2-deoxy-2-((18)F)fluoro-beta-D-glucose : no description available [CHeBI]
ID Source | ID |
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PubMed CID | 9920539 |
CHEMBL ID | 497613 |
CHEBI ID | 49131 |
Synonym |
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2-deoxy-2-((18)f)fluoro-beta-d-glucopyranose |
2-deoxy-2-((18)f)fluoro-beta-d-glucose |
CHEBI:49131 , |
CHEMBL497613 |
fludeoxyglucose-f18 |
105851-18-1 |
2-deoxy-2-(fluoro-18f)-beta-d-glucopyranose |
7R6S3C8YL2 , |
unii-7r6s3c8yl2 |
beta-d-fludeoxyglucopyranose f-18 |
.beta.-d-fludeoxyglucopyranose f-18 |
2-deoxy-2-(fluoro-18f)-.beta.-d-glucopyranose |
(2r,3r,4s,5s,6r)-3-(18f)fluoranyl-6-(hydroxymethyl)oxane-2,4,5-triol |
2-[18f]fluoro-2-deoxy-beta-d-glucopyranose |
Class | Description |
---|---|
2-deoxy-2-((18)F)fluoro-D-glucopyranose | |
2-deoxy-2-fluoro-beta-D-glucose |
Assay ID | Title | Year | Journal | Article |
---|---|---|---|---|
AID476419 | Ratio of drug uptake in tumor to blood of mouse S180 cells xenografted Kunming mouse at 10 to 20 uCi, iv after 120 mins by gamma counting | 2010 | Bioorganic & medicinal chemistry, Apr-01, Volume: 18, Issue:7 ISSN: 1464-3391 | (18)F Labeled benzimidazole derivatives as potential radiotracer for positron emission tomography (PET) tumor imaging. |
AID476215 | Ratio of drug uptake in tumor to blood of mouse S180 cells xenografted Kunming mouse at 10 to 20 uCi, iv after 5 mins by gamma counting | 2010 | Bioorganic & medicinal chemistry, Apr-01, Volume: 18, Issue:7 ISSN: 1464-3391 | (18)F Labeled benzimidazole derivatives as potential radiotracer for positron emission tomography (PET) tumor imaging. |
AID476216 | Ratio of drug uptake in tumor to muscle of mouse S180 cells xenografted Kunming mouse at 10 to 20 uCi, iv after 5 mins by gamma counting | 2010 | Bioorganic & medicinal chemistry, Apr-01, Volume: 18, Issue:7 ISSN: 1464-3391 | (18)F Labeled benzimidazole derivatives as potential radiotracer for positron emission tomography (PET) tumor imaging. |
AID696418 | Ratio of drug uptake in tumor to lung of mouse Colon 26 cells xenografted BALB/c mouse at 150 uCi administered parenterally after 2 hrs by PET analysis | 2011 | Journal of medicinal chemistry, Oct-13, Volume: 54, Issue:19 ISSN: 1520-4804 | In vitro cellular uptake and dimerization of signal transducer and activator of transcription-3 (STAT3) identify the photosensitizing and imaging-potential of isomeric photosensitizers derived from chlorophyll-a and bacteriochlorophyll-a. |
AID434403 | Biodistribution in S180 tumor-bearing KM mouse liver assessed per gram of tissue at 240 to 370 kBq, iv after 30 mins | 2009 | Bioorganic & medicinal chemistry letters, Aug-15, Volume: 19, Issue:16 ISSN: 1464-3405 | Synthesis and evaluation of novel F-18 labeled fluoroarylvaline derivatives: potential PET imaging agents for tumor detection. |
AID476225 | Biodistribution in mouse S180 cells xenografted Kunming mouse blood at 10 to 20 uCi, iv after 15 mins by gamma counting | 2010 | Bioorganic & medicinal chemistry, Apr-01, Volume: 18, Issue:7 ISSN: 1464-3391 | (18)F Labeled benzimidazole derivatives as potential radiotracer for positron emission tomography (PET) tumor imaging. |
AID434402 | Biodistribution in S180 tumor-bearing KM mouse liver assessed per gram of tissue at 240 to 370 kBq, iv after 60 mins | 2009 | Bioorganic & medicinal chemistry letters, Aug-15, Volume: 19, Issue:16 ISSN: 1464-3405 | Synthesis and evaluation of novel F-18 labeled fluoroarylvaline derivatives: potential PET imaging agents for tumor detection. |
