| Assay ID | Title | Year | Journal | Article |
|---|
| AID233940 | Ratio between Ki of L1210-P enzyme and Michaelis-Menten constant (kM) | 2000 | Journal of medicinal chemistry, Nov-30, Volume: 43, Issue:24
| 5-Substituted N(4)-hydroxy-2'-deoxycytidines and their 5'-monophosphates: synthesis, conformation, interaction with tumor thymidylate synthase, and in vitro antitumor activity. |
| AID233942 | Ratio between Ki of L1210-R enzyme and Michaelis-Menten constant (kM) | 2000 | Journal of medicinal chemistry, Nov-30, Volume: 43, Issue:24
| 5-Substituted N(4)-hydroxy-2'-deoxycytidines and their 5'-monophosphates: synthesis, conformation, interaction with tumor thymidylate synthase, and in vitro antitumor activity. |
| AID1134942 | Competitive inhibition of thymidylate synthase purified from methotrexate-resistant Lactobacillus casei using 2'-deoxy[5-3H]uridine 5'-phosphate by radioisotope assay | 1979 | Journal of medicinal chemistry, Sep, Volume: 22, Issue:9
| 5-Cyano-2'-deoxyuridine 5'-phosphate: a potent competitive inhibitor of thymidylate synthetase. |
| AID228252 | Time-independent inhibition of thymidylate synthase from parenteral L1210 cells | 2000 | Journal of medicinal chemistry, Nov-30, Volume: 43, Issue:24
| 5-Substituted N(4)-hydroxy-2'-deoxycytidines and their 5'-monophosphates: synthesis, conformation, interaction with tumor thymidylate synthase, and in vitro antitumor activity. |
| AID1147594 | Inhibition of amethopterin-resistant Lactobacillus casei thymidylate synthetase-catalyzed 5-BrdUMP dehalogenation by absorbance analysis in absence of CH2-H4-folate | 1977 | Journal of medicinal chemistry, Nov, Volume: 20, Issue:11
| Inhibition of Lactobacillus casei thymidylate synthetase by 5-substituted 2'-deoxyuridylates. Preliminary quantitative structure-activity relationship. |
| AID228251 | Time-independent inhibition of thymidylate synthase from FdUrd-resistant L1210 cells | 2000 | Journal of medicinal chemistry, Nov-30, Volume: 43, Issue:24
| 5-Substituted N(4)-hydroxy-2'-deoxycytidines and their 5'-monophosphates: synthesis, conformation, interaction with tumor thymidylate synthase, and in vitro antitumor activity. |
| AID220360 | The compound was evaluated for the inhibition of dTMP synthetase from Lactobacillus casei | 1981 | Journal of medicinal chemistry, Dec, Volume: 24, Issue:12
| Inhibition of thymidylate synthetase by 5-alkynyl-2'-deoxyuridylates. |
| AID1147592 | Inhibition of amethopterin-resistant Lactobacillus casei thymidylate synthetase-catalyzed dTMP formation using dUMP as substrate by spectrophotometric analysis in presence of CH2-H4-folate | 1977 | Journal of medicinal chemistry, Nov, Volume: 20, Issue:11
| Inhibition of Lactobacillus casei thymidylate synthetase by 5-substituted 2'-deoxyuridylates. Preliminary quantitative structure-activity relationship. |
| AID99552 | Inhibition of dTMP synthetase in the absence of CH2-H4 folate Lactobacillus casei | 1983 | Journal of medicinal chemistry, Aug, Volume: 26, Issue:8
| Mechanism of action of 2',5-difluoro-1-arabinosyluracil. |
| [information is prepared from bioassay data collected from National Library of Medicine (NLM), extracted Dec-2023] |