)phenyl]-2-furancarboxamidearomatic amide;
furans
00low000000
N-(5-ethyl-1,3,4-thiadiazol-2-yl)-2-[[5-(2-methyl-3-furanyl)-4-(2-methylpropyl)-1,2,4-triazol-3-yl]thio]acetamidearomatic amide00low000000
5-(2-furanyl)-N-(4-methylphenyl)-3-isoxazolecarboxamidearomatic amide00low000000
N-[5-(ethylthio)-1,3,4-thiadiazol-2-yl]-3,3,3-trifluoro-2-methyl-2-(trifluoromethyl)propanamidearomatic amide00low000000
4-amino-N-(2-oxolanylmethyl)-3-prop-2-enyl-2-sulfanylidene-5-thiazolecarboxamidearomatic amide;
thiazoles
00low000000
3-amino-5-methyl-4-[[3-(4-morpholinyl)propylamino]-oxomethyl]-2-thiophenecarboxylic acid ethyl esteraromatic amide;
thiophenes
00low000000
N-[5-(ethylthio)-1,3,4-thiadiazol-2-yl]-2,2-bis(trifluoromethyl)butanamidearomatic amide00low000000
N-[(7-methyl-2-oxo-1H-quinolin-3-yl)methyl]-N-phenyl-2-furancarboxamidearomatic amide;
furans
00low000000
N-[5-[2-(4-morpholinyl)ethyl]-1,3,4-thiadiazol-2-yl]cyclohexanecarboxamidearomatic amide00low000000
N-(5-cyclohexyl-1,3,4-thiadiazol-2-yl)-2-furancarboxamidearomatic amide;
heteroarene
00low000000
5-(3-chlorophenyl)-N-[2-methyl-5-(3-methyl-[1,2,4]triazolo[3,4-b][1,3,4]thiadiazol-6-yl)phenyl]-2-furancarboxamidearomatic amide;
furans
00low000000
4-amino-3-methyl-N-(phenylmethyl)-2-sulfanylidene-5-thiazolecarboxamidearomatic amide;
thiazoles
00low000000
N-[4-(diethylamino)phenyl]-2-furancarboxamidearomatic amide;
furans
00low000000
3-[[2-benzofuranyl(oxo)methyl]amino]benzoic acid ethyl esteraromatic amide;
furans
00low000000
N-(4-fluorophenyl)-2,1,3-benzothiadiazole-5-carboxamidearomatic amide00low000000
N-[5-(2-methylpropyl)-1,3,4-thiadiazol-2-yl]-2-thiophen-2-ylacetamidearomatic amide00low000000
N-(3-pyridinyl)-2,3-dihydrothieno[3,4-b][1,4]dioxin-5-carboxamidearomatic amide;
thiophenes
00low000000
2-[[2,3-dihydro-1,4-benzodioxin-6-yl(oxo)methyl]amino]benzoic acid methyl esteraromatic amide00low000000
5-(2,4-dichlorophenyl)-N-(2-methylphenyl)-2-furancarboxamidearomatic amide;
furans
00low000000
4-[[2-furanyl(oxo)methyl]amino]benzoic acid propan-2-yl esteraromatic amide;
furans;
isopropyl ester;
secondary carboxamide
00low000000
N-(2,5-dimethylphenyl)-2-benzofurancarboxamidearomatic amide;
furans
00low000000
N-(4-methoxyphenyl)-2-benzofurancarboxamidearomatic amide;
furans
00low000000
1-cyclohexyl-3-[[oxo(thiophen-2-yl)methyl]amino]thioureaaromatic amide;
thiophenes
00low000000
N-[4-(3,4-dimethylphenyl)-2-thiazolyl]-2-furancarboxamidearomatic amide;
heteroarene
00low000000
Methyl 3-(isonicotinoylamino)-4-methylbenzoatearomatic amide00low000000
N-[[(5-chloro-2-pyridinyl)amino]-sulfanylidenemethyl]-2-thiophenecarboxamidearomatic amide;
thiophenes
00low000000
N-phenethyl-2-furamidearomatic amide;
heteroarene
00low000000
4-[[oxo(thiophen-2-yl)methyl]amino]benzoic acidaromatic amide00low000000
N-(2,6-dimethoxy-4-pyrimidinyl)-3-phenylpropanamidearomatic amide00low000000
N-(4-ethylphenyl)-4-oxo-3H-phthalazine-1-carboxamidearomatic amide00low000000
N-(2-tert-butyl-5-oxo-4,6-dihydrothieno[3,4-c]pyrazol-3-yl)-2-thiophenecarboxamidearomatic amide;
thiophenes
00low000000
N-[4-[oxo(1-piperidinyl)methyl]phenyl]-2-thiophenecarboxamidearomatic amide00low000000
5-bromo-N-(2,4-dichlorophenyl)-2-furancarboxamidearomatic amide;
furans
00low000000
N-[3-chloro-4-(1-pyrrolidinyl)phenyl]-2-furancarboxamidearomatic amide;
furans
00low000000
2-hydroxy-5-[[(5-methyl-2-furanyl)-oxomethyl]amino]benzoic acidaromatic amide;
furans
00low000000
N-[3-[[2-furanyl(oxo)methyl]amino]phenyl]-5-nitro-2-furancarboxamidearomatic amide;
furans
00low000000
4-cyano-3-methyl-5-(4-methylphenyl)-2-thiophenecarbohydrazidearomatic amide;
thiophenes
00low000000
3-[[(2,5-dimethyl-3-furanyl)-oxomethyl]amino]benzoic acidaromatic amide;
furans
00low000000
4-methyl-N-(3-nitrophenyl)-5-phenyl-3-thiophenecarboxamidearomatic amide00low000000
5-bromo-N-(4-propan-2-ylphenyl)-2-furancarboxamidearomatic amide;
furans
00low000000
N-(cyclopentylideneamino)-4,5,6,7-tetrahydro-1H-indazole-3-carboxamidearomatic amide;
pyrazoles
00low000000
N,4-dimethyl-5-phenyl-2-thiophenecarboxamidearomatic amide;
thiophenes
00low000000
5-[anilino(oxo)methyl]-4-methyl-2-(1-oxopropylamino)-3-thiophenecarboxylic acid methyl esteraromatic amide00low000000
4-methyl-N,5-diphenyl-3-thiophenecarboxamidearomatic amide00low000000
N-(2-pyridinyl)-4,5,6,7-tetrahydro-1-benzothiophene-3-carboxamidearomatic amide;
thiophenes
00low000000
N-(4-bromo-2-fluorophenyl)-2-methyl-3-furancarboxamidearomatic amide;
furans
00low000000
N-(3-chlorophenyl)-1-ethyl-5-methyl-4-pyrazolecarboxamidearomatic amide00low000000
N-[5-(methylthio)-1,3,4-thiadiazol-2-yl]-3-phenylpropanamidearomatic amide00low000000
4-phenyl-N-(2-pyridinyl)butanamidearomatic amide00low000000
2-[[(5-bromo-2-furanyl)-oxomethyl]amino]benzoic acidaromatic amide;
furans
00low000000
N-(4-fluoro-3-nitrophenyl)-3-methyl-2-thiophenecarboxamidearomatic amide00low000000
N-[1-[(4-fluorophenyl)methyl]-3-pyrazolyl]-5-methyl-2-furancarboxamidearomatic amide;
heteroarene
00low000000
N-(3-carbamoyl-5,6-dihydro-4H-cyclopenta[b]thiophen-2-yl)-4-chloro-2-methyl-3-pyrazolecarboxamidearomatic amide;
thiophenes
00low000000
N-(4,5-dihydrothiazol-2-yl)-1-ethyl-3-pyrazolecarboxamidearomatic amide;
pyrazoles
00low000000
N-(2-bromo-4-methylphenyl)-5-ethyl-3-thiophenecarboxamidearomatic amide00low000000
1-[[(1,3-dimethyl-4-pyrazolyl)-oxomethyl]amino]-3-(4-methylphenyl)thioureaaromatic amide;
pyrazoles
00low000000
2,5-dimethyl-4-nitro-N-[4-(1-pyrazolylmethyl)phenyl]-3-pyrazolecarboxamidearomatic amide00low000000
1-(2-methylphenyl)-3-[[(5-methyl-3-thiophenyl)-oxomethyl]amino]thioureaaromatic amide;
thiophenes
00low000000
1-(3-methylphenyl)-3-[[(5-methyl-3-thiophenyl)-oxomethyl]amino]thioureaaromatic amide;
thiophenes
00low000000
1-(3-methylphenyl)-3-[[oxo-(5-propyl-3-thiophenyl)methyl]amino]thioureaaromatic amide;
thiophenes
00low000000
N-(2-chlorophenyl)-5-nitro-2-furancarboxamidearomatic amide;
furans
00low000000
4-chloro-N-[2-fluoro-5-(trifluoromethyl)phenyl]-2-methyl-3-pyrazolecarboxamidearomatic amide00low000000
5-methyl-N-(5-methyl-3-isoxazolyl)-3-isoxazolecarboxamidearomatic amide;
heteroarene
00low000000
N-[4-(5-bromo-2-thiophenyl)-2-thiazolyl]acetamideacetamides;
aromatic amide
00low000000
N-(4-methoxyphenyl)-2-(2-methylpropyl)-4-quinolinecarboxamidearomatic amide00low000000
N-(2-chlorophenyl)-2-[[cyclopropyl(oxo)methyl]amino]-4-methyl-5-thiazolecarboxamidearomatic amide00low000000
5-methyl-N-(3-pyridinyl)-3-isoxazolecarboxamidearomatic amide;
heteroarene
00low000000
2-[[oxo(thiophen-2-yl)methyl]amino]-4,5,6,7-tetrahydro-1-benzothiophene-3-carboxylic acid propan-2-yl esteraromatic amide;
isopropyl ester;
secondary carboxamide;
thiophenes
00low000000
N-(3-hydroxyphenyl)-5-methyl-3-furancarboxamidearomatic amide;
furans
00low000000
5-(4-chlorophenyl)-N-(5-ethyl-1,3,4-thiadiazol-2-yl)-2-furancarboxamidearomatic amide;
heteroarene
00low000000
N-(5-fluoro-2-methylphenyl)-1,3-benzodioxole-5-carboxamidearomatic amide00low000000
N-(2-cyano-1-cyclopentenyl)-1-ethyl-3-pyrazolecarboxamidearomatic amide;
heteroarene
00low000000
N-[4-[[acetamido(sulfanylidene)methyl]amino]phenyl]-2-thiophenecarboxamidearomatic amide00low000000
N-[3-[(1,3-dioxo-5-isoindolyl)oxy]phenyl]-2-furancarboxamidearomatic amide;
furans
00low000000
2-methyl-N-(2,4,6-trimethylphenyl)-3-furancarboxamidearomatic amide;
furans
00low000000
4-[[(2-methyl-1,3-benzothiazol-6-yl)-oxomethyl]amino]benzoic acid methyl esteraromatic amide00low000000
N-(4-ethoxyphenyl)-1,2,5-thiadiazole-3-carboxamidearomatic amide00low000000