AID476230 | Ratio of drug uptake in tumor to brain of mouse S180 cells xenografted Kunming mouse at 10 to 20 uCi, iv after 15 mins by gamma counting | 2010 | Bioorganic & medicinal chemistry, Apr-01, Volume: 18, Issue:7 ISSN: 1464-3391 | (18)F Labeled benzimidazole derivatives as potential radiotracer for positron emission tomography (PET) tumor imaging. |
AID434412 | Biodistribution in S180 tumor-bearing KM mouse blood assessed per gram of tissue weight at 240 to 370 kBq, iv after 60 mins | 2009 | Bioorganic & medicinal chemistry letters, Aug-15, Volume: 19, Issue:16 ISSN: 1464-3405 | Synthesis and evaluation of novel F-18 labeled fluoroarylvaline derivatives: potential PET imaging agents for tumor detection. |
AID434436 | Ratio of drug level in S180 tumor to muscleKM mouse at 240 to 370 kBq, iv after 15 mins | 2009 | Bioorganic & medicinal chemistry letters, Aug-15, Volume: 19, Issue:16 ISSN: 1464-3405 | Synthesis and evaluation of novel F-18 labeled fluoroarylvaline derivatives: potential PET imaging agents for tumor detection. |
AID434439 | Ratio of drug level in S180 tumor to muscleKM mouse at 240 to 370 kBq, iv after 120 mins | 2009 | Bioorganic & medicinal chemistry letters, Aug-15, Volume: 19, Issue:16 ISSN: 1464-3405 | Synthesis and evaluation of novel F-18 labeled fluoroarylvaline derivatives: potential PET imaging agents for tumor detection. |
AID434405 | Biodistribution in S180 tumor-bearing KM mouse liver assessed per gram of tissue weight at 240 to 370 kBq, iv after 5 mins | 2009 | Bioorganic & medicinal chemistry letters, Aug-15, Volume: 19, Issue:16 ISSN: 1464-3405 | Synthesis and evaluation of novel F-18 labeled fluoroarylvaline derivatives: potential PET imaging agents for tumor detection. |
AID434419 | Biodistribution in S180 tumor-bearing KM mouse brain assessed per gram of tissue at 240 to 370 kBq, iv after 120 mins | 2009 | Bioorganic & medicinal chemistry letters, Aug-15, Volume: 19, Issue:16 ISSN: 1464-3405 | Synthesis and evaluation of novel F-18 labeled fluoroarylvaline derivatives: potential PET imaging agents for tumor detection. |
AID434434 | Ratio of drug level in S180 tumor to brain KM mouse at 240 to 370 kBq, iv after 120 mins | 2009 | Bioorganic & medicinal chemistry letters, Aug-15, Volume: 19, Issue:16 ISSN: 1464-3405 | Synthesis and evaluation of novel F-18 labeled fluoroarylvaline derivatives: potential PET imaging agents for tumor detection. |
AID476263 | Biodistribution in mouse S180 cells xenografted Kunming mouse muscle at 10 to 20 uCi, iv after 120 mins by gamma counting | 2010 | Bioorganic & medicinal chemistry, Apr-01, Volume: 18, Issue:7 ISSN: 1464-3391 | (18)F Labeled benzimidazole derivatives as potential radiotracer for positron emission tomography (PET) tumor imaging. |
AID434392 | Biodistribution in S180 tumor-bearing KM mouse kidney assessed per gram of tissue at 240 to 370 kBq, iv after 60 mins | 2009 | Bioorganic & medicinal chemistry letters, Aug-15, Volume: 19, Issue:16 ISSN: 1464-3405 | Synthesis and evaluation of novel F-18 labeled fluoroarylvaline derivatives: potential PET imaging agents for tumor detection. |
AID1060655 | Drug uptake in mouse xenografted with human K562 cells expressing Bcr-Abl after 45 mins by PET analysis | 2014 | Bioorganic & medicinal chemistry, Jan-01, Volume: 22, Issue:1 ISSN: 1464-3391 | Imatinib analogs as potential agents for PET imaging of Bcr-Abl and c-KIT expression at a kinase level. |
AID434422 | Biodistribution in S180 tumor present in KM mouse assessed per gram of tissue at 240 to 370 kBq, iv after 30 mins | 2009 | Bioorganic & medicinal chemistry letters, Aug-15, Volume: 19, Issue:16 ISSN: 1464-3405 | Synthesis and evaluation of novel F-18 labeled fluoroarylvaline derivatives: potential PET imaging agents for tumor detection. |
