| Assay ID | Title | Year | Journal | Article |
|---|
| AID1296008 | Cytotoxic Profiling of Annotated Libraries Using Quantitative High-Throughput Screening | 2020 | SLAS discovery : advancing life sciences R & D, 01, Volume: 25, Issue:1
| Cytotoxic Profiling of Annotated and Diverse Chemical Libraries Using Quantitative High-Throughput Screening. |
| AID1346986 | P-glycoprotein substrates identified in KB-3-1 adenocarcinoma cell line, qHTS therapeutic library screen | 2019 | Molecular pharmacology, 11, Volume: 96, Issue:5
| A High-Throughput Screen of a Library of Therapeutics Identifies Cytotoxic Substrates of P-glycoprotein. |
| AID1347160 | Primary screen NINDS Rhodamine qHTS for Zika virus inhibitors | 2020 | Proceedings of the National Academy of Sciences of the United States of America, 12-08, Volume: 117, Issue:49
| Therapeutic candidates for the Zika virus identified by a high-throughput screen for Zika protease inhibitors. |
| AID1346987 | P-glycoprotein substrates identified in KB-8-5-11 adenocarcinoma cell line, qHTS therapeutic library screen | 2019 | Molecular pharmacology, 11, Volume: 96, Issue:5
| A High-Throughput Screen of a Library of Therapeutics Identifies Cytotoxic Substrates of P-glycoprotein. |
| AID1347159 | Primary screen GU Rhodamine qHTS for Zika virus inhibitors: Unlinked NS2B-NS3 protease assay | 2020 | Proceedings of the National Academy of Sciences of the United States of America, 12-08, Volume: 117, Issue:49
| Therapeutic candidates for the Zika virus identified by a high-throughput screen for Zika protease inhibitors. |
| AID392917 | Inhibition of human immunoprecipitated histone acetyltransferase p300 in U937 cell nuclear extracts assessed as remaining enzyme activity at 50 uM | 2009 | Bioorganic & medicinal chemistry letters, Feb-15, Volume: 19, Issue:4
| Identification of 4-hydroxyquinolines inhibitors of p300/CBP histone acetyltransferases. |
| AID392678 | Inhibition of human histone acetyltransferase in U937 cell nuclear extracts at 50 uM | 2009 | Bioorganic & medicinal chemistry letters, Feb-15, Volume: 19, Issue:4
| Identification of 4-hydroxyquinolines inhibitors of p300/CBP histone acetyltransferases. |
| AID1422590 | Inhibition of recombinant human GCN5 using histone peptide as substrate in presence of [14C]-acetyl CoA by microbeta counting method | 2018 | Bioorganic & medicinal chemistry, 11-01, Volume: 26, Issue:20
| Discovery and biological evaluation of thiobarbituric derivatives as potent p300/CBP inhibitors. |
| AID1408177 | Inhibition of recombinant human GST-tagged Gcn5 using H3 as substrate in presence of [3H]-acetyl-CoA by phosphor image analysis | 2018 | European journal of medicinal chemistry, Sep-05, Volume: 157 | Identification of novel inhibitors of histone acetyltransferase hMOF through high throughput screening. |
| AID331953 | Inhibition of recombinant CBP in human U937 cells at 50 uM | 2008 | Bioorganic & medicinal chemistry letters, May-01, Volume: 18, Issue:9
| Identification of long chain alkylidenemalonates as novel small molecule modulators of histone acetyltransferases. |
| AID392681 | Inhibition of human histone acetyltransferase GCN5 in U937 cell nuclear extracts assessed as remaining enzyme activity at 50 uM | 2009 | Bioorganic & medicinal chemistry letters, Feb-15, Volume: 19, Issue:4
| Identification of 4-hydroxyquinolines inhibitors of p300/CBP histone acetyltransferases. |
| AID272386 | Inhibition of HAT in human U937 cells at 50 uM | 2006 | Journal of medicinal chemistry, Nov-16, Volume: 49, Issue:23
| Small-molecule inhibitors of histone acetyltransferase activity: identification and biological properties. |
| AID392682 | Inhibition of human GST-fused histone acetyltransferase PCAF in U937 cell nuclear extracts assessed as remaining enzyme activity at 50 uM | 2009 | Bioorganic & medicinal chemistry letters, Feb-15, Volume: 19, Issue:4
| Identification of 4-hydroxyquinolines inhibitors of p300/CBP histone acetyltransferases. |
| AID392680 | Inhibition of human GST-fused histone acetyltransferase CBP in U937 cell nuclear extracts assessed as remaining enzyme activity at 50 uM | 2009 | Bioorganic & medicinal chemistry letters, Feb-15, Volume: 19, Issue:4
| Identification of 4-hydroxyquinolines inhibitors of p300/CBP histone acetyltransferases. |
| [information is prepared from bioassay data collected from National Library of Medicine (NLM), extracted Dec-2023] |