4-bromo-1-methyl-N-(2-thiazolyl)-3-pyrazolecarboxamidearomatic amide;
heteroarene
00low000000
N-(3-methoxyphenyl)-4,5,6,7-tetrahydro-1-benzothiophene-3-carboxamidearomatic amide00low000000
3-[[(5-bromo-2-furanyl)-oxomethyl]amino]-2-methylbenzoic acidaromatic amide;
furans
00low000000
5-phenyl-N-(3-pyridinyl)-3-isoxazolecarboxamidearomatic amide;
heteroarene
00low000000
(5-phenyl-3-isoxazolyl)-(1-pyrrolidinyl)methanonearomatic amide;
heteroarene
00low000000
N-(2-pyridinyl)-2-[[5-(3-pyridinyl)-1,3,4-oxadiazol-2-yl]thio]acetamidearomatic amide00low000000
4-[oxo-(pyridin-4-ylamino)methyl]-1H-imidazole-5-carboxylic acid ethyl esteraromatic amide;
heteroarene
00low000000
N-(2-hydroxy-5-methylphenyl)-1,3-dioxo-2-propyl-5-isoindolecarboxamidearomatic amide00low000000
N-[3-[oxo-(3-pyridinylmethylamino)methyl]phenyl]-2-furancarboxamidearomatic amide;
furans
00low000000
N-[(1-ethyl-2-oxo-6-benzo[cd]indolyl)sulfonyl]-N-(4-methoxyphenyl)-3-pyridinecarboxamidearomatic amide00low000000
5-chloro-N-[4-[(3,4-dimethyl-5-isoxazolyl)sulfamoyl]phenyl]-3-methyl-2-benzofurancarboxamidearomatic amide;
furans
00low000000
3-amino-2-[(4-methoxyanilino)-oxomethyl]-4-(4-methoxyphenyl)-6-methyl-5-thieno[2,3-b]pyridinecarboxylic acid ethyl esteraromatic amide00low000000
2-[[4-(2-furanyl)-6-(trifluoromethyl)-2-pyrimidinyl]thio]-N-(5-methyl-3-isoxazolyl)acetamidearomatic amide00low000000
N-(4-methoxyphenyl)-N-thiophen-2-ylsulfonyl-2-furancarboxamidearomatic amide;
furans
00low000000
5-[(2,4-dichlorophenoxy)methyl]-N-(2-fluorophenyl)-2-furancarboxamidearomatic amide;
furans
00low000000
2-[(3-cyano-6,7-dihydro-5H-cyclopenta[b]pyridin-2-yl)thio]-N-(3-cyano-5,6-dihydro-4H-cyclopenta[b]thiophen-2-yl)acetamidearomatic amide00low000000
3-amino-N-(2-fluorophenyl)-6-(phenylmethyl)-4-(trifluoromethyl)-2-thieno[2,3-b]pyridinecarboxamidearomatic amide00low000000
5-(4-bromophenyl)-N-(2-methoxyphenyl)-2-furancarboxamidearomatic amide;
furans
00low000000
5-bromo-N-[4-(4-methyl-1-piperazinyl)phenyl]-2-furancarboxamidearomatic amide;
furans
00low000000
N-[3-chloro-2-(4-morpholinyl)phenyl]-2,3-dihydro-1,4-benzodioxin-6-carboxamidearomatic amide00low000000
N-[3-[oxo-(3-pyridinylmethylamino)methyl]-4,5,6,7-tetrahydro-1-benzothiophen-2-yl]-2-furancarboxamidearomatic amide;
thiophenes
00low000000
N-(4-chlorophenyl)-7,8-dimethoxy-1-oxo-2-benzothiopyran-3-carboxamidearomatic amide00low000000
N-(2-methoxyphenyl)-5-methyl-3-[(2-methylphenyl)methyl]-4-oxo-6-thieno[2,3-d]pyrimidinecarboxamidearomatic amide00low000000
2-[acetyl(2-furanylmethyl)amino]-N-(4-chlorophenyl)-5-methyl-4-thiazolecarboxamidearomatic amide00low000000
N-[2-[2-[2-(4-ethoxyanilino)-2-oxoethyl]-5-tetrazolyl]phenyl]-2-thiophenecarboxamidearomatic amide00low000000
N-(3-methylphenyl)-4-(4-nitrophenyl)-2-phenyl-5-thiazolecarboxamidearomatic amide00low000000
N-(5-chloro-2-pyridinyl)-2-ethyl-3-pyrazolecarboxamidearomatic amide;
heteroarene
00low000000
5-amino-4-[anilino(oxo)methyl]-3-methyl-2-thiophenecarboxylic acid ethyl esteraromatic amide00low000000
5-(3-chlorophenyl)-N-(2-propyl-5-tetrazolyl)-2-furancarboxamidearomatic amide;
heteroarene
00low000000
N-[5-[(4-chlorophenoxy)methyl]-1,3,4-thiadiazol-2-yl]-2-thiophenecarboxamidearomatic amide;
thiophenes
00low000000
N-[5-(1,3-benzothiazol-2-yl)-2-chlorophenyl]-1,3-benzodioxole-5-carboxamidearomatic amide00low000000
N-[4-[[2-furanyl(oxo)methyl]amino]phenyl]-1,3-benzodioxole-5-carboxamidearomatic amide;
furans
00low000000
5-(4-methylphenyl)-N-(3-pyridinylmethyl)-3-isoxazolecarboxamidearomatic amide;
heteroarene
00low000000
N-(4-cyano-2-methyl-3-pyrazolyl)-5-(4-methylphenyl)-3-isoxazolecarboxamidearomatic amide;
heteroarene
00low000000
N-(6-methyl-2-pyridinyl)-2-(phenylmethyl)sulfonylacetamidearomatic amide00low000000
5-nitro-N-[4-(2-oxazolo[4,5-b]pyridinyl)phenyl]-2-furancarboxamidearomatic amide;
furans
00low000000
N-[4-[[2-(4-hydroxyphenyl)-1,3-dioxo-5-isoindolyl]oxy]phenyl]-2-thiophenecarboxamidearomatic amide00low000000
2-furanyl-(4,4,8-trimethyl-1-sulfanylidene-5-dithiolo[3,4-c]quinolinyl)methanonearomatic amide;
heteroarene
00low000000
3-(2-chloro-6-fluorophenyl)-N-(3-fluoro-4-methylphenyl)-5-methyl-4-isoxazolecarboxamidearomatic amide00low000000
N-[4-[[[[oxo(thiophen-2-yl)methyl]amino]-sulfanylidenemethyl]amino]phenyl]-2-furancarboxamidearomatic amide;
furans
00low000000
N-[3-chloro-4-[[2-furanyl(oxo)methyl]amino]phenyl]-2,3-dihydro-1,4-benzodioxin-6-carboxamidearomatic amide;
furans
00low000000
2-methyl-N-(3-methylphenyl)-3-imidazo[1,2-a]pyridinecarboxamidearomatic amide00low000000
N-[2,5-diethoxy-4-[[(2-methylpropylamino)-sulfanylidenemethyl]amino]phenyl]-2-furancarboxamidearomatic amide;
furans
00low000000
N-[2,5-diethoxy-4-[[ethylamino(sulfanylidene)methyl]amino]phenyl]-2-thiophenecarboxamidearomatic amide00low000000
N-[2,5-diethoxy-4-[[(2-furanylmethylamino)-sulfanylidenemethyl]amino]phenyl]-2-furancarboxamidearomatic amide;
furans
00low000000
N-(4-methylphenyl)-4,5,6,7-tetrahydro-1-benzothiophene-2-carboxamidearomatic amide00low000000
N2,N5-bis(3-acetamidophenyl)pyridine-2,5-dicarboxamidearomatic amide00low000000
4-chloro-1-methyl-N-[1-[(4-methylphenyl)methyl]-3-pyrazolyl]-3-pyrazolecarboxamidearomatic amide;
heteroarene
00low000000
N-(5-chloro-2-pyridinyl)-2-(3,5-dimethyl-4-nitro-1-pyrazolyl)acetamidearomatic amide00low000000
N-[4-[methyl(phenyl)sulfamoyl]phenyl]-2-thiophenecarboxamidearomatic amide00low000000
3-[[(2-cyclohexyl-1,3-dioxo-5-isoindolyl)-oxomethyl]amino]benzoic acidaromatic amide00low000000
2-[(3-cyano-6-methyl-2-pyridinyl)thio]-N-(2-thiazolyl)acetamidearomatic amide00low000000
N-(benzenesulfonyl)-N-(4-methoxyphenyl)-3-pyridinecarboxamidearomatic amide00low000000
5-bromo-N-[3-chloro-2-(1-pyrrolidinyl)phenyl]-2-furancarboxamidearomatic amide;
furans
00low000000
N-[(2-fluorophenyl)methyl]-2-thiophenecarboxamidearomatic amide;
thiophenes
00low000000
N-(3-carbamoyl-5-propyl-2-thiophenyl)-2-methyl-3-furancarboxamidearomatic amide;
thiophenes
00low000000
N-(2-carbamoylphenyl)-4-ethyl-5-methyl-3-thiophenecarboxamidearomatic amide00low000000
5-methyl-N-[2-(methylthio)phenyl]-2-furancarboxamidearomatic amide;
furans
00low000000
N-(2-furanylmethyl)-5-methyl-4-phenyl-3-thiophenecarboxamidearomatic amide;
thiophenes
00low000000
5-methyl-N-[5-(trifluoromethyl)-1,3,4-thiadiazol-2-yl]-3-isoxazolecarboxamidearomatic amide;
heteroarene
00low000000
4-ethyl-5-methyl-N-[1-[(3-methylphenyl)methyl]-1,2,4-triazol-3-yl]-3-thiophenecarboxamidearomatic amide;
thiophenes
00low000000
5-bromo-N-[2-(4-chlorophenyl)ethyl]-2-thiophenecarboxamidearomatic amide;
thiophenes
00low000000
5-bromo-N-(5-cyclohexyl-1,3,4-thiadiazol-2-yl)-2-thiophenecarboxamidearomatic amide;
thiophenes
00low000000
2-acetamido-5-propyl-3-thiophenecarboxamideacetamides;
aromatic amide
00low000000
N-(5-tert-butyl-2-methoxyphenyl)-3,5-dimethyl-4-isoxazolecarboxamidearomatic amide00low000000
N-[1-[(4-chlorophenyl)methyl]-4-pyrazolyl]cyclopentanecarboxamidearomatic amide00low000000
3,5-dimethyl-N-[2-(methylthio)phenyl]-4-isoxazolecarboxamidearomatic amide00low000000
N-[2-(4-fluorophenyl)ethyl]-5-methyl-2-thiophenecarboxamidearomatic amide;
thiophenes
00low000000
N-(3-hydroxyphenyl)-3-pyrazolo[1,5-a]pyrimidinecarboxamidearomatic amide00low000000
propanoic acid [4-[[2-furanyl(oxo)methyl]amino]phenyl] esteraromatic amide;
furans
00low000000
N-[4-[4-(1-oxopropyl)-1-piperazinyl]phenyl]-2-furancarboxamidearomatic amide;
furans
00low000000