AID476242 | Ratio of drug uptake in tumor to muscle of mouse S180 cells xenografted Kunming mouse at 10 to 20 uCi, iv after 30 mins by gamma counting | 2010 | Bioorganic & medicinal chemistry, Apr-01, Volume: 18, Issue:7 ISSN: 1464-3391 | (18)F Labeled benzimidazole derivatives as potential radiotracer for positron emission tomography (PET) tumor imaging. |
AID434395 | Biodistribution in S180 tumor-bearing KM mouse kidney assessed per gram of tissue at 240 to 370 kBq, iv after 5 mins | 2009 | Bioorganic & medicinal chemistry letters, Aug-15, Volume: 19, Issue:16 ISSN: 1464-3405 | Synthesis and evaluation of novel F-18 labeled fluoroarylvaline derivatives: potential PET imaging agents for tumor detection. |
AID434423 | Biodistribution in S180 tumor present in KM mouse assessed per gram of tissue at 240 to 370 kBq, iv after 60 mins | 2009 | Bioorganic & medicinal chemistry letters, Aug-15, Volume: 19, Issue:16 ISSN: 1464-3405 | Synthesis and evaluation of novel F-18 labeled fluoroarylvaline derivatives: potential PET imaging agents for tumor detection. |
AID476231 | Biodistribution in mouse S180 cells xenografted Kunming mouse heart at 10 to 20 uCi, iv after 30 mins by gamma counting | 2010 | Bioorganic & medicinal chemistry, Apr-01, Volume: 18, Issue:7 ISSN: 1464-3391 | (18)F Labeled benzimidazole derivatives as potential radiotracer for positron emission tomography (PET) tumor imaging. |
AID463482 | Biodistribution in tumor of Fischer 344 rat bearing rat 9L cells at 20 uCi, iv after 60 mins | 2010 | Journal of medicinal chemistry, Jan-28, Volume: 53, Issue:2 ISSN: 1520-4804 | Synthesis, radiolabeling, and biological evaluation of (R)- and (S)-2-amino-3-[(18)F]fluoro-2-methylpropanoic acid (FAMP) and (R)- and (S)-3-[(18)F]fluoro-2-methyl-2-N-(methylamino)propanoic acid (NMeFAMP) as potential PET radioligands for imaging brain t |
AID696416 | Ratio of drug uptake in tumor to spleen of mouse Colon 26 cells xenografted BALB/c mouse at 150 uCi administered parenterally after 2 hrs by PET analysis | 2011 | Journal of medicinal chemistry, Oct-13, Volume: 54, Issue:19 ISSN: 1520-4804 | In vitro cellular uptake and dimerization of signal transducer and activator of transcription-3 (STAT3) identify the photosensitizing and imaging-potential of isomeric photosensitizers derived from chlorophyll-a and bacteriochlorophyll-a. |
AID434435 | Ratio of drug level in S180 tumor to muscleKM mouse at 240 to 370 kBq, iv after 5 mins | 2009 | Bioorganic & medicinal chemistry letters, Aug-15, Volume: 19, Issue:16 ISSN: 1464-3405 | Synthesis and evaluation of novel F-18 labeled fluoroarylvaline derivatives: potential PET imaging agents for tumor detection. |
AID476213 | Biodistribution in mouse S180 cells xenografted Kunming mouse brain at 10 to 20 uCi, iv after 5 mins by gamma counting | 2010 | Bioorganic & medicinal chemistry, Apr-01, Volume: 18, Issue:7 ISSN: 1464-3391 | (18)F Labeled benzimidazole derivatives as potential radiotracer for positron emission tomography (PET) tumor imaging. |
AID434413 | Biodistribution in S180 tumor-bearing KM mouse blood assessed per gram of tissue weight at 240 to 370 kBq, iv after 30 mins | 2009 | Bioorganic & medicinal chemistry letters, Aug-15, Volume: 19, Issue:16 ISSN: 1464-3405 | Synthesis and evaluation of novel F-18 labeled fluoroarylvaline derivatives: potential PET imaging agents for tumor detection. |
