Assay ID | Title | Year | Journal | Article |
AID488691 | Selectivity ratio of IC50 for SERT to IC50 for NET | 2010 | Bioorganic & medicinal chemistry, Jun-01, Volume: 18, Issue:11
| Synthesis and in vitro toxicity of 4-MTA, its characteristic clandestine synthesis byproducts and related sulfur substituted alpha-alkylthioamphetamines. |
AID488700 | Cytotoxicity against human SH-SY5Y cells assessed as cell viability after 48 hrs by neutral red assay | 2010 | Bioorganic & medicinal chemistry, Jun-01, Volume: 18, Issue:11
| Synthesis and in vitro toxicity of 4-MTA, its characteristic clandestine synthesis byproducts and related sulfur substituted alpha-alkylthioamphetamines. |
AID395043 | Inhibition of MAOA in rat brain mitochondria | 2009 | Bioorganic & medicinal chemistry, Mar-15, Volume: 17, Issue:6
| Naphthylisopropylamine and N-benzylamphetamine derivatives as monoamine oxidase inhibitors. |
AID576805 | Cytotoxicity against human chemoresistant DG75 cells expressing SERT assessed as decrease in cell viability 10 or 50 uM after 72 hrs Alamar blue assay | 2011 | Bioorganic & medicinal chemistry, Feb-01, Volume: 19, Issue:3
| Synthesis and serotonin transporter activity of 1,3-bis(aryl)-2-nitro-1-propenes as a new class of anticancer agents. |
AID488690 | Selectivity ratio of IC50 for SERT to IC50 for DAT | 2010 | Bioorganic & medicinal chemistry, Jun-01, Volume: 18, Issue:11
| Synthesis and in vitro toxicity of 4-MTA, its characteristic clandestine synthesis byproducts and related sulfur substituted alpha-alkylthioamphetamines. |
AID145706 | Compound was tested for the ability to inhibit [3H]norepinephrine binding to Norepinephrine transporter in rat synaptosomes | 1998 | Journal of medicinal chemistry, Mar-12, Volume: 41, Issue:6
| Synthesis and pharmacological evaluation of ring-methylated derivatives of 3,4-(methylenedioxy)amphetamine (MDA). |
AID234659 | selectivity is the ratio between IC50 values of 5-HTand NE | 1998 | Journal of medicinal chemistry, Mar-12, Volume: 41, Issue:6
| Synthesis and pharmacological evaluation of ring-methylated derivatives of 3,4-(methylenedioxy)amphetamine (MDA). |
AID471634 | Cytotoxicity against human HEK293 cells after 48 hrs by neutral red assay | 2009 | European journal of medicinal chemistry, Dec, Volume: 44, Issue:12
| Synthesis and serotonin transporter activity of sulphur-substituted alpha-alkyl phenethylamines as a new class of anticancer agents. |
AID488695 | Cytotoxicity against human HEK293 cells assessed as cell viability after 48 hrs by neutral red assay | 2010 | Bioorganic & medicinal chemistry, Jun-01, Volume: 18, Issue:11
| Synthesis and in vitro toxicity of 4-MTA, its characteristic clandestine synthesis byproducts and related sulfur substituted alpha-alkylthioamphetamines. |
AID488698 | Cytotoxicity against human HEK293 cells over expressing human DAT assessed as cell viability after 48 hrs by neutral red assay | 2010 | Bioorganic & medicinal chemistry, Jun-01, Volume: 18, Issue:11
| Synthesis and in vitro toxicity of 4-MTA, its characteristic clandestine synthesis byproducts and related sulfur substituted alpha-alkylthioamphetamines. |
AID471639 | Cytotoxicity against human SH-SY5Y cells after 48 hrs by neutral red assay | 2009 | European journal of medicinal chemistry, Dec, Volume: 44, Issue:12
| Synthesis and serotonin transporter activity of sulphur-substituted alpha-alkyl phenethylamines as a new class of anticancer agents. |
AID576811 | Cytotoxicity against human HEK293 cells assessed as decrease in cell viability after 48 hrs neutral red dye assay | 2011 | Bioorganic & medicinal chemistry, Feb-01, Volume: 19, Issue:3
| Synthesis and serotonin transporter activity of 1,3-bis(aryl)-2-nitro-1-propenes as a new class of anticancer agents. |
AID241440 | Inhibitory concentration against monoamine oxidase A in rat brain mitochondrial suspension | 2005 | Journal of medicinal chemistry, Apr-07, Volume: 48, Issue:7