8-chloro-N-(4-fluorophenyl)-2-(2-pyridinyl)-4-quinolinecarboxamidearomatic amide00low000000
N-[4-[(3,4-dimethyl-5-isoxazolyl)sulfamoyl]phenyl]-6,8-dimethyl-2-(3-pyridinyl)-4-quinolinecarboxamidearomatic amide00low000000
N-[4-[(3,4-dimethyl-5-isoxazolyl)sulfamoyl]phenyl]-6,8-dimethyl-2-(2-pyridinyl)-4-quinolinecarboxamidearomatic amide00low000000
6,8-dimethyl-N-[4-[(5-methyl-3-isoxazolyl)sulfamoyl]phenyl]-2-(2-pyridinyl)-4-quinolinecarboxamidearomatic amide00low000000
N-(4-methyl-2-thiazolyl)-2-[(5-pyridin-4-yl-1,3,4-oxadiazol-2-yl)thio]acetamidearomatic amide00low000000
2-[[5-(3-fluorophenyl)-1,3,4-oxadiazol-2-yl]thio]-N-(1,3,4-thiadiazol-2-yl)acetamidearomatic amide00low000000
N-[2-[4-[(4-chlorophenyl)-oxomethyl]-1-piperazinyl]phenyl]-1,3-benzodioxole-5-carboxamidearomatic amide00low000000
4-[[(4-bromo-2-ethyl-3-pyrazolyl)-oxomethyl]amino]benzoic acid propan-2-yl esteraromatic amide;
isopropyl ester;
secondary carboxamide
00low000000
N-[4-[[[[(4-tert-butylphenyl)-oxomethyl]amino]-sulfanylidenemethyl]amino]-2-methoxyphenyl]-2-thiophenecarboxamidearomatic amide00low000000
3-(2-chlorophenyl)-5-methyl-N-[4-[2-(4-morpholinyl)-2-oxoethoxy]phenyl]-4-isoxazolecarboxamidearomatic amide00low000000
5-[(cyclohexylamino)-oxomethyl]-4-methyl-2-[(1-oxo-2-thiophen-2-ylethyl)amino]-3-thiophenecarboxylic acid ethyl esteraromatic amide;
thiophenes
00low000000
N-[3-[[2-(2-bromo-4,6-dimethylphenoxy)-1-oxoethyl]amino]phenyl]-2-furancarboxamidearomatic amide;
furans
00low000000
5-(2-chlorophenyl)-N-phenyl-2-furancarboxamidearomatic amide;
furans
00low000000
N-[4-(4-morpholinyl)phenyl]-5-(2-nitrophenyl)-2-furancarboxamidearomatic amide;
furans
00low000000
5-[(3-aminoanilino)-oxomethyl]-4-methyl-2-(1-oxobutylamino)-3-thiophenecarboxylic acid methyl esteraromatic amide00low000000
3-amino-8-methyl-N-[4-(4-morpholinyl)phenyl]-2-thieno[2,3-b]quinolinecarboxamidearomatic amide00low000000
N-[5-[(2,2-dimethyl-1-oxopropyl)amino]-2-pyridinyl]-2-furancarboxamidearomatic amide00low000000
5-tert-butyl-N-[2-(cyclopentylamino)-2-oxoethyl]-N-(2,5-dimethylphenyl)-3-methyl-2-furancarboxamidearomatic amide;
furans
00low000000
4-methyl-2-[(1-oxo-2-phenoxyethyl)amino]-N-phenyl-5-thiazolecarboxamidearomatic amide00low000000
N-(4-bromophenyl)-1-[3-chloro-5-(trifluoromethyl)-2-pyridinyl]-2-pyrrolecarboxamidearomatic amide00low000000
[[[3-[(4-methylphenyl)methoxy]-2-thiophenyl]-oxomethyl]amino]thioureaaromatic amide;
thiophenes
00low000000
N,5-bis(4-methoxyphenyl)-2-thiophenecarboxamidearomatic amide00low000000
1-(6-methyl-2-pyridinyl)-N-(3-pyridinyl)-4-imidazolecarboxamidearomatic amide;
heteroarene
00low000000
5-(4-chlorophenyl)-N-[4-(4-methyl-1-piperazinyl)phenyl]-2-furancarboxamidearomatic amide;
furans
00low000000
4-chloro-N-(3,4-dimethoxyphenyl)-1-ethyl-3-pyrazolecarboxamidearomatic amide00low000000
N-(4-fluorophenyl)-3H-benzimidazole-5-carboxamidearomatic amide00low000000
2-[2-[[1-oxo-2-[(5-pyridin-4-yl-1,3,4-oxadiazol-2-yl)thio]ethyl]amino]-4-thiazolyl]acetic acid ethyl esteraromatic amide00low000000
N-[4-[[(1-oxohexylamino)-sulfanylidenemethyl]amino]phenyl]-2-furancarboxamidearomatic amide;
furans
00low000000
5-[diethylamino(oxo)methyl]-4-methyl-2-(1-oxopentylamino)-3-thiophenecarboxylic acid methyl esteraromatic amide;
thiophenes
00low000000
5-bromo-N-[[[oxo(thiophen-2-yl)methyl]hydrazo]-sulfanylidenemethyl]-2-furancarboxamidearomatic amide;
thiophenes
00low000000
N-[5-(ethoxymethyl)-1,3,4-thiadiazol-2-yl]-2-(phenylthio)acetamidearomatic amide00low000000
5-bromo-N-(2-fluorophenyl)-6-oxo-3-pyrancarboxamidearomatic amide00low000000
4-[[3-[(2-methoxyanilino)-oxomethyl]-5,6,7,8-tetrahydro-4H-cyclohepta[b]thiophen-2-yl]amino]-4-oxobutanoic acidaromatic amide00low000000
3-amino-N-(2-fluorophenyl)-6-(2-furanyl)-2-thieno[2,3-b]pyridinecarboxamidearomatic amide00low000000
3-amino-N-(2-fluorophenyl)-6-(3-pyridinyl)-2-thieno[2,3-b]pyridinecarboxamidearomatic amide00low000000
LSM-20401aromatic amide00low000000
N-(4-bromophenyl)-5-tert-butyl-2-methyl-4-nitro-3-pyrazolecarboxamidearomatic amide00low000000
1-[(2-chlorophenyl)methyl]-3-methyl-N-(4-methyl-2-thiazolyl)-5-thieno[2,3-c]pyrazolecarboxamidearomatic amide;
thiophenes
00low000000
2-[[2-furanyl(oxo)methyl]amino]benzoic acid [2-(cyclohexylmethylamino)-2-oxoethyl] esteraromatic amide;
furans
00low000000
2-[2-[[2-[(3-carbamoyl-5,6-dihydro-4H-cyclopenta[b]thiophen-2-yl)amino]-2-oxoethyl]thio]-4-thiazolyl]acetic acid ethyl esteraromatic amide;
thiophenes
00low000000
5-bromo-N-[2-(4-morpholinyl)-5-(trifluoromethyl)phenyl]-3-pyridinecarboxamidearomatic amide00low000000
2-[[2-[5-(4-morpholinylsulfonyl)-2-thiophenyl]-1-oxoethyl]amino]-5-phenyl-3-thiophenecarboxamidearomatic amide;
thiophenes
00low000000
4-[[oxo-(1-phenyl-3-pyridin-4-yl-4-pyrazolyl)methyl]amino]benzoic acid methyl esteraromatic amide00low000000
N-(4-acetylphenyl)-5-[(phenylthio)methyl]-2-furancarboxamidearomatic amide;
furans
00low000000
N-(4-methoxyphenyl)-5-(phenoxymethyl)-2-furancarboxamidearomatic amide;
furans
00low000000
3-cyclohexyl-N-(1,3-dimethyl-2,6-dioxo-4-pyrimidinyl)propanamidearomatic amide00low000000
4-[[(2-methyl-3-furanyl)-oxomethyl]amino]benzoic acid butyl esteraromatic amide;
furans
00low000000
4-[[[5-[(4-chloro-3,5-dimethyl-1-pyrazolyl)methyl]-2-furanyl]-oxomethyl]amino]benzoic acid propan-2-yl esteraromatic amide;
furans;
isopropyl ester
00low000000
2-methyl-N-(2,3,4,5,6-pentafluorophenyl)-3-furancarboxamidearomatic amide;
furans
00low000000
N-[2,2-dimethyl-3-[[oxo(thiophen-2-yl)methyl]amino]propyl]-2-thiophenecarboxamidearomatic amide;
thiophenes
00low000000
5-bromo-N-(2-phenylphenyl)-2-furancarboxamidearomatic amide;
furans
00low000000
N-(2-methoxyphenyl)-5-methyl-3-(1-naphthalenylmethyl)-4-oxo-6-thieno[2,3-d]pyrimidinecarboxamidearomatic amide00low000000
N-[2-[4-[(4-chlorophenyl)-oxomethyl]-1-piperazinyl]phenyl]-2-benzofurancarboxamidearomatic amide;
furans
00low000000
N-[5-(3-methoxyphenyl)-1,3,4-thiadiazol-2-yl]-2-thiophenecarboxamidearomatic amide;
thiophenes
00low000000
1-[[(4-ethyl-5-methyl-3-thiophenyl)-oxomethyl]amino]-3-(2-phenylethyl)thioureaaromatic amide;
thiophenes
00low000000
2,3-bis(2-furanyl)-N-[4-(4-morpholinyl)phenyl]-6-quinoxalinecarboxamidearomatic amide00low000000
6-bromo-2-(3-pyridinyl)-N-[4-(trifluoromethyl)phenyl]-4-quinolinecarboxamidearomatic amide00low000000
4-[[oxo-[2-(2-pyridinyl)-4-quinolinyl]methyl]amino]benzoic acid methyl esteraromatic amide00low000000
N-[3-[[2-(2,6-dimethylphenoxy)-1-oxoethyl]amino]phenyl]-2-furancarboxamidearomatic amide;
furans
00low000000
5-bromo-N-[2-(4-methyl-1-piperazinyl)phenyl]-2-furancarboxamidearomatic amide;
furans
00low000000
N-[2-(1-cyclohexenyl)ethyl]-5-methyl-3-isoxazolecarboxamidearomatic amide;
heteroarene
00low000000
N-[3-[(cyclopropylamino)-oxomethyl]-4,5,6,7,8,9-hexahydrocycloocta[b]thiophen-2-yl]-2-furancarboxamidearomatic amide;
thiophenes
00low000000
2-[[(2-methyl-3-furanyl)-oxomethyl]amino]benzoic acidaromatic amide;
furans
00low000000
N-(3-acetylphenyl)-5,7-dimethyl-2-pyrazolo[1,5-a]pyrimidinecarboxamidearomatic amide00low000000
[3,5-bis[(phenylmethyl)amino]-1,2,4-triazol-1-yl]-thiophen-2-ylmethanonearomatic amide;
thiophenes
00low000000
2-[[[5-(3-chlorophenyl)-2-furanyl]-oxomethyl]amino]benzoic acid methyl esteraromatic amide;
furans
00low000000
N-[4-(4-morpholinyl)phenyl]-2-pyridin-4-yl-4-quinolinecarboxamidearomatic amide00low000000
5-chloro-N-(3,4-dimethylphenyl)-2,1-benzothiazole-3-carboxamidearomatic amide00low000000
[[2-[[4-(4-bromophenyl)-2-thiazolyl]amino]-2-oxoethyl]thio]methanethioic acid O-ethyl esteraromatic amide00low000000