AID476420 | Ratio of drug uptake in tumor to muscle of mouse S180 cells xenografted Kunming mouse at 10 to 20 uCi, iv after 120 mins by gamma counting | 2010 | Bioorganic & medicinal chemistry, Apr-01, Volume: 18, Issue:7 ISSN: 1464-3391 | (18)F Labeled benzimidazole derivatives as potential radiotracer for positron emission tomography (PET) tumor imaging. |
AID476237 | Biodistribution in mouse S180 cells xenografted Kunming mouse muscle at 10 to 20 uCi, iv after 30 mins by gamma counting | 2010 | Bioorganic & medicinal chemistry, Apr-01, Volume: 18, Issue:7 ISSN: 1464-3391 | (18)F Labeled benzimidazole derivatives as potential radiotracer for positron emission tomography (PET) tumor imaging. |
AID434421 | Biodistribution in S180 tumor present in KM mouse assessed per gram of tissue at 240 to 370 kBq, iv after 15 mins | 2009 | Bioorganic & medicinal chemistry letters, Aug-15, Volume: 19, Issue:16 ISSN: 1464-3405 | Synthesis and evaluation of novel F-18 labeled fluoroarylvaline derivatives: potential PET imaging agents for tumor detection. |
AID434428 | Ratio of drug level in S180 tumor to blood in KM mouse at 240 to 370 kBq, iv after 60 mins | 2009 | Bioorganic & medicinal chemistry letters, Aug-15, Volume: 19, Issue:16 ISSN: 1464-3405 | Synthesis and evaluation of novel F-18 labeled fluoroarylvaline derivatives: potential PET imaging agents for tumor detection. |
AID1060654 | Drug uptake in intestine of mouse xenografted with human U87WT cells expressing human wild type c-KIT after 45 mins by PET analysis | 2014 | Bioorganic & medicinal chemistry, Jan-01, Volume: 22, Issue:1 ISSN: 1464-3391 | Imatinib analogs as potential agents for PET imaging of Bcr-Abl and c-KIT expression at a kinase level. |
AID476243 | Ratio of drug uptake in tumor to brain of mouse S180 cells xenografted Kunming mouse at 10 to 20 uCi, iv after 30 mins by gamma counting | 2010 | Bioorganic & medicinal chemistry, Apr-01, Volume: 18, Issue:7 ISSN: 1464-3391 | (18)F Labeled benzimidazole derivatives as potential radiotracer for positron emission tomography (PET) tumor imaging. |
AID434384 | Biodistribution in S180 tumor-bearing KM mouse muscle assessed per gram of tissue at 240 to 370 kBq, iv after 15 mins | 2009 | Bioorganic & medicinal chemistry letters, Aug-15, Volume: 19, Issue:16 ISSN: 1464-3405 | Synthesis and evaluation of novel F-18 labeled fluoroarylvaline derivatives: potential PET imaging agents for tumor detection. |
AID434420 | Biodistribution in S180 tumor present in KM mouse assessed per gram of tissue at 240 to 370 kBq, iv after 5 mins | 2009 | Bioorganic & medicinal chemistry letters, Aug-15, Volume: 19, Issue:16 ISSN: 1464-3405 | Synthesis and evaluation of novel F-18 labeled fluoroarylvaline derivatives: potential PET imaging agents for tumor detection. |
AID434399 | Biodistribution in S180 tumor-bearing KM mouse lung assessed per gram of tissue at 240 to 370 kBq, iv after 15 mins | 2009 | Bioorganic & medicinal chemistry letters, Aug-15, Volume: 19, Issue:16 ISSN: 1464-3405 | Synthesis and evaluation of novel F-18 labeled fluoroarylvaline derivatives: potential PET imaging agents for tumor detection. |
AID476264 | Biodistribution in mouse S180 cells xenografted Kunming mouse blood at 10 to 20 uCi, iv after 120 mins by gamma counting | 2010 | Bioorganic & medicinal chemistry, Apr-01, Volume: 18, Issue:7 ISSN: 1464-3391 | (18)F Labeled benzimidazole derivatives as potential radiotracer for positron emission tomography (PET) tumor imaging. |
AID434430 | Ratio of drug level in S180 tumor to brain KM mouse at 240 to 370 kBq, iv after 5 mins | 2009 | Bioorganic & medicinal chemistry letters, Aug-15, Volume: 19, Issue:16 ISSN: 1464-3405 | Synthesis and evaluation of novel F-18 labeled fluoroarylvaline derivatives: potential PET imaging agents for tumor detection. |
