Assay ID | Title | Year | Journal | Article |
AID504810 | Antagonists of the Thyroid Stimulating Hormone Receptor: HTS campaign | 2010 | Endocrinology, Jul, Volume: 151, Issue:7
| A small molecule inverse agonist for the human thyroid-stimulating hormone receptor. |
AID504812 | Inverse Agonists of the Thyroid Stimulating Hormone Receptor: HTS campaign | 2010 | Endocrinology, Jul, Volume: 151, Issue:7
| A small molecule inverse agonist for the human thyroid-stimulating hormone receptor. |
AID213175 | Concentration required to inhibit 50% of I-T3 binding to hTR1 (Thyroid hormone receptor beta) was determined | 2003 | Journal of medicinal chemistry, Apr-24, Volume: 46, Issue:9
| Thyroid receptor ligands. 1. Agonist ligands selective for the thyroid receptor beta1. |
AID75733 | Effect on rat hepatic glycerophosphate dehydrogenase alpha (GPD) activity 3 days after injection of 10e-6 mol/kg. | 1992 | Journal of medicinal chemistry, Feb-07, Volume: 35, Issue:3
| alpha-Methylated analogues of triiodothyroalkanoic acids: synthesis and biological activity. |
AID213163 | Concentration required to inhibit 50% of I-T3 binding to hTR1 (Thyroid hormone receptor alpha) was determined | 2003 | Journal of medicinal chemistry, Apr-24, Volume: 46, Issue:9
| Thyroid receptor ligands. 1. Agonist ligands selective for the thyroid receptor beta1. |
AID739861 | Inhibition of human recombinant PCNA interaction with PIP box protein N-5-carboxyfluorescein-SAVLQKKITDYFHPKK after 30 mins by fluorescence polarization assay | 2013 | Bioorganic & medicinal chemistry, Apr-01, Volume: 21, Issue:7
| Small molecule inhibitors of PCNA/PIP-box interaction suppress translesion DNA synthesis. |
AID170336 | Effect on the plasma cholesterol levels after subcutaneous administration of 8 nmol/kg in Dawley rats. | 1992 | Journal of medicinal chemistry, Feb-07, Volume: 35, Issue:3
| alpha-Methylated analogues of triiodothyroalkanoic acids: synthesis and biological activity. |
AID104520 | Effect on rat hepatic Malic enzyme activity 3 days after injection of 10e-6 mol/kg. | 1992 | Journal of medicinal chemistry, Feb-07, Volume: 35, Issue:3
| alpha-Methylated analogues of triiodothyroalkanoic acids: synthesis and biological activity. |
AID170334 | Effect on the plasma cholesterol levels after subcutaneous administration of 16 nmol/kg in Dawley rats. p < 0.01 | 1992 | Journal of medicinal chemistry, Feb-07, Volume: 35, Issue:3
| alpha-Methylated analogues of triiodothyroalkanoic acids: synthesis and biological activity. |
AID299948 | Inhibition of human thyroid hormone receptor beta 1 | 2007 | Bioorganic & medicinal chemistry, Aug-01, Volume: 15, Issue:15
| QSAR study of selective ligands for the thyroid hormone receptor beta. |
AID104519 | Effect on rat hepatic Malic enzyme activity 3 days after injection of 10e-5 mol/kg. | 1992 | Journal of medicinal chemistry, Feb-07, Volume: 35, Issue:3
| alpha-Methylated analogues of triiodothyroalkanoic acids: synthesis and biological activity. |
AID231783 | Ratio of concentration required to inhibit 50% of I-T3 binding to hTR-alpha1 to that of concentration required to inhibit 50% of I-T3 binding to hTR-beta1 was determined | 2003 | Journal of medicinal chemistry, Apr-24, Volume: 46, Issue:9
| Thyroid receptor ligands. 1. Agonist ligands selective for the thyroid receptor beta1. |
AID75734 | Effect on rat hepatic glycerophosphate dehydrogenase alpha (GPD) activity relative to L-T3. | 1992 | Journal of medicinal chemistry, Feb-07, Volume: 35, Issue:3
| alpha-Methylated analogues of triiodothyroalkanoic acids: synthesis and biological activity. |
AID311017 | Inhibition of thyroid hormone receptor beta | 2007 | Bioorganic & medicinal chemistry, Jul-01, Volume: 15, Issue:13
| 2D QSAR studies on thyroid hormone receptor ligands. |
AID311016 | Inhibition of thyroid hormone receptor alpha | 2007 | Bioorganic & medicinal chemistry, Jul-01, Volume: 15, Issue:13
| 2D QSAR studies on thyroid hormone receptor ligands. |
AID104517 | Effect on rat hepatic Malic enzyme activity relative to L-T3. | 1992 | Journal of medicinal chemistry, Feb-07, Volume: 35, Issue:3
| alpha-Methylated analogues of triiodothyroalkanoic acids: synthesis and biological activity. |
AID1797782 | TRalpha-Binding Assay. from Article 10.1021/jm021080f: \\Thyroid receptor ligands. 1. Agonist ligands selective for the thyroid receptor beta1.\\ | 2003 | Journal of medicinal chemistry, Apr-24, Volume: 46, Issue:9
| Thyroid receptor ligands. 1. Agonist ligands selective for the thyroid receptor beta1. |
AID1797784 | TRbeta-Binding Assay from Article 10.1021/jm021080f: \\Thyroid receptor ligands. 1. Agonist ligands selective for the thyroid receptor beta1.\\ | 2003 | Journal of medicinal chemistry, Apr-24, Volume: 46, Issue:9
| Thyroid receptor ligands. 1. Agonist ligands selective for the thyroid receptor beta1. |
[information is prepared from bioassay data collected from National Library of Medicine (NLM), extracted Dec-2023] |