N-(2-sulfanylidene-3H-1,3,4-thiadiazol-5-yl)-2-furancarboxamidearomatic amide;
heteroarene
00low000000
5-methyl-N-(4-propan-2-ylphenyl)-2-pyrazinecarboxamidearomatic amide00low000000
2-pyridin-4-yl-N-[4-(2-thiazolylsulfamoyl)phenyl]-4-quinolinecarboxamidearomatic amide00low000000
N-[4-(1-piperidinyl)phenyl]-2-quinolinecarboxamidearomatic amide00low000000
2,5-dimethyl-1-(3-methylphenyl)-N-(4-methylphenyl)-3-pyrrolecarboxamidearomatic amide00low000000
N-[4-(difluoromethylthio)phenyl]-5-[(2-hydroxy-5-methoxyphenyl)-oxomethyl]-2-imino-3-pyrancarboxamidearomatic amide00low000000
N-(2-tert-butylphenyl)-2,2-dioxo-3,4-dihydro-[1,2,4]thiadiazino[3,4-b][1,3]benzothiazole-8-carboxamidearomatic amide00low000000
N-(4-tert-butyl-2-thiazolyl)-5-methyl-2-thiophenecarboxamidearomatic amide;
thiophenes
00low000000
2-[[2-furanyl(oxo)methyl]amino]-4,5-dimethoxybenzoic acid [2-[(3,5-dichloro-2-pyridinyl)amino]-2-oxoethyl] esteraromatic amide;
furans
00low000000
4-acetyl-N-[4-(4-chlorophenyl)-2-thiazolyl]-3,5-dimethyl-1H-pyrrole-2-carboxamidearomatic amide;
heteroarene
00low000000
N-(6-methoxy-3-pyridinyl)-3-methyl-2-thiophenecarboxamidearomatic amide;
thiophenes
00low000000
N-(4-chloro-2-fluorophenyl)-3-(methoxymethyl)-2-benzofurancarboxamidearomatic amide;
furans
00low000000
7-methyl-N-[4-(4-morpholinyl)phenyl]-[1,2,4]triazolo[1,5-a]pyrimidine-2-carboxamidearomatic amide00low000000
N-[4-(2-pyridinyl)-2-thiazolyl]cyclopentanecarboxamidearomatic amide00low000000
5-[2-[[2-[[2-furanyl(oxo)methyl]amino]phenyl]-oxomethoxy]-1-oxoethyl]-2,4-dimethyl-1H-pyrrole-3-carboxylic acid ethyl esteraromatic amide;
furans
00low000000
N-[2-[(1,3-benzodioxol-5-ylmethylamino)-oxomethyl]phenyl]-2-ethoxy-3-pyridinecarboxamidearomatic amide00low000000
N-(5-methyl-2-thiazolyl)cyclopentanecarboxamidearomatic amide00low000000
2-[[2-[[5-(4-ethylanilino)-1,3,4-thiadiazol-2-yl]thio]-1-oxoethyl]amino]-3-thiophenecarboxamidearomatic amide;
thiophenes
00low000000
N-(4-chlorophenyl)-N-ethyl-6-(propan-2-ylamino)-4-(trifluoromethyl)-3-pyridinecarboxamidearomatic amide00low000000
N-(4-chlorophenyl)-2,5-dimethyl-1-(thiophen-2-ylmethyl)-3-pyrrolecarboxamidearomatic amide00low000000
N-(3,5-dimethylphenyl)-2,5-dimethyl-1-(thiophen-2-ylmethyl)-3-pyrrolecarboxamidearomatic amide00low000000
N-(4-chlorophenyl)-5-methyl-2-[(4-methylphenyl)methyl]-3-pyrazolecarboxamidearomatic amide00low000000
N-(6-methoxy-3-pyridinyl)-2-thiophenecarboxamidearomatic amide;
thiophenes
00low000000
3-[5-[anilino(oxo)methyl]-2-furanyl]-2-thiophenecarboxylic acid methyl esteraromatic amide;
furans
00low000000
5-(4-morpholinylsulfonyl)-N-[4-(trifluoromethoxy)phenyl]-2-furancarboxamidearomatic amide;
furans
00low000000
5-tert-butyl-N-(4-fluorophenyl)-2-[(4-fluorophenyl)methyl]-3-pyrazolecarboxamidearomatic amide00low000000
N-(4-oxo-2-thieno[3,2-d][1,3]thiazinyl)-2-furancarboxamidearomatic amide;
heteroarene
00low000000
5-[[[5-(2-chlorophenyl)-2-(trifluoromethyl)-3-furanyl]-oxomethyl]amino]-2-(4-morpholinyl)benzoic acid methyl esteraromatic amide;
furans
00low000000
2-(4-morpholinyl)-5-[[oxo-[2-(trifluoromethyl)-5-[4-(trifluoromethyl)phenyl]-3-furanyl]methyl]amino]benzoic acid methyl esteraromatic amide;
furans
00low000000
5-[[[5-(4-chlorophenyl)-2-(trifluoromethyl)-3-furanyl]-oxomethyl]amino]-2-(4-morpholinyl)benzoic acid methyl esteraromatic amide;
furans
00low000000
2-[[(5-tert-butyl-2-methyl-3-furanyl)-oxomethyl]amino]-4,5-dimethoxybenzoic acid methyl esteraromatic amide;
furans
00low000000
N-[3-(aminosulfonyl)phenyl]-2-phenoxynicotinamidearomatic amide00low000000
5-tert-butyl-N-[5-(dimethylsulfamoyl)-2-methylphenyl]-2-(phenylmethyl)-3-pyrazolecarboxamidearomatic amide00low000000
N'-[4-(3-methoxyphenyl)-2-thiazolyl]-2-thiophenecarbohydrazidearomatic amide;
thiophenes
00low000000
4-(4-chlorophenyl)sulfonyl-N-(2,4-difluorophenyl)-3-methyl-2-thiophenecarboxamidearomatic amide00low000000
3-chloro-4-propan-2-ylsulfonyl-2-thiophenecarbohydrazidearomatic amide;
thiophenes
00low000000
N-(2-chlorophenyl)-5-(2-pyridinyl)-2-thiophenecarboxamidearomatic amide00low000000
4-hydroxy-3-(methylthio)-4,5,6,7-tetrahydro-2-benzothiophene-1-carbohydrazidearomatic amide;
thiophenes
00low000000
N-phenyl-2-benzo[g][1]benzothiolecarboxamide1-benzothiophenes;
aromatic amide
00low000000
N-(4-methyl-2-nitrophenyl)-2-furancarboxamidearomatic amide;
furans
00low000000
N-(5-nitro-2-pyridinyl)cyclopropanecarboxamidearomatic amide00low000000
3-ethyl-N-(2H-tetrazol-5-yl)-1-adamantanecarboxamidearomatic amide00low000000
2-[[oxo(thiophen-2-yl)methyl]amino]-6-propyl-4,5,6,7-tetrahydro-1-benzothiophene-3-carboxamidearomatic amide;
thiophenes
00low000000
N-(2-hydroxy-5-methylphenyl)-2-furancarboxamidearomatic amide;
furans
00low000000
3-[[[1,3-dioxo-2-(2-oxolanylmethyl)-5-isoindolyl]-oxomethyl]amino]benzoic acidaromatic amide00low000000
alanyl-alanyl-alanyl-alanine, (d-ala-l-ala-l-ala-l-ala)-isomeraromatic amide;
furans
00low000000
N-[5-[(4-methylphenyl)methyl]-2-thiazolyl]-2-oxolanecarboxamidearomatic amide00low000000
[3-methyl-4-[oxo(thiophen-2-yl)methyl]-1-piperazinyl]-thiophen-2-ylmethanonearomatic amide;
thiophenes
00low000000
N-[(2-ethyl-1-piperidinyl)-sulfanylidenemethyl]-2-thiophenecarboxamidearomatic amide;
thiophenes
00low000000
N-(3,3,5-trimethylcyclohexyl)-1H-1,2,4-triazole-5-carboxamidearomatic amide;
heteroarene
00low000000
6-[[[5-(ethylthio)-1,3,4-thiadiazol-2-yl]amino]-oxomethyl]-1-cyclohex-3-enecarboxylic acidaromatic amide00low000000
4-amino-3-(4-ethoxyphenyl)-N-(2-oxolanylmethyl)-2-sulfanylidene-5-thiazolecarboxamidearomatic amide;
thiazoles
00low000000
N-[4-[[[4-(4-methoxyphenyl)-4-oxanyl]methylamino]-oxomethyl]phenyl]-2-furancarboxamidearomatic amide;
furans
00low000000
N4-(4-fluorophenyl)-N5-(2-nitrophenyl)-1H-imidazole-4,5-dicarboxamidearomatic amide00low000000
N-[5-(2-oxolanyl)-1,3,4-thiadiazol-2-yl]-2-thiophenecarboxamidearomatic amide;
thiophenes
00low000000
N-(3-carbamoyl-5-propyl-2-thiophenyl)-2-oxolanecarboxamidearomatic amide;
thiophenes
00low000000
N-(3-cyano-6-methyl-4,5,6,7-tetrahydro-1-benzothiophen-2-yl)-5-methyl-3-isoxazolecarboxamidearomatic amide;
heteroarene
00low000000
5-bromo-N-[1-(2,5-dimethylphenyl)ethyl]-2-furancarboxamidearomatic amide;
heteroarene
00low000000
2-[(4-methylphenyl)thio]-N-(1H-1,2,4-triazol-5-yl)propanamidearomatic amide00low000000
N-[4-(4-acetyl-1-piperazinyl)-3-chlorophenyl]-2-furancarboxamidearomatic amide;
furans
00low000000
N-(3-cyano-2-thiophenyl)-2-[(1-methyl-2-imidazolyl)thio]acetamidearomatic amide00low000000
5-[[[2-[[2-furanyl(oxo)methyl]amino]phenyl]-oxomethoxy]methyl]-3-methyl-1H-pyrrole-2,4-dicarboxylic acid diethyl esteraromatic amide;
furans
00low000000
N-(4,5,6,7-tetrahydro-1,3-benzothiazol-2-yl)-4-thiophen-2-ylbutanamidearomatic amide00low000000
2-[[5-[1-(dimethylamino)ethyl]-4-(phenylmethyl)-1,2,4-triazol-3-yl]thio]-N-(5-methyl-3-isoxazolyl)acetamidearomatic amide00low000000
2,2,3,3-tetrafluoro-N-(1H-1,2,4-triazol-5-yl)propanamidearomatic amide00low000000
4-[[3-[(4-methylanilino)-oxomethyl]-5,6,7,8-tetrahydro-4H-cyclohepta[b]thiophen-2-yl]amino]-4-oxobutanoic acidaromatic amide00low000000
N-(2-methoxyphenyl)-6-methyl-4,5,6,7-tetrahydro-1-benzothiophene-3-carboxamidearomatic amide00low000000
6-methyl-N-(5-methyl-1,3,4-thiadiazol-2-yl)-4,5,6,7-tetrahydro-1-benzothiophene-3-carboxamidearomatic amide;
thiophenes
00low000000
N-[3-chloro-4-(4-methyl-1-piperazinyl)phenyl]-2,3-dihydro-1,4-benzodioxin-6-carboxamidearomatic amide00low000000