AID434374 | Biodistribution in S180 tumor-bearing KM mouse brain assessed per gram of tissue at 240 to 370 kBq, iv after 15 mins | 2009 | Bioorganic & medicinal chemistry letters, Aug-15, Volume: 19, Issue:16 ISSN: 1464-3405 | Synthesis and evaluation of novel F-18 labeled fluoroarylvaline derivatives: potential PET imaging agents for tumor detection. |
AID476207 | Biodistribution in mouse S180 cells xenografted Kunming mouse pancreas at 10 to 20 uCi, iv after 5 mins by gamma counting | 2010 | Bioorganic & medicinal chemistry, Apr-01, Volume: 18, Issue:7 ISSN: 1464-3391 | (18)F Labeled benzimidazole derivatives as potential radiotracer for positron emission tomography (PET) tumor imaging. |
AID476255 | Ratio of drug uptake in tumor to muscle of mouse S180 cells xenografted Kunming mouse at 10 to 20 uCi, iv after 60 mins by gamma counting | 2010 | Bioorganic & medicinal chemistry, Apr-01, Volume: 18, Issue:7 ISSN: 1464-3391 | (18)F Labeled benzimidazole derivatives as potential radiotracer for positron emission tomography (PET) tumor imaging. |
AID476211 | Biodistribution in mouse S180 cells xenografted Kunming mouse muscle at 10 to 20 uCi, iv after 5 mins by gamma counting | 2010 | Bioorganic & medicinal chemistry, Apr-01, Volume: 18, Issue:7 ISSN: 1464-3391 | (18)F Labeled benzimidazole derivatives as potential radiotracer for positron emission tomography (PET) tumor imaging. |
AID1060653 | Drug uptake in intestine of mouse xenografted with human U87 cells after 45 mins by PET analysis | 2014 | Bioorganic & medicinal chemistry, Jan-01, Volume: 22, Issue:1 ISSN: 1464-3391 | Imatinib analogs as potential agents for PET imaging of Bcr-Abl and c-KIT expression at a kinase level. |
AID476418 | Biodistribution in mouse S180 cells xenografted Kunming mouse tumor at 10 to 20 uCi, iv after 120 mins by gamma counting | 2010 | Bioorganic & medicinal chemistry, Apr-01, Volume: 18, Issue:7 ISSN: 1464-3391 | (18)F Labeled benzimidazole derivatives as potential radiotracer for positron emission tomography (PET) tumor imaging. |
AID434426 | Ratio of drug level in S180 tumor to blood in KM mouse at 240 to 370 kBq, iv after 15mins | 2009 | Bioorganic & medicinal chemistry letters, Aug-15, Volume: 19, Issue:16 ISSN: 1464-3405 | Synthesis and evaluation of novel F-18 labeled fluoroarylvaline derivatives: potential PET imaging agents for tumor detection. |
AID476228 | Ratio of drug uptake in tumor to blood of mouse S180 cells xenografted Kunming mouse at 10 to 20 uCi, iv after 15 mins by gamma counting | 2010 | Bioorganic & medicinal chemistry, Apr-01, Volume: 18, Issue:7 ISSN: 1464-3391 | (18)F Labeled benzimidazole derivatives as potential radiotracer for positron emission tomography (PET) tumor imaging. |
AID594522 | Drug uptake in human SY-cells xenografted mouse tumor at 200 kBq, iv after 15 to 25 mins by positron emission tomography | 2011 | Bioorganic & medicinal chemistry letters, Apr-15, Volume: 21, Issue:8 ISSN: 1464-3405 | An efficient and expedient method for the synthesis of 11C-labeled α-aminoisobutyric acid: a tumor imaging agent potentially useful for cancer diagnosis. |
AID476227 | Biodistribution in mouse S180 cells xenografted Kunming mouse tumor at 10 to 20 uCi, iv after 15 mins by gamma counting | 2010 | Bioorganic & medicinal chemistry, Apr-01, Volume: 18, Issue:7 ISSN: 1464-3391 | (18)F Labeled benzimidazole derivatives as potential radiotracer for positron emission tomography (PET) tumor imaging. |
