Assay ID | Title | Year | Journal | Article |
AID716291 | Ratio of ZnPhe EC50 to compound EC50 for human CCR8 transfected in COS7 cells coexpressing chimeric Gqi4myr assessed as IP3 turnover by liquid scintillation counting analysis | 2012 | Journal of medicinal chemistry, Sep-27, Volume: 55, Issue:18
| Modulation in selectivity and allosteric properties of small-molecule ligands for CC-chemokine receptors. |
AID716298 | Allosteric modulation at human CCR5 transfected in COS7 cells coexpressing chimeric Gqi4myr assessed as [3H]IP3 turnover by liquid scintillation counting analysis relative to basal level | 2012 | Journal of medicinal chemistry, Sep-27, Volume: 55, Issue:18
| Modulation in selectivity and allosteric properties of small-molecule ligands for CC-chemokine receptors. |
AID716294 | Allosteric modulation at human CCR8 transfected in COS7 cells assessed as [3H]IP3 turnover by liquid scintillation counting analysis | 2012 | Journal of medicinal chemistry, Sep-27, Volume: 55, Issue:18
| Modulation in selectivity and allosteric properties of small-molecule ligands for CC-chemokine receptors. |
AID716289 | Displacement of [125I]-CCL3 from human CCR1 transfected in COS7 cells coexpressing chimeric Gqi4myr after 3 hrs | 2012 | Journal of medicinal chemistry, Sep-27, Volume: 55, Issue:18
| Modulation in selectivity and allosteric properties of small-molecule ligands for CC-chemokine receptors. |
AID218537 | Inhibition of beta-hematin formation; Not active | 2004 | Journal of medicinal chemistry, May-20, Volume: 47, Issue:11
| In vitro antimalarial activity of a series of cationic 2,2'-bipyridyl- and 1,10-phenanthrolineplatinum(II) benzoylthiourea complexes. |
AID158223 | In vitro antimalarial activity against chloroquine-sensitive Plasmodium falciparum D10; Not determined | 2004 | Journal of medicinal chemistry, May-20, Volume: 47, Issue:11
| In vitro antimalarial activity of a series of cationic 2,2'-bipyridyl- and 1,10-phenanthrolineplatinum(II) benzoylthiourea complexes. |
AID716295 | Allosteric modulation at human CCR5 transfected in COS7 cells coexpressing chimeric Gqi4myr assessed as [3H]IP3 turnover by liquid scintillation counting analysis | 2012 | Journal of medicinal chemistry, Sep-27, Volume: 55, Issue:18
| Modulation in selectivity and allosteric properties of small-molecule ligands for CC-chemokine receptors. |
AID716297 | Allosteric modulation at human CCR1 transfected in COS7 cells coexpressing chimeric Gqi4myr assessed as [3H]IP3 turnover by liquid scintillation counting analysis relative to basal level | 2012 | Journal of medicinal chemistry, Sep-27, Volume: 55, Issue:18
| Modulation in selectivity and allosteric properties of small-molecule ligands for CC-chemokine receptors. |
AID716300 | Ratio of ZnPhe EC50 to compound EC50 for human CCR1 transfected in COS7 cells coexpressing chimeric Gqi4myr assessed as IP3 turnover by liquid scintillation counting analysis | 2012 | Journal of medicinal chemistry, Sep-27, Volume: 55, Issue:18
| Modulation in selectivity and allosteric properties of small-molecule ligands for CC-chemokine receptors. |
AID716302 | Ratio of ZnPhe EC50 to compound EC50 for human CCR5 transfected in COS7 cells coexpressing chimeric Gqi4myr assessed as IP3 turnover by liquid scintillation counting analysis | 2012 | Journal of medicinal chemistry, Sep-27, Volume: 55, Issue:18
| Modulation in selectivity and allosteric properties of small-molecule ligands for CC-chemokine receptors. |
AID716290 | Allosteric modulation at human CCR8 transfected in COS7 cells coexpressing chimeric Gqi4myr assessed as [3H]IP3 turnover by liquid scintillation counting analysis relative to basal level | 2012 | Journal of medicinal chemistry, Sep-27, Volume: 55, Issue:18
| Modulation in selectivity and allosteric properties of small-molecule ligands for CC-chemokine receptors. |
AID716296 | Allosteric modulation at human CCR1 transfected in COS7 cells coexpressing chimeric Gqi4myr assessed as {3H]IP3 turnover by liquid scintillation counting analysis | 2012 | Journal of medicinal chemistry, Sep-27, Volume: 55, Issue:18
| Modulation in selectivity and allosteric properties of small-molecule ligands for CC-chemokine receptors. |
AID716287 | Displacement of [125I]-CCL3 from human CCR5 transfected in COS7 cells coexpressing chimeric Gqi4myr after 3 hrs | 2012 | Journal of medicinal chemistry, Sep-27, Volume: 55, Issue:18
| Modulation in selectivity and allosteric properties of small-molecule ligands for CC-chemokine receptors. |
AID158225 | In vitro antimalarial activity against chloroquine-sensitive Plasmodium falciparum K1; Not determined | 2004 | Journal of medicinal chemistry, May-20, Volume: 47, Issue:11
| In vitro antimalarial activity of a series of cationic 2,2'-bipyridyl- and 1,10-phenanthrolineplatinum(II) benzoylthiourea complexes. |
AID72977 | Ability to associate with ferriprotoporphyrin IX | 2004 | Journal of medicinal chemistry, May-20, Volume: 47, Issue:11
| In vitro antimalarial activity of a series of cationic 2,2'-bipyridyl- and 1,10-phenanthrolineplatinum(II) benzoylthiourea complexes. |
AID716288 | Displacement of [125I]-CCL3 from human CCR1 transfected in COS7 cells coexpressing chimeric Gqi4myr after 3 hrs relative to basal level | 2012 | Journal of medicinal chemistry, Sep-27, Volume: 55, Issue:18
| Modulation in selectivity and allosteric properties of small-molecule ligands for CC-chemokine receptors. |
AID716293 | Binding affinity to Zn(II) after 2 hrs using FluoZin-3 by fuorescence assay | 2012 | Journal of medicinal chemistry, Sep-27, Volume: 55, Issue:18
| Modulation in selectivity and allosteric properties of small-molecule ligands for CC-chemokine receptors. |
[information is prepared from bioassay data collected from National Library of Medicine (NLM), extracted Dec-2023] |