N-[2-(3-oxo-4H-quinoxalin-2-yl)phenyl]-2-thiophenecarboxamidearomatic amide00low000000
4-amino-N5-(4-butoxyphenyl)-N5-[2-(cyclohexylamino)-2-oxoethyl]isothiazole-3,5-dicarboxamidearomatic amide00low000000
N-(4-Butan-2-ylphenyl)-N-[2-(cyclopentylamino)-2-oxo-1-pyridin-3-ylethyl]furan-2-carboxamidearomatic amide;
furans
anticoronaviral agent00low000000
N-[2-(Cyclopentylamino)-2-oxo-1-pyridin-3-ylethyl]-N-(4-propan-2-ylphenyl)furan-2-carboxamidearomatic amide;
furans
anticoronaviral agent00low000000
4-amino-3-[(cyclohexylamino)-oxomethyl]-5-isothiazolecarboxylic acid [1-(cyclohexylamino)-1-oxopropan-2-yl] esteraromatic amide;
thiazoles
00low000000
4-[[(4-methyl-5-thieno[3,2-b]pyrrolyl)-oxomethyl]amino]benzoic acid methyl esteraromatic amide00low000000
1-[(4-fluorophenyl)methyl]-N-[4-(4-methyl-1-piperazinyl)phenyl]-2-oxo-3H-benzimidazole-5-carboxamidearomatic amide00low000000
5-(2-furanyl)-N-(3-pyridinylmethyl)-3-isoxazolecarboxamidearomatic amide;
heteroarene
00low000000
5-bromo-N-[6-[[(5-bromo-2-furanyl)-oxomethyl]amino]-2-pyridinyl]-2-furancarboxamidearomatic amide;
heteroarene
00low000000
N-(2,4-dimethoxyphenyl)-3-[[2-(2-methoxyphenoxy)-1-oxoethyl]amino]-2-benzofurancarboxamidearomatic amide;
furans
00low000000
N-(2,4-dimethoxyphenyl)-3-[[2-furanyl(oxo)methyl]amino]-2-benzofurancarboxamidearomatic amide;
furans
00low000000
N-(2-furanylmethyl)-5-(4-morpholinyl)-4-phenyl-2-thiophenecarboxamidearomatic amide;
thiophenes
00low000000
5-(4-bromophenyl)-N,N-diethyl-3-isoxazolecarboxamidearomatic amide;
heteroarene
00low000000
N-[4-[5-[(2-methylphenoxy)methyl]-1,2,4-oxadiazol-3-yl]phenyl]-2-furancarboxamidearomatic amide;
furans
00low000000
5-[(4-fluorophenyl)methylsulfonylmethyl]-N-(2-oxolanylmethyl)-2-furancarboxamidearomatic amide;
heteroarene
00low000000
N-(5-chloro-2-methoxyphenyl)-2,4-dimethyl-5-oxazolecarboxamidearomatic amide00low000000
3-[[oxo(2-quinoxalinyl)methyl]amino]benzoic acid ethyl esteraromatic amide00low000000
N-(3-chlorophenyl)-5-(1,4-dioxa-8-azaspiro[4.5]decan-8-ylsulfonyl)-3-methyl-2-benzofurancarboxamidearomatic amide;
furans
00low000000
3-[[2-furanyl(oxo)methyl]amino]-N-(4-methoxyphenyl)-2-benzofurancarboxamidearomatic amide;
furans
00low000000
N-(1,1-dioxo-2,3-dihydrothiophen-3-yl)-N-(2-ethylphenyl)-2-thiophenecarboxamidearomatic amide00low000000
1-[oxo-[4-oxo-6-[(4-propan-2-ylphenyl)sulfamoyl]-1H-quinolin-3-yl]methyl]-4-piperidinecarboxamidearomatic amide;
quinolines
00low000000
3-methyl-N,6-diphenyl-2-imidazo[2,1-b]thiazolecarboxamidearomatic amide00low000000
N-(3,4-dimethoxyphenyl)-7-methoxy-4,5-dihydrobenzo[g][1,2]benzoxazole-3-carboxamidearomatic amide00low000000
6-[(2-ethylphenyl)sulfamoyl]-N-(2-furanylmethyl)-4-oxo-1H-quinoline-3-carboxamidearomatic amide;
quinolines
00low000000
N-ethyl-3-[4-morpholinyl(oxo)methyl]-4-oxo-N-phenyl-1H-quinoline-6-sulfonamidearomatic amide;
quinolines
00low000000
6-[(2-ethylphenyl)sulfamoyl]-4-oxo-N-(2-oxolanylmethyl)-1H-quinoline-3-carboxamidearomatic amide;
quinolines
00low000000
6-(1-azepanylsulfonyl)-1-ethyl-N-(2-furanylmethyl)-4-oxo-3-quinolinecarboxamidearomatic amide;
quinolines
00low000000
3-(2-chlorophenyl)-5-methyl-N-[3-(3-methyl-2-imidazo[1,2-a]pyrimidinyl)phenyl]-4-isoxazolecarboxamidearomatic amide00low000000
N-(4-ethylphenyl)-5-(2-furanyl)-3-isoxazolecarboxamidearomatic amide00low000000
N-(2-chlorophenyl)-5-(1,4-dioxa-8-azaspiro[4.5]decan-8-ylsulfonyl)-3-methyl-2-benzofurancarboxamidearomatic amide;
furans
00low000000
N4,N5-bis(2-ethoxyphenyl)-1H-imidazole-4,5-dicarboxamidearomatic amide00low000000
N-(4-acetylphenyl)-5,6,7,8-tetrahydro-4H-cyclohepta[d]isoxazole-3-carboxamidearomatic amide00low000000
N-[1-[(4-fluorophenyl)methyl]-3,5-dimethyl-4-pyrazolyl]-5-(2-furanyl)-3-isoxazolecarboxamidearomatic amide;
heteroarene
00low000000
5-(4-chlorophenyl)-N-(2-furanylmethyl)-3-isoxazolecarboxamidearomatic amide;
heteroarene
00low000000
N-(2,3-dimethylphenyl)-3-methyl-5-(4-morpholinylsulfonyl)-2-benzofurancarboxamidearomatic amide;
furans
00low000000
N-(3,4-dimethylphenyl)-5-(2-furanyl)-3-isoxazolecarboxamidearomatic amide00low000000
5-(4-bromophenyl)-N-propan-2-yl-3-isoxazolecarboxamidearomatic amide;
heteroarene
00low000000
N-(3-pyridinyl)-5,6,7,8-tetrahydro-4H-cyclohepta[d]isoxazole-3-carboxamidearomatic amide;
heteroarene
00low000000
N-[1-(2,3-dihydro-1,4-benzodioxin-6-yl)ethyl]-1-methyl-4-oxo-6-(1-pyrrolidinylsulfonyl)-3-quinolinecarboxamidearomatic amide;
quinolines
00low000000
N-butan-2-yl-6-[(4-ethoxyphenyl)sulfamoyl]-4-oxo-1H-quinoline-3-carboxamidearomatic amide;
quinolines
00low000000
1-methyl-6-[(4-methyl-1-piperidinyl)sulfonyl]-3-[oxo(1-piperidinyl)methyl]-4-quinolinonearomatic amide;
quinolines
00low000000
N-(3,4-dimethylphenyl)-3-methyl-5-(4-morpholinylsulfonyl)-2-benzofurancarboxamidearomatic amide;
furans
00low000000
1-methyl-N-(2-methylcyclohexyl)-4-oxo-6-(1-pyrrolidinylsulfonyl)-3-quinolinecarboxamidearomatic amide;
quinolines
00low000000
N-cyclohexyl-5,6,7,8-tetrahydro-4H-cyclohepta[d]isoxazole-3-carboxamidearomatic amide;
heteroarene
00low000000
N-[5-(dimethylsulfamoyl)-2-methylphenyl]-2-quinolinecarboxamidearomatic amide00low000000
N-[5-(diethylsulfamoyl)-2-(4-morpholinyl)phenyl]-2-oxo-1H-quinoline-4-carboxamidearomatic amide00low000000
3-(2-benzofuranyl)-N-(4-nitrophenyl)-1-phenyl-4-pyrazolecarboxamidearomatic amide00low000000
LSM-20806aromatic amide00low000000
N-[(4-methoxyphenyl)methyl]-2-(phenylmethyl)-4-thiazolecarboxamidearomatic amide;
thiazoles
00low000000
5-bromo-N-[3-[methyl(phenyl)sulfamoyl]phenyl]-3-pyridinecarboxamidearomatic amide00low000000
N-(3-carbamoyl-4,5,6,7-tetrahydro-1-benzothiophen-2-yl)-2-methyl-3-pyrazolecarboxamidearomatic amide;
thiophenes
00low000000
1-butyl-3-[[(4,5-dimethyl-3-thiophenyl)-oxomethyl]amino]thioureaaromatic amide;
thiophenes
00low000000
4-[[3-[anilino(oxo)methyl]-5,6,7,8-tetrahydro-4H-cyclohepta[b]thiophen-2-yl]amino]-4-oxobutanoic acidaromatic amide00low000000
6-bromo-1-(dibromomethyl)-5,5-dimethyl-N-(6-methyl-2-pyridinyl)-4-bicyclo[2.1.1]hexanecarboxamidearomatic amide00low000000
N1',N6'-bis[(5-methyl-1H-pyrazol-3-yl)-oxomethyl]hexanedihydrazidearomatic amide;
pyrazoles
00low000000
1-amino-N-methyl-5-(4-morpholinyl)-N-phenyl-6,7,8,9-tetrahydrothieno[2,3-c]isoquinoline-2-carboxamidearomatic amide00low000000
N-(2-fluorophenyl)-6-(1,2,4-triazol-1-yl)-3-pyridinecarboxamidearomatic amide00low000000
N-methyl-5-phenyl-2-thiophenecarboxamidearomatic amide;
thiophenes
00low000000
N-(4-fluorophenyl)-5-methyl-1H-indole-2-carboxamidearomatic amide00low000000
N-[3-(1,3-dioxo-2-benzo[de]isoquinolinyl)propyl]-N-(2-methoxy-4-methylphenyl)-2-thiophenecarboxamidearomatic amide00low000000
N-[3-(dimethylsulfamoyl)-4-methylphenyl]-2-quinolinecarboxamidearomatic amide00low000000
N-[3-[(2-methoxyphenyl)sulfamoyl]phenyl]-2-quinolinecarboxamidearomatic amide00low000000
N-(2,4-dimethylphenyl)-3-methyl-5-(4-morpholinylsulfonyl)-2-benzofurancarboxamidearomatic amide;
furans
00low000000
N-[3-(1,3-benzothiazol-2-yl)phenyl]-4-oxo-1-benzopyran-2-carboxamidearomatic amide00low000000
3-(4-methylphenyl)-N-[3-(4-morpholinylsulfonyl)phenyl]-1-phenyl-4-pyrazolecarboxamidearomatic amide00low000000
4-amino-3-(3,4-dimethylphenyl)-N-(2-fluorophenyl)-2-sulfanylidene-5-thiazolecarboxamidearomatic amide00low000000
5-oxo-N-[3-(trifluoromethyl)phenyl]-2,3-dihydrothiazolo[3,2-a]pyrimidine-6-carboxamidearomatic amide00low000000
N-[5-(2-chlorophenyl)-1,3,4-thiadiazol-2-yl]-2-[(4-methyl-1,2,4-triazol-3-yl)thio]butanamidearomatic amide00low000000
LSM-19765aromatic amide00low000000