| Sulfur-substituted alpha-alkyl phenethylamines as selective and reversible MAO-A inhibitors: biological activities, CoMFA analysis, and active site modeling. |
AID576803 | Cytotoxicity against human SH-SY5Y cells expressing human SERT assessed as decrease in cell viability after 48 hrs neutral red dye assay | 2011 | Bioorganic & medicinal chemistry, Feb-01, Volume: 19, Issue:3
| Synthesis and serotonin transporter activity of 1,3-bis(aryl)-2-nitro-1-propenes as a new class of anticancer agents. |
AID471630 | Inhibition of [3H]5-HT reuptake at rat SERT expressed in HEK293 cells after 2 mins by liquid scintillation counting | 2009 | European journal of medicinal chemistry, Dec, Volume: 44, Issue:12
| Synthesis and serotonin transporter activity of sulphur-substituted alpha-alkyl phenethylamines as a new class of anticancer agents. |
AID471638 | Induction of human SERT-dependent cytotoxicity in SERT expressing human DG75 cells after 48 hrs by neutral red assay | 2009 | European journal of medicinal chemistry, Dec, Volume: 44, Issue:12
| Synthesis and serotonin transporter activity of sulphur-substituted alpha-alkyl phenethylamines as a new class of anticancer agents. |
AID471670 | Selectivity ratio of IC50 for DAT in rat brain synaptosome to IC50 for SERT in rat brain synaptosome | 2009 | European journal of medicinal chemistry, Dec, Volume: 44, Issue:12
| Synthesis and serotonin transporter activity of sulphur-substituted alpha-alkyl phenethylamines as a new class of anticancer agents. |
AID471673 | Induction of human NET-dependent cytotoxicity in NET expressing HEK293 cells after 48 hrs by neutral red assay | 2009 | European journal of medicinal chemistry, Dec, Volume: 44, Issue:12
| Synthesis and serotonin transporter activity of sulphur-substituted alpha-alkyl phenethylamines as a new class of anticancer agents. |
AID471665 | Inhibition of [3H]5-HT uptake at SERT in rat brain synaptosome | 2009 | European journal of medicinal chemistry, Dec, Volume: 44, Issue:12
| Synthesis and serotonin transporter activity of sulphur-substituted alpha-alkyl phenethylamines as a new class of anticancer agents. |
AID471671 | Selectivity ratio of IC50 for NET in rat brain synaptosome to IC50 for SERT in rat brain synaptosome | 2009 | European journal of medicinal chemistry, Dec, Volume: 44, Issue:12
| Synthesis and serotonin transporter activity of sulphur-substituted alpha-alkyl phenethylamines as a new class of anticancer agents. |
AID576813 | Inhibition of [3H]-serotonin reuptake at human SERT expressed in HEK293 cells after 15 to 20 mins by fluorescence neurotransmitter transporter assay | 2011 | Bioorganic & medicinal chemistry, Feb-01, Volume: 19, Issue:3
| Synthesis and serotonin transporter activity of 1,3-bis(aryl)-2-nitro-1-propenes as a new class of anticancer agents. |
AID471635 | Induction of human SERT-dependent cytotoxicity in SERT expressing HEK293 cells after 48 hrs by neutral red assay | 2009 | European journal of medicinal chemistry, Dec, Volume: 44, Issue:12
| Synthesis and serotonin transporter activity of sulphur-substituted alpha-alkyl phenethylamines as a new class of anticancer agents. |
AID471672 | Induction of human DAT-dependent cytotoxicity in DAT expressing HEK293 cells after 48 hrs by neutral red assay | 2009 | European journal of medicinal chemistry, Dec, Volume: 44, Issue:12
| Synthesis and serotonin transporter activity of sulphur-substituted alpha-alkyl phenethylamines as a new class of anticancer agents. |
AID471667 | Inhibition of human noradrenaline transporter | 2009 | European journal of medicinal chemistry, Dec, Volume: 44, Issue:12
| Synthesis and serotonin transporter activity of sulphur-substituted alpha-alkyl phenethylamines as a new class of anticancer agents. |
AID471666 | Inhibition of [3H]5-HT uptake at SERT | 2009 | European journal of medicinal chemistry, Dec, Volume: 44, Issue:12
| Synthesis and serotonin transporter activity of sulphur-substituted alpha-alkyl phenethylamines as a new class of anticancer agents. |
