Assay ID | Title | Year | Journal | Article |
AID313111 | Displacement of [3H]SCH-23390 from rat dopamine D1 receptor | 2007 | Journal of medicinal chemistry, Jan-25, Volume: 50, Issue:2
| Advances in development of dopaminergic aporphinoids. |
AID569899 | Binding affinity to dopamine D1 receptor low binding site by radioligand displacement assay | 2011 | ACS medicinal chemistry letters, Mar-10, Volume: 2, Issue:3
| Synthesis and Evaluation of Fluorinated Aporphines: Potential Positron Emission Tomography Ligands for D2 Receptors |
AID226917 | Ratio of binding affinity of D2 to binding affinity of D1 | 1990 | Journal of medicinal chemistry, Jun, Volume: 33, Issue:6
| Synthesis and dopamine receptor affinities of enantiomers of 2-substituted apomorphines and their N-n-propyl analogues. |
AID317241 | Displacement of [3H]neomonapride from dopamine D2 receptor in rat striatum | 2008 | Journal of medicinal chemistry, Feb-28, Volume: 51, Issue:4
| Synthesis and dopamine receptor affinities of N-alkyl-11-hydroxy-2-methoxynoraporphines: N-alkyl substituents determine D1 versus D2 receptor selectivity. |
AID317240 | Displacement of [3H]SCH-23390 from dopamine D1 receptor in rat striatum | 2008 | Journal of medicinal chemistry, Feb-28, Volume: 51, Issue:4
| Synthesis and dopamine receptor affinities of N-alkyl-11-hydroxy-2-methoxynoraporphines: N-alkyl substituents determine D1 versus D2 receptor selectivity. |
AID65113 | Binding affinity at rat striatal Dopamine receptor D2 using [3H]- piperone radioligand | 1990 | Journal of medicinal chemistry, Jun, Volume: 33, Issue:6
| Synthesis and dopamine receptor affinities of enantiomers of 2-substituted apomorphines and their N-n-propyl analogues. |
AID61403 | Binding affinity against Dopamine receptor D2 from rat brain corpus striatum membrane | 1990 | Journal of medicinal chemistry, Dec, Volume: 33, Issue:12
| Synthesis and dopamine receptor affinity of (R)-(-)-2-fluoro-N-n-propylnorapomorphine: a highly potent and selective dopamine D2 agonist. |
AID317242 | Selectivity ratio of rat dopamine D2 receptor to rat dopamine D1 receptor | 2008 | Journal of medicinal chemistry, Feb-28, Volume: 51, Issue:4
| Synthesis and dopamine receptor affinities of N-alkyl-11-hydroxy-2-methoxynoraporphines: N-alkyl substituents determine D1 versus D2 receptor selectivity. |
AID313112 | Displacement of [3H]raclopride from rat dopamine D2 receptor | 2007 | Journal of medicinal chemistry, Jan-25, Volume: 50, Issue:2
| Advances in development of dopaminergic aporphinoids. |
AID569896 | Displacement of [3H]SCH23390 from dopamine D2 receptor low binding site in Sprague-Dawley rat striatum by scintillation counting | 2011 | ACS medicinal chemistry letters, Mar-10, Volume: 2, Issue:3
| Synthesis and Evaluation of Fluorinated Aporphines: Potential Positron Emission Tomography Ligands for D2 Receptors |
AID569900 | Binding affinity to dopamine D1 receptor high binding site by radioligand displacement assay | 2011 | ACS medicinal chemistry letters, Mar-10, Volume: 2, Issue:3
| Synthesis and Evaluation of Fluorinated Aporphines: Potential Positron Emission Tomography Ligands for D2 Receptors |
AID569901 | Displacement of [3H]domperidone from human dopamine D3 receptor expressed in human HEK293 cells by scintillation counting | 2011 | ACS medicinal chemistry letters, Mar-10, Volume: 2, Issue:3
| Synthesis and Evaluation of Fluorinated Aporphines: Potential Positron Emission Tomography Ligands for D2 Receptors |
AID62464 | Agonistic activity against calf striatal Dopamine receptor using [3H]- ADTN radioligand | 1990 | Journal of medicinal chemistry, Jun, Volume: 33, Issue:6
| Synthesis and dopamine receptor affinities of enantiomers of 2-substituted apomorphines and their N-n-propyl analogues. |
AID226901 | Potency ratio as ratio of IC50 of D2 receptor to that of D1 receptor | 1990 | Journal of medicinal chemistry, Dec, Volume: 33, Issue:12
| Synthesis and dopamine receptor affinity of (R)-(-)-2-fluoro-N-n-propylnorapomorphine: a highly potent and selective dopamine D2 agonist. |
AID61026 | Binding affinity against Dopamine receptor D1 from rat brain corpus striatum membrane | 1990 | Journal of medicinal chemistry, Dec, Volume: 33, Issue:12
| Synthesis and dopamine receptor affinity of (R)-(-)-2-fluoro-N-n-propylnorapomorphine: a highly potent and selective dopamine D2 agonist. |
AID61497 | Binding affinity at rat striatal Dopamine receptor D1 using [3H]- SCH-23390 radioligand | 1990 | Journal of medicinal chemistry, Jun, Volume: 33, Issue:6
| Synthesis and dopamine receptor affinities of enantiomers of 2-substituted apomorphines and their N-n-propyl analogues. |
AID569897 | Displacement of [3H]domperidone from dopamine D2 receptor high binding site in Sprague-Dawley rat striatum by scintillation counting | 2011 | ACS medicinal chemistry letters, Mar-10, Volume: 2, Issue:3
| Synthesis and Evaluation of Fluorinated Aporphines: Potential Positron Emission Tomography Ligands for D2 Receptors |
[information is prepared from bioassay data collected from National Library of Medicine (NLM), extracted Dec-2023] |