N-[4-methyl-3-(1-piperidinylsulfonyl)phenyl]-4-oxo-1-benzopyran-2-carboxamidearomatic amide00low000000
N-(2,5-dimethoxyphenyl)-4-oxo-3-(2-phenylethyl)-2-sulfanylidene-1H-quinazoline-7-carboxamidearomatic amide00low000000
N-[3-(dimethylsulfamoyl)-4-methylphenyl]-5-methyl-2-pyrazinecarboxamidearomatic amide00low000000
N-(4-methylphenyl)-6-(1-pyrazolyl)-3-pyridinecarboxamidearomatic amide00low000000
N-[4-[(cyclohexylamino)-oxomethyl]phenyl]-3-pyridinecarboxamidearomatic amide00low000000
N-[3-[(2,4-dimethylphenyl)sulfamoyl]-4-methylphenyl]-3-oxo-4H-1,4-benzothiazine-6-carboxamidearomatic amide00low000000
N-(3-methoxyphenyl)-1,3-dioxo-2-(2-oxolanylmethyl)-5-isoindolecarboxamidearomatic amide00low000000
ver-49009aromatic amide;
monochlorobenzenes;
monomethoxybenzene;
pyrazoles;
resorcinols
Hsp90 inhibitor00low000000
N2,N6-bis[4-(dimethylamino)phenyl]pyridine-2,6-dicarboxamidearomatic amide00low000000
2,5-dichloro-N-[5-(4-fluorophenyl)-1,3,4-oxadiazol-2-yl]-3-thiophenecarboxamidearomatic amide;
thiophenes
00low000000
N-[4-[5-(3,4-dimethoxyphenyl)-1,2,4-oxadiazol-3-yl]phenyl]-4-pyridinecarboxamidearomatic amide00low000000
5-(2-chlorophenyl)-N-(4-methoxyphenyl)-2-furancarboxamidearomatic amide;
furans
00low000000
N-[3-(1-azepanylsulfonyl)phenyl]-4-oxo-1-benzopyran-2-carboxamidearomatic amide00low000000
N-[4-[(3,4-dimethyl-5-isoxazolyl)sulfamoyl]phenyl]-3-methyl-5-oxo-6-thiazolo[3,2-a]pyrimidinecarboxamidearomatic amide00low000000
N-(2,4-difluorophenyl)-6-(propylthio)-3-pyridinecarboxamidearomatic amide00low000000
N,N,4-trimethyl-2-[[(5-methyl-2-furanyl)-oxomethyl]amino]-5-thiazolecarboxamidearomatic amide;
thiazoles
00low000000
5-bromo-N-(5-pyridin-4-yl-1,3,4-oxadiazol-2-yl)-2-thiophenecarboxamidearomatic amide;
thiophenes
00low000000
N-[5-(diethylsulfamoyl)-2-(4-morpholinyl)phenyl]-2,3-dihydro-1H-cyclopenta[b]quinoline-9-carboxamidearomatic amide00low000000
N-(2-chloro-3-pyridinyl)-2-[[5-(3-methylanilino)-1,3,4-thiadiazol-2-yl]thio]acetamidearomatic amide00low000000
N-[5-(4-morpholinylsulfonyl)-2-(1-pyrrolidinyl)phenyl]-2-oxo-1H-quinoline-4-carboxamidearomatic amide00low000000
6-chloro-N-[3-[(2-chlorophenyl)sulfamoyl]phenyl]-3-pyridinecarboxamidearomatic amide00low000000
N-[4-methoxy-3-(4-morpholinylsulfonyl)phenyl]-5-methyl-4,5,6,7-tetrahydro-1-benzothiophene-2-carboxamidearomatic amide00low000000
N-[5-(diethylsulfamoyl)-2-methoxyphenyl]-5-methyl-3-isoxazolecarboxamidearomatic amide00low000000
N-(4-Nitro-1,2,5-oxadiazol-3-yl)-2-pyridin-2-ylsulfanylacetamidearomatic amideanticoronaviral agent00low000000
N-[3-(1,3-dioxo-2-benzo[de]isoquinolinyl)propyl]-N-(4-methoxyphenyl)-2-thiophenecarboxamidearomatic amide00low000000
N-(3-carbamoyl-6-methyl-4,5,6,7-tetrahydro-1-benzothiophen-2-yl)-3-(2-chlorophenyl)-5-methyl-4-isoxazolecarboxamidearomatic amide;
thiophenes
00low000000
[3-(2-hydroxyphenyl)-5-(4-methoxyphenyl)-3,4-dihydropyrazol-2-yl]-thiophen-2-ylmethanonearomatic amide;
thiophenes
00low000000
2-(4,5-dihydrothiazol-2-ylthio)-N-[5-(ethylthio)-1,3,4-thiadiazol-2-yl]acetamidearomatic amide00low000000
1-butyl-3-[[oxo-(5-propan-2-yl-3-thiophenyl)methyl]amino]thioureaaromatic amide;
thiophenes
00low000000
5-bromo-N-[4-[5-(2-methylphenyl)-1,2,4-oxadiazol-3-yl]phenyl]-2-furancarboxamidearomatic amide;
furans
00low000000
N-[1-[(4-fluorophenyl)methyl]-4-pyrazolyl]-5-(2-furanyl)-3-isoxazolecarboxamidearomatic amide;
heteroarene
00low000000
N-ethyl-3-(1-pyrrolyl)-2-thiophenecarboxamidearomatic amide;
thiophenes
00low000000
N-(4-methoxyphenyl)-5-[2-(trifluoromethyl)phenyl]-2-furancarboxamidearomatic amide;
furans
00low000000
N-[5-(diethylsulfamoyl)-2-(4-morpholinyl)phenyl]-2-oxo-1-benzopyran-3-carboxamidearomatic amide00low000000
N-(3-nitrophenyl)-1,3-benzodioxole-5-carboxamidearomatic amide00low000000
granisetronaromatic amide;
indazoles
00low000000
N-(3-chlorophenyl)-1H-imidazole-5-carboxamidearomatic amide00low000000
N-[3-(3-chlorophenyl)-5-isoxazolyl]-2-(4,5,6,7-tetrahydroindazol-2-yl)acetamidearomatic amide00low000000
N-(3-cyano-5,6-dihydro-4H-cyclopenta[b]thiophen-2-yl)-5-cyclopropyl-3-isoxazolecarboxamidearomatic amide;
heteroarene
00low000000
N-cyclohexyl-5-propyl-3-isoxazolecarboxamidearomatic amide;
heteroarene
00low000000
N-(3-cyano-4,5,6,7-tetrahydro-1-benzothiophen-2-yl)-5-(2-methylpropyl)-3-isoxazolecarboxamidearomatic amide;
heteroarene
00low000000
2-[[oxo-(5-propyl-3-isoxazolyl)methyl]amino]benzoic acid methyl esteraromatic amide00low000000
N-(4-ethylphenyl)-2-(2-furanylmethyl)-1,3-dioxo-5-isoindolecarboxamidearomatic amide00low000000
N-(5-bromo-2-hydroxyphenyl)-5-propyl-3-isoxazolecarboxamidearomatic amide00low000000
N-(2-ethylphenyl)-5-(3-hydroxyphenyl)-3-isoxazolecarboxamidearomatic amide00low000000
N-(3-acetylphenyl)-5-propan-2-yl-3-isoxazolecarboxamidearomatic amide00low000000
N,N-dicyclohexyl-5-propyl-3-isoxazolecarboxamidearomatic amide;
heteroarene
00low000000
N-(6-tert-butyl-3-cyano-4,5,6,7-tetrahydro-1-benzothiophen-2-yl)-5-cyclopropyl-3-isoxazolecarboxamidearomatic amide;
heteroarene
00low000000
5-amino-1-[(3-methoxyphenyl)methyl]-N-(4-methylphenyl)-4-triazolecarboxamidearomatic amide00low000000
2-[[cyclohexyl(oxo)methyl]amino]-3-thiophenecarboxamidearomatic amide;
thiophenes
00low000000
5-(4-methyl-1-naphthalenyl)-N-phenyl-2-furancarboxamidearomatic amide;
furans
00low000000
5-(2-methylphenyl)-N-(phenylmethyl)-2-furancarboxamidearomatic amide;
heteroarene
00low000000
N-[3-(7-methyl-2-imidazo[1,2-a]pyridinyl)phenyl]-2-thiophenecarboxamidearomatic amide00low000000
2-chloro-N-(1-methyl-3-pyrazolyl)acetamidearomatic amide00low000000
N-(5-carbamoyl-2-methoxyphenyl)-3-(2,4-dimethoxyphenyl)-4-oxo-2-sulfanylidene-1H-quinazoline-7-carboxamidearomatic amide00low000000
N-(4-chloro-2,5-dimethoxyphenyl)-5-cyclopropyl-3-isoxazolecarboxamidearomatic amide00low000000
4-[3-[(3-chloro-4-fluoroanilino)-oxomethyl]-7-oxo-1H-pyrazolo[1,5-a]pyrimidin-5-yl]-1-piperidinecarboxylic acid tert-butyl esteraromatic amide00low000000
N-(4-ethoxyphenyl)-1,5-dimethyl-4-oxo-2-pyrrolo[3,2-c]quinolinecarboxamidearomatic amide00low000000
platensimycinaromatic amide;
cyclic ether;
cyclic ketone;
dihydroxybenzoic acid;
monocarboxylic acid amide;
polycyclic cage
antibacterial agent;
antimicrobial agent;
bacterial metabolite;
EC 2.3.1.85 (fatty acid synthase) inhibitor
00low000000
granisetron hydrochloridearomatic amide;
indazoles
00low000000
2-chloro-N-[3-(2-thiazolo[5,4-b]pyridinyl)phenyl]-3-pyridinecarboxamidearomatic amide00low000000
N-(5-methyl-1,3,4-thiadiazol-2-yl)-2-[[1-(phenylmethyl)-2-imidazolyl]thio]acetamidearomatic amide00low000000
N-[5-[(2-methylphenyl)methylthio]-1,3,4-thiadiazol-2-yl]-2-thiophen-2-ylacetamidearomatic amide00low000000
a 770041aromatic amide00low000000
N-[4-(1-adamantylsulfamoyl)phenyl]-4-bromo-1-methyl-3-pyrazolecarboxamidearomatic amide00low000000
N-[3-(3,5-dimethyl-1-piperidinyl)propyl]-4,5,6,7-tetrahydro-1-benzothiophene-3-carboxamidearomatic amide;
thiophenes
00low000000
4-chloro-N-(4-ethylphenyl)-3-methyl-5-isoxazolecarboxamidearomatic amide00low000000
lenvatinibaromatic amide;
aromatic ether;
cyclopropanes;
monocarboxylic acid amide;
monochlorobenzenes;
phenylureas;
quinolines
antineoplastic agent;
EC 2.7.10.1 (receptor protein-tyrosine kinase) inhibitor;
fibroblast growth factor receptor antagonist;
orphan drug;
vascular endothelial growth factor receptor antagonist
00low000000
cfm 1571aromatic amide00low000000
mirabegron1,3-thiazoles;
aromatic amide;
ethanolamines;
monocarboxylic acid amide