AID576812 | Cytotoxicity against human HEK293 cells expressing human SERT assessed as decrease in cell viability after 48 hrs neutral red dye assay | 2011 | Bioorganic & medicinal chemistry, Feb-01, Volume: 19, Issue:3
| Synthesis and serotonin transporter activity of 1,3-bis(aryl)-2-nitro-1-propenes as a new class of anticancer agents. |
AID179206 | Compound was tested for its ability to inhibit [3H]dopamine uptake in rat synaptosomes | 1998 | Journal of medicinal chemistry, Mar-12, Volume: 41, Issue:6
| Synthesis and pharmacological evaluation of ring-methylated derivatives of 3,4-(methylenedioxy)amphetamine (MDA). |
AID471640 | Cytotoxicity against human HEK293 cells at 1 uM after 48 hrs by neutral red assay | 2009 | European journal of medicinal chemistry, Dec, Volume: 44, Issue:12
| Synthesis and serotonin transporter activity of sulphur-substituted alpha-alkyl phenethylamines as a new class of anticancer agents. |
AID204225 | Activity towards Serotonin transporter was determined by the ability to inhibit [3H]5-HT uptake in rat synaptosomes | 1998 | Journal of medicinal chemistry, Mar-12, Volume: 41, Issue:6
| Synthesis and pharmacological evaluation of ring-methylated derivatives of 3,4-(methylenedioxy)amphetamine (MDA). |
AID471668 | Inhibition of human dopamine transporter | 2009 | European journal of medicinal chemistry, Dec, Volume: 44, Issue:12
| Synthesis and serotonin transporter activity of sulphur-substituted alpha-alkyl phenethylamines as a new class of anticancer agents. |
AID471669 | Inhibition of [3H]5-HT uptake at human SERT expressed in HEK293 cells after 10 mins by scintillation counting | 2009 | European journal of medicinal chemistry, Dec, Volume: 44, Issue:12
| Synthesis and serotonin transporter activity of sulphur-substituted alpha-alkyl phenethylamines as a new class of anticancer agents. |
AID234658 | selectivity is the ratio between IC50 values of 5-HTand DA | 1998 | Journal of medicinal chemistry, Mar-12, Volume: 41, Issue:6
| Synthesis and pharmacological evaluation of ring-methylated derivatives of 3,4-(methylenedioxy)amphetamine (MDA). |
AID488697 | Cytotoxicity against human HEK293 cells over expressing human NET assessed as cell viability after 48 hrs by neutral red assay | 2010 | Bioorganic & medicinal chemistry, Jun-01, Volume: 18, Issue:11
| Synthesis and in vitro toxicity of 4-MTA, its characteristic clandestine synthesis byproducts and related sulfur substituted alpha-alkylthioamphetamines. |
AID471641 | Induction of human SERT-dependent cytotoxicity in SERT expressing HEK293 cells at 1 uM after 48 hrs by neutral red assay | 2009 | European journal of medicinal chemistry, Dec, Volume: 44, Issue:12
| Synthesis and serotonin transporter activity of sulphur-substituted alpha-alkyl phenethylamines as a new class of anticancer agents. |
AID488699 | Cytotoxicity against rat PC12 cells assessed as cell viability after 48 hrs by neutral red assay | 2010 | Bioorganic & medicinal chemistry, Jun-01, Volume: 18, Issue:11
| Synthesis and in vitro toxicity of 4-MTA, its characteristic clandestine synthesis byproducts and related sulfur substituted alpha-alkylthioamphetamines. |
AID488696 | Cytotoxicity against human HEK293 cells over expressing human SERT assessed as cell viability after 48 hrs by neutral red assay | 2010 | Bioorganic & medicinal chemistry, Jun-01, Volume: 18, Issue:11
| Synthesis and in vitro toxicity of 4-MTA, its characteristic clandestine synthesis byproducts and related sulfur substituted alpha-alkylthioamphetamines. |
AID395041 | Inhibition of MAOB in rat brain mitochondria at 100 uM | 2009 | Bioorganic & medicinal chemistry, Mar-15, Volume: 17, Issue:6
| Naphthylisopropylamine and N-benzylamphetamine derivatives as monoamine oxidase inhibitors. |
[information is prepared from bioassay data collected from National Library of Medicine (NLM), extracted Dec-2023] |