| Assay ID | Title | Year | Journal | Article |
|---|
| AID739283 | Displacement of [3H]-CP55940 from human CB2 receptor after 90 mins by liquid scintillation spectrophotometer analysis | 2013 | Bioorganic & medicinal chemistry, Apr-01, Volume: 21, Issue:7
| Novel antiobesity agents: synthesis and pharmacological evaluation of analogues of Rimonabant and of LH21. |
| AID739282 | Displacement of [3H]-CP55940 from human CB1 receptor after 90 mins by liquid scintillation spectrophotometer analysis | 2013 | Bioorganic & medicinal chemistry, Apr-01, Volume: 21, Issue:7
| Novel antiobesity agents: synthesis and pharmacological evaluation of analogues of Rimonabant and of LH21. |
| AID127386 | Effect on electrically evoked contractions in mouse vas deferens at 10E-8 to 10E-6 M concentration; No effect | 2004 | Journal of medicinal chemistry, May-20, Volume: 47, Issue:11
| Discovery of 5-(4-chlorophenyl)-1-(2,4-dichlorophenyl)-3-hexyl-1h-1,2,4-triazole, a novel in vivo cannabinoid antagonist containing a 1,2,4-triazole motif. |
| AID227373 | Effect on cannabinoid tetrad (nociception, temperature, spontaneous motility and catalepsy) of behavioral test; no significant effect | 2004 | Journal of medicinal chemistry, May-20, Volume: 47, Issue:11
| Discovery of 5-(4-chlorophenyl)-1-(2,4-dichlorophenyl)-3-hexyl-1h-1,2,4-triazole, a novel in vivo cannabinoid antagonist containing a 1,2,4-triazole motif. |
| AID49488 | Ability to displace [3H]SR-141,716A radioligand from cannabinoid receptor 1 in rat cerebellar membrane | 2004 | Journal of medicinal chemistry, May-20, Volume: 47, Issue:11
| Discovery of 5-(4-chlorophenyl)-1-(2,4-dichlorophenyl)-3-hexyl-1h-1,2,4-triazole, a novel in vivo cannabinoid antagonist containing a 1,2,4-triazole motif. |
| AID1177626 | Inverse agonist activity at human CB1 receptor | 2013 | Bioorganic & medicinal chemistry letters, Sep-01, Volume: 23, Issue:17
| Peripherally restricted CB1 receptor blockers. |
| AID49489 | Ability to displace [3H]WIN-55212-2 radioligand from cannabinoid receptor 1 in rat cerebellar membrane | 2004 | Journal of medicinal chemistry, May-20, Volume: 47, Issue:11
| Discovery of 5-(4-chlorophenyl)-1-(2,4-dichlorophenyl)-3-hexyl-1h-1,2,4-triazole, a novel in vivo cannabinoid antagonist containing a 1,2,4-triazole motif. |
| AID1177627 | Inverse agonist activity at rat CB1 receptor | 2013 | Bioorganic & medicinal chemistry letters, Sep-01, Volume: 23, Issue:17
| Peripherally restricted CB1 receptor blockers. |
| AID74172 | Effect on electrically evoked contractions in mesenteric plexus longitudinal muscles of guinea pig at 10E-8 to 2.4E-6 M; No effect | 2004 | Journal of medicinal chemistry, May-20, Volume: 47, Issue:11
| Discovery of 5-(4-chlorophenyl)-1-(2,4-dichlorophenyl)-3-hexyl-1h-1,2,4-triazole, a novel in vivo cannabinoid antagonist containing a 1,2,4-triazole motif. |
| [information is prepared from bioassay data collected from National Library of Medicine (NLM), extracted Dec-2023] |