AID476261 | Biodistribution in mouse S180 cells xenografted Kunming mouse kidney at 10 to 20 uCi, iv after 120 mins by gamma counting | 2010 | Bioorganic & medicinal chemistry, Apr-01, Volume: 18, Issue:7 ISSN: 1464-3391 | (18)F Labeled benzimidazole derivatives as potential radiotracer for positron emission tomography (PET) tumor imaging. |
AID410815 | Biodistribution in tumor of iv dosed C3H/HeJ mouse bearing mouse RIF cells assessed as relative uptake value after 3 days by PET imaging | 2009 | Journal of medicinal chemistry, Jan-22, Volume: 52, Issue:2 ISSN: 1520-4804 | Comparative positron-emission tomography (PET) imaging and phototherapeutic potential of 124I- labeled methyl- 3-(1'-iodobenzyloxyethyl)pyropheophorbide-a vs the corresponding glucose and galactose conjugates. |
AID476246 | Biodistribution in mouse S180 cells xenografted Kunming mouse pancreas at 10 to 20 uCi, iv after 60 mins by gamma counting | 2010 | Bioorganic & medicinal chemistry, Apr-01, Volume: 18, Issue:7 ISSN: 1464-3391 | (18)F Labeled benzimidazole derivatives as potential radiotracer for positron emission tomography (PET) tumor imaging. |
AID463483 | Biodistribution in tumor of Fischer 344 rat bearing rat 9L cells at 20 uCi, iv after 120 mins | 2010 | Journal of medicinal chemistry, Jan-28, Volume: 53, Issue:2 ISSN: 1520-4804 | Synthesis, radiolabeling, and biological evaluation of (R)- and (S)-2-amino-3-[(18)F]fluoro-2-methylpropanoic acid (FAMP) and (R)- and (S)-3-[(18)F]fluoro-2-methyl-2-N-(methylamino)propanoic acid (NMeFAMP) as potential PET radioligands for imaging brain t |
AID476232 | Biodistribution in mouse S180 cells xenografted Kunming mouse liver at 10 to 20 uCi, iv after 30 mins by gamma counting | 2010 | Bioorganic & medicinal chemistry, Apr-01, Volume: 18, Issue:7 ISSN: 1464-3391 | (18)F Labeled benzimidazole derivatives as potential radiotracer for positron emission tomography (PET) tumor imaging. |
AID476220 | Biodistribution in mouse S180 cells xenografted Kunming mouse pancreas at 10 to 20 uCi, iv after 15 mins by gamma counting | 2010 | Bioorganic & medicinal chemistry, Apr-01, Volume: 18, Issue:7 ISSN: 1464-3391 | (18)F Labeled benzimidazole derivatives as potential radiotracer for positron emission tomography (PET) tumor imaging. |
AID476221 | Biodistribution in mouse S180 cells xenografted Kunming mouse lung at 10 to 20 uCi, iv after 15 mins by gamma counting | 2010 | Bioorganic & medicinal chemistry, Apr-01, Volume: 18, Issue:7 ISSN: 1464-3391 | (18)F Labeled benzimidazole derivatives as potential radiotracer for positron emission tomography (PET) tumor imaging. |
AID434411 | Biodistribution in S180 tumor-bearing KM mouse blood assessed per gram of tissue weight at 240 to 370 kBq, iv after 120 mins | 2009 | Bioorganic & medicinal chemistry letters, Aug-15, Volume: 19, Issue:16 ISSN: 1464-3405 | Synthesis and evaluation of novel F-18 labeled fluoroarylvaline derivatives: potential PET imaging agents for tumor detection. |
AID434408 | Biodistribution in S180 tumor-bearing KM mouse heart assessed per gram of tissue weight at 240 to 370 kBq, iv after 30 mins | 2009 | Bioorganic & medicinal chemistry letters, Aug-15, Volume: 19, Issue:16 ISSN: 1464-3405 | Synthesis and evaluation of novel F-18 labeled fluoroarylvaline derivatives: potential PET imaging agents for tumor detection. |
AID476239 | Biodistribution in mouse S180 cells xenografted Kunming mouse brain at 10 to 20 uCi, iv after 30 mins by gamma counting | 2010 | Bioorganic & medicinal chemistry, Apr-01, Volume: 18, Issue:7 ISSN: 1464-3391 | (18)F Labeled benzimidazole derivatives as potential radiotracer for positron emission tomography (PET) tumor imaging. |
AID476247 | Biodistribution in mouse S180 cells xenografted Kunming mouse lung at 10 to 20 uCi, iv after 60 mins by gamma counting | 2010 | Bioorganic & medicinal chemistry, Apr-01, Volume: 18, Issue:7 ISSN: 1464-3391 | (18)F Labeled benzimidazole derivatives as potential radiotracer for positron emission tomography (PET) tumor imaging. |
AID434381 | Biodistribution in S180 tumor-bearing KM mouse muscle assessed per gram of tissue at 240 to 370 kBq, iv after 120 mins | 2009 | Bioorganic & medicinal chemistry letters, Aug-15, Volume: 19, Issue:16 ISSN: 1464-3405 | Synthesis and evaluation of novel F-18 labeled fluoroarylvaline derivatives: potential PET imaging agents for tumor detection. |
AID476252 | Biodistribution in mouse S180 cells xenografted Kunming mouse brain at 10 to 20 uCi, iv after 60 mins by gamma counting | 2010 | Bioorganic & medicinal chemistry, Apr-01, Volume: 18, Issue:7 ISSN: 1464-3391 | (18)F Labeled benzimidazole derivatives as potential radiotracer for positron emission tomography (PET) tumor imaging. |
AID476206 | Biodistribution in mouse S180 cells xenografted Kunming mouse liver at 10 to 20 uCi, iv after 5 mins by gamma counting | 2010 | Bioorganic & medicinal chemistry, Apr-01, Volume: 18, Issue:7 ISSN: 1464-3391 | (18)F Labeled benzimidazole derivatives as potential radiotracer for positron emission tomography (PET) tumor imaging. |
AID476248 | Biodistribution in mouse S180 cells xenografted Kunming mouse kidney at 10 to 20 uCi, iv after 60 mins by gamma counting | 2010 | Bioorganic & medicinal chemistry, Apr-01, Volume: 18, Issue:7 ISSN: 1464-3391 | (18)F Labeled benzimidazole derivatives as potential radiotracer for positron emission tomography (PET) tumor imaging. |
AID476208 | Biodistribution in mouse S180 cells xenografted Kunming mouse lung at 10 to 20 uCi, iv after 5 mins by gamma counting | 2010 | Bioorganic & medicinal chemistry, Apr-01, Volume: 18, Issue:7 ISSN: 1464-3391 | (18)F Labeled benzimidazole derivatives as potential radiotracer for positron emission tomography (PET) tumor imaging. |
AID434380 | Biodistribution in S180 tumor-bearing KM mouse spleen assessed per gram of tissue at 240 to 370 kBq, iv after 5 mins | 2009 | Bioorganic & medicinal chemistry letters, Aug-15, Volume: 19, Issue:16 ISSN: 1464-3405 | Synthesis and evaluation of novel F-18 labeled fluoroarylvaline derivatives: potential PET imaging agents for tumor detection. |
AID434396 | Biodistribution in S180 tumor-bearing KM mouse lung assessed per gram of tissue at 240 to 370 kBq, iv after 120 mins | 2009 | Bioorganic & medicinal chemistry letters, Aug-15, Volume: 19, Issue:16 ISSN: 1464-3405 | Synthesis and evaluation of novel F-18 labeled fluoroarylvaline derivatives: potential PET imaging agents for tumor detection. |
AID434393 | Biodistribution in S180 tumor-bearing KM mouse kidney assessed per gram of tissue at 240 to 370 kBq, iv after 30 mins | 2009 | Bioorganic & medicinal chemistry letters, Aug-15, Volume: 19, Issue:16 ISSN: 1464-3405 | Synthesis and evaluation of novel F-18 labeled fluoroarylvaline derivatives: potential PET imaging agents for tumor detection. |
AID696412 | Drug uptake in BALB/c mouse heart xenografted with mouse Colon 26 cells at 150 uCi administered parenterally after 2 hrs by PET analysis | 2011 | Journal of medicinal chemistry, Oct-13, Volume: 54, Issue:19 ISSN: 1520-4804 | In vitro cellular uptake and dimerization of signal transducer and activator of transcription-3 (STAT3) identify the photosensitizing and imaging-potential of isomeric