beta-adrenergic agonist00low000000
jte 907aromatic amide;
quinolines
00low000000
osi 930aromatic amide00low000000
avanafilaromatic amide;
monocarboxylic acid amide;
organochlorine compound;
prolinols;
pyrimidines
EC 3.1.4.* (phosphoric diester hydrolase) inhibitor;
vasodilator agent
00low000000
scio-469aromatic amide;
aromatic ketone;
chloroindole;
dicarboxylic acid diamide;
indolecarboxamide;
monofluorobenzenes;
N-acylpiperazine;
N-alkylpiperazine
antineoplastic agent;
apoptosis inducer;
EC 2.7.11.24 (mitogen-activated protein kinase) inhibitor
00low000000
rivaroxabanaromatic amide;
lactam;
monocarboxylic acid amide;
morpholines;
organochlorine compound;
oxazolidinone;
thiophenes
anticoagulant;
EC 3.4.21.6 (coagulation factor Xa) inhibitor
00low000000
2-((aminocarbonyl)amino)-5-(4-fluorophenyl)-3-thiophenecarboxamidearomatic amide;
thiophenes
00low000000
ym 201636aromatic amide00low000000
osu 03012antibiotic antifungal drug;
aromatic amide;
glycine derivative;
organofluorine compound;
phenanthrenes;
pyrazoles
antineoplastic agent;
apoptosis inducer;
EC 2.7.11.1 (non-specific serine/threonine protein kinase) inhibitor
00low000000
ly-2157299aromatic amide;
methylpyridines;
monocarboxylic acid amide;
pyrrolopyrazole;
quinolines
antineoplastic agent;
TGFbeta receptor antagonist
00low000000
tolfenpyradaromatic amide;
aromatic ether;
organochlorine compound;
pyrazole insecticide
agrochemical;
antifungal agent;
EC 1.3.5.1 [succinate dehydrogenase (quinone)] inhibitor;
mitochondrial NADH:ubiquinone reductase inhibitor
00low000000
azd 7762aromatic amide;
thiophenes
00low000000
ethaboxam1,3-thiazoles;
aromatic amide;
aromatic amine;
nitrile;
secondary amino compound;
thiophenes
00low000000
penthiopyradaromatic amide;
organofluorine compound;
pyrazoles;
thiophenes
00low000000
[5-hydroxy-3-(4-methoxyphenyl)-5-(trifluoromethyl)-4H-pyrazol-1-yl]-thiophen-2-ylmethanonearomatic amide;
thiophenes
00low000000
VPC 23019aromatic amide;
D-serine derivative;
organic phosphate;
phosphoric ester;
secondary carboxamide
sphingosine-1-phosphate receptor 1 antagonist;
sphingosine-1-phosphate receptor 3 antagonist
00low000000
4-[2-(2-chloro-4-fluoroanilino)-5-methyl-4-pyrimidinyl]-N-[(1S)-1-(3-chlorophenyl)-2-hydroxyethyl]-1H-pyrrole-2-carboxamidearomatic amide;
heteroarene
00low000000
4-cyano-N-[4-(4-methyl-1-piperazinyl)-2-(4-methyl-1-piperidinyl)phenyl]-1H-pyrrole-2-carboxamidearomatic amide00low000000
5-fluoro-1,3-dimethyl-N-[2-(4-methylpentan-2-yl)phenyl]pyrazole-4-carboxamidearomatic amide;
organofluorine compound;
pyrazoles
00low000000
n-(2-(1,1'-bicyclopropyl)-2-ylphenyl)-3-(difluoromethyl)-1-methyl-1h-pyrazole-4-carboxamidearomatic amide;
cyclopropanes;
organofluorine compound;
pyrazoles;
ring assembly
00low000000
N-[2-methoxy-5-(4-morpholinylsulfonyl)phenyl]-4,5,6,7-tetrahydro-1-benzothiophene-2-carboxamidearomatic amide00low000000
3-(2,4-dimethoxyphenyl)-N-(3-fluoro-4-methylphenyl)-4-oxo-2-sulfanylidene-1H-quinazoline-7-carboxamidearomatic amide00low000000
N-Cyclohexyl-5-(2-thienyl)-1,2-oxazole-3-carboxamidearomatic amide;
heteroarene
00low000000
2-[[1,3-dimethyl-7-(4-methylphenyl)-2,4-dioxo-5-pyrimido[4,5-d]pyrimidinyl]thio]-N-(5-methyl-3-isoxazolyl)acetamidearomatic amide00low000000
fluxapyroxadanilide fungicide;
aromatic amide;
biphenyls;
pyrazoles;
trifluorobenzene
antifungal agrochemical;
EC 1.3.5.1 [succinate dehydrogenase (quinone)] inhibitor
00low000000
N-(3-cyano-4,5,6,7-tetrahydro-1-benzothiophen-2-yl)-5-methyl-4-nitro-3-isoxazolecarboxamidearomatic amide;
heteroarene
00low000000
N-(3-carbamoyl-4,5,6,7-tetrahydro-1-benzothiophen-2-yl)-5-methyl-4-nitro-3-isoxazolecarboxamidearomatic amide;
thiophenes
00low000000
N-(4-acetylphenyl)-5,6-dihydro-4H-cyclopenta[d]isoxazole-3-carboxamidearomatic amide00low000000
dafadine Caromatic amide;
aromatic ether;
difluorobenzene;
isoxazoles;
N-acylpiperidine;
pyridines
P450 inhibitor00low000000
dafadine Baromatic amide;
aromatic ether;
isoxazoles;
monochlorobenzenes;
monofluorobenzenes;
N-acylpiperidine;
pyridines
P450 inhibitor00low000000
5-amino-N-(2-methoxy-5-methylphenyl)-1-[[3-(trifluoromethyl)phenyl]methyl]-4-triazolecarboxamidearomatic amide00low000000
vx-770aromatic amide;
monocarboxylic acid amide;
phenols;
quinolone
CFTR potentiator;
orphan drug
00low000000
lumacaftoraromatic amide;
benzodioxoles;
benzoic acids;
cyclopropanes;
organofluorine compound;
pyridines
CFTR potentiator;
orphan drug
00low000000
platencinaromatic amide;
cyclic ketone;
dihydroxybenzoic acid;
monocarboxylic acid amide;
polycyclic cage
antibacterial agent;
antimicrobial agent;
bacterial metabolite;
EC 2.3.1.85 (fatty acid synthase) inhibitor
00low000000
4-methyl-N-(3-methylbutyl)-5-(5-methyl-3-phenyl-4H-isoxazol-5-yl)-2-thiazolecarboxamidearomatic amide;
thiazoles
00low000000
4-[[[5-[[[(2S)-1-[(2-methylpropan-2-yl)oxy]-6-[[(2-methylpropan-2-yl)oxy-oxomethyl]amino]-1-oxohexan-2-yl]amino]-oxomethyl]-1H-imidazol-4-yl]-oxomethyl]amino]benzoic acid ethyl esteraromatic amide;
tert-butyl ester
00low000000
2-[[[4-[(3-methylanilino)-oxomethyl]-1H-imidazol-5-yl]-oxomethyl]amino]acetic acid (phenylmethyl) esteraromatic amide00low000000
N4-(4-methoxyphenyl)-N5-[(1S)-1-phenylethyl]-1H-imidazole-4,5-dicarboxamidearomatic amide00low000000
2-[[[4-[(4-chloroanilino)-oxomethyl]-1H-imidazol-5-yl]-oxomethyl]amino]acetic acid tert-butyl esteraromatic amide;
tert-butyl ester
00low000000
(2S)-2-[[[4-[(4-chloroanilino)-oxomethyl]-1H-imidazol-5-yl]-oxomethyl]amino]-6-[[(2-methylpropan-2-yl)oxy-oxomethyl]amino]hexanoic acid tert-butyl esteraromatic amide;
tert-butyl ester
00low000000
(2S)-2-[[[4-[[4-[[[(2-methylpropan-2-yl)oxy-oxomethyl]amino]methyl]anilino]-oxomethyl]-1H-imidazol-5-yl]-oxomethyl]amino]propanoic acid tert-butyl esteraromatic amide;
tert-butyl ester
00low000000
N4-(4-methoxyphenyl)-N5-[(1R)-1-phenylethyl]-1H-imidazole-4,5-dicarboxamidearomatic amide00low000000
amg 1aromatic amide00low000000
N-(2-aminophenyl)-2-pyrazinecarboxamidearomatic amide00low000000
5-(3-hydroxyphenyl)-N-[2-(4-morpholinyl)ethyl]-3-isoxazolecarboxamidearomatic amide;
heteroarene
00low000000
n-cyclopropyl-5-(thiophen-2-yl)isoxazole-3-carboxamidearomatic amide;
heteroarene
00low000000
N-(5-chloro-2,4-dimethoxyphenyl)-1-methyl-4-(4-morpholinylsulfonyl)-2-pyrrolecarboxamidearomatic amide00low000000
4-(1-((5-((2,6-dimethylphenoxy)methyl)-3-isoxazolyl)carbonyl)-4-piperidinyl)pyridinearomatic amide;
aromatic ether;
isoxazoles;
N-acylpiperidine;
pyridines
geroprotector;
P450 inhibitor
00low000000
dafadine Daromatic amide;
aromatic ether;
isoxazoles;
N-acylpiperidine;
organofluorine compound;
pyridines
P450 inhibitor00low000000
dafadine Oaromatic amide;
aromatic ether;
isoxazoles;
N-acylpiperidine;
pyridines;
ring assembly
P450 inhibitor00low000000
bms 777607aromatic amide00low000000
suvorexant1,3-benzoxazoles;
aromatic amide;
diazepine;
organochlorine compound;
triazoles
central nervous system depressant;
orexin receptor antagonist
00low000000
N-[(2R,3S)-2-[[[[(3,5-dimethyl-4-isoxazolyl)amino]-oxomethyl]-methylamino]methyl]-5-[(2S)-1-hydroxypropan-2-yl]-3-methyl-6-oxo-2,3,4,7-tetrahydro-1,5-benzoxazonin-9-yl]-4,4,4-trifluorobutanamidearomatic amide00low000000
N-[(2S,3S)-5-[(2R)-1-hydroxypropan-2-yl]-3-methyl-2-[[methyl-[oxo-(propan-2-ylamino)methyl]amino]methyl]-6-oxo-3,4-dihydro-2H-1,5-benzoxazocin-10-yl]cyclopropanecarboxamidearomatic amide00low000000
N-[(2S,3S)-5-[(2R)-1-hydroxypropan-2-yl]-3-methyl-2-(methylaminomethyl)-6-oxo-3,4-dihydro-2H-1,5-benzoxazocin-10-yl]cyclopropanecarboxamidearomatic amide00low000000
N-[(2S,3S)-2-[[[[(3,5-dimethyl-4-isoxazolyl)amino]-oxomethyl]-methylamino]methyl]-5-[(2R)-1-hydroxypropan-2-yl]-3-methyl-6-oxo-3,4-dihydro-2H-1,5-benzoxazocin-8-yl]-4,4,4-trifluorobutanamidearomatic amide00low000000
N-[(2S,3S)-2-[[[(cyclohexylamino)-oxomethyl]-methylamino]methyl]-5-[(2R)-1-hydroxypropan-2-yl]-3-methyl-6-oxo-3,4-dihydro-2H-1,5-benzoxazocin-8-yl]-4,4,4-trifluorobutanamidearomatic amide00low000000
N-[(2S,3S)-5-[(2R)-1-hydroxypropan-2-yl]-3-methyl-2-[[methyl-[oxo-(propan-2-ylamino)methyl]amino]methyl]-6-oxo-3,4-dihydro-2H-1,5-benzoxazocin-8-yl]cyclopropanecarboxamidearomatic amide00low000000
N-[(2R,3S)-2-[[cyclopropylmethyl(methyl)amino]methyl]-5-[(2S)-1-hydroxypropan-2-yl]-3-methyl-6-oxo-2,3,4,7-tetrahydro-1,5-benzoxazonin-9-yl]-4,4,4-trifluorobutanamidearomatic amide00low000000
N-[(2S,3S)-2-[[[(cyclohexylamino)-oxomethyl]-methylamino]methyl]-5-[(2R)-1-hydroxypropan-2-yl]-3-methyl-6-oxo-3,4-dihydro-2H-1,5-benzoxazocin-8-yl]cyclohexanecarboxamidearomatic amide00low000000
5-(2,5-difluorophenyl)-N-(2,6-dimethylphenyl)-2-furancarboxamidearomatic amide;
furans
00low000000
5-(2,5-dichlorophenyl)-N-(2,6-dimethoxyphenyl)-2-furancarboxamidearomatic amide;
furans
00low000000
5-(2,5-dichlorophenyl)-N-[2,6-di(propan-2-yl)phenyl]-2-furancarboxamidearomatic amide;
furans
00low000000
5-(2,5-dichlorophenyl)-N-(2,6-diethylphenyl)-2-furancarboxamidearomatic amide;
furans
00low000000
N-(2,6-dimethylphenyl)-5-(4-methyl-3-thiophenyl)-2-furancarboxamidearomatic amide;
furans
00low000000
N-[(1R)-2-(tert-butylamino)-2-oxo-1-(3-pyridinyl)ethyl]-N-(4-tert-butylphenyl)-2-furancarboxamidearomatic amide;
furans
00low000000
fluazaindolizinearomatic amide;
imidazopyridine;
monocarboxylic acid amide;
monochlorobenzenes;
monomethoxybenzene;
N-sulfonylcarboxamide;
organofluorine pesticide
agrochemical;
nematicide
00low000000
ve 821aromatic amide00low000000
N-[2-(3-oxo-4H-quinoxalin-2-yl)-4-propan-2-ylphenyl]-2-thiophenecarboxamidearomatic amide00low000000
N-[9-(dichloromethylene)-1,2,3,4-tetrahydro-1,4-methanonaphthalen-5-yl]-3-(difluoromethyl)-1-methylpyrazole-4-carboxamidearomatic amide;
bridged compound;
olefinic compound;
organochlorine compound;
organofluorine compound;
pyrazoles
00low000000
coumermycinaromatic amide;
coumarins;
glycoside;
heteroarenecarboxylate ester;
pyrroles
antimicrobial agent;
antineoplastic agent;
bacterial metabolite;
DNA synthesis inhibitor;
Hsp90 inhibitor;
topoisomerase IV inhibitor
00low000000
1-butyl-4-hydroxy-N-(3-methyl-2-pyridinyl)-2-oxo-3-quinolinecarboxamidearomatic amide;
quinolines
00low000000
roquinimexaromatic amide00low000000
N-(2-chlorophenyl)-4-hydroxy-2-oxo-1-pentyl-3-quinolinecarboxamidearomatic amide00low000000
4-hydroxy-1-(2-methylpropyl)-2-oxo-N-(2-sulfamoylphenyl)-3-quinolinecarboxamidearomatic amide00low000000
4-hydroxy-2-oxo-1-propyl-N-(pyridin-4-ylmethyl)-3-quinolinecarboxamidearomatic amide;
quinolines
00low000000
lfm a13aromatic amide;
dibromobenzene;
enamide;
enol;
nitrile;
secondary carboxamide
antineoplastic agent;
apoptosis inducer;
EC 2.7.10.2 (non-specific protein-tyrosine kinase) inhibitor;
EC 2.7.11.21 (polo kinase) inhibitor;
geroprotector;
platelet aggregation inhibitor
00low000000
laquinimodaromatic amide00low000000
N-[(4-chlorophenyl)methyl]-4-hydroxy-2-oxo-1-prop-2-enyl-3-quinolinecarboxamidearomatic amide;
quinolines
00low000000
4-hydroxy-2-oxo-N-[3-(trifluoromethyl)phenyl]-1H-quinoline-3-carboxamidearomatic amide00low000000
4-hydroxy-1-methyl-2-oxo-N-(4-oxo-2-propyl-3-quinazolinyl)-3-quinolinecarboxamidearomatic amide;
quinolines
00low000000
1-butyl-N-[(4-chlorophenyl)methyl]-4-hydroxy-2-oxo-3-quinolinecarboxamidearomatic amide;
quinolines
00low000000
N'-[(2-chlorophenyl)-oxomethyl]-1-ethyl-4-hydroxy-2-oxo-3-quinolinecarbohydrazidearomatic amide;
quinolines
00low000000
4-hydroxy-1-methyl-N'-[(3-methylphenyl)-oxomethyl]-2-oxo-3-quinolinecarbohydrazidearomatic amide;
quinolines
00low000000
N-(2-aminophenyl)-1-butyl-4-hydroxy-2-oxo-3-quinolinecarboxamidearomatic amide00low000000
4-hydroxy-2-oxo-1-prop-2-enyl-N-(3-pyridinyl)-3-quinolinecarboxamidearomatic amide;
quinolines
00low000000
LSM-23565aromatic amide;
quinolines
00low000000
1-ethyl-4-hydroxy-2-oxo-N'-(1-oxoheptyl)-3-quinolinecarbohydrazidearomatic amide;
quinolines
00low000000
1-ethyl-N-(2-fluorophenyl)-4-hydroxy-2-oxo-3-quinolinecarboxamidearomatic amide00low000000
N-(2-aminophenyl)-4-hydroxy-2-oxo-1-pentyl-3-quinolinecarboxamidearomatic amide00low000000
teriflunomide(trifluoromethyl)benzenes;
aromatic amide;
enamide;
enol;
nitrile;
secondary carboxamide
drug metabolite;
EC 1.3.98.1 [dihydroorotate oxidase (fumarate)] inhibitor;
hepatotoxic agent;
non-steroidal anti-inflammatory drug;
tyrosine kinase inhibitor
00low000000
1-ethyl-4-hydroxy-2-oxo-N'-(1-oxodecyl)-3-quinolinecarbohydrazidearomatic amide;
quinolines
00low000000
LSM-31922aromatic amide;
quinolines
00low000000
1-ethyl-4-hydroxy-2-oxo-N-(3-pyridinylmethyl)-3-quinolinecarboxamidearomatic amide;
quinolines
00low000000
N-(1H-benzimidazol-2-yl)-1-ethyl-4-hydroxy-2-oxo-3-quinolinecarboxamidearomatic amide;
quinolines
00low000000
N-[(3,4-dimethoxyphenyl)methyl]-4-hydroxy-2-oxo-1-propyl-3-quinolinecarboxamidearomatic amide;
quinolines
00low000000
4-hydroxy-N-(2-methyl-4-oxo-3-quinazolinyl)-1-(2-methylpropyl)-2-oxo-5,6,7,8-tetrahydroquinoline-3-carboxamidearomatic amide;
quinolines
00low000000
4-hydroxy-1-(2-methylpropyl)-2-oxo-N-[4-oxo-2-(phenylmethyl)-3-quinazolinyl]-5,6,7,8-tetrahydroquinoline-3-carboxamidearomatic amide;
quinolines
00low000000
4-hydroxy-2-oxo-1-pentyl-N-(2-pyridinylmethyl)-3-quinolinecarboxamidearomatic amide;
quinolines
00low000000
N-[2-(4-chlorophenyl)ethyl]-4-hydroxy-2-oxo-1-propyl-3-quinolinecarboxamidearomatic amide;
quinolines
00low000000
abt-267aromatic amide;
carbamate ester;
dipeptide;
pyrrolidines
antiviral drug;
hepatitis C virus nonstructural protein 5A inhibitor
00low000000
3-(difluoromethyl)-N-methoxy-1-methyl-N-[1-(2,4,6-trichlorophenyl)propan-2-yl]pyrazole-4-carboxamidearomatic amide;
monocarboxylic acid amide;
organofluorine compound;
pyrazoles;
trichlorobenzene
00low000000
AKB48aromatic amide;
indazoles
00low000000
Adb-fubinacaaromatic amide;
indazoles
00low000000
n-(1-adamantyl)-1-(5-fluoropentyl)-1h-indazole-3-carboxamidearomatic amide;
indazoles
00low000000
4-chloro-N-[(4-chlorophenyl)methyl]-3-nitro-1H-pyrazole-5-carboxamidearomatic amide;
heteroarene
00low000000
1-[4-[[oxo-(7-oxo-4H-isothiazolo[4,3-d]pyrimidin-3-yl)methyl]amino]phenyl]-3-piperidinecarboxylic acid ethyl esteraromatic amide00low000000
1-[4-[[(5-methyl-7-oxo-4H-isothiazolo[4,3-d]pyrimidin-3-yl)-oxomethyl]amino]phenyl]-3-piperidinecarboxylic acid ethyl esteraromatic amide00low000000
5-(3-hydroxymethyl-3-methyl-1-triazeno)imidazole-4-carboxamidearomatic amide;
heteroarene
00low000000
ver 52296aromatic amide;
isoxazoles;
monocarboxylic acid amide;
morpholines;
resorcinols
angiogenesis inhibitor;
antineoplastic agent;
Hsp90 inhibitor
00low000000
dabigatran etexilatearomatic amide;
benzimidazoles;
beta-alanine derivative;
carboxamidine;
carboxylic ester;
pyridines
anticoagulant;
EC 3.4.21.5 (thrombin) inhibitor;
prodrug
00low000000
ConditionIndicatedStudiesFirst YearLast YearAverage AgeRelationship StrengthTrialspre-19901990's2000's2010'spost-2020
Inflammation02010201014.0high000100
Innate Inflammatory Response02010201014.0high000100
Malaria, Falciparum02014201410.0high000010
Plasmodium falciparum Malaria02014201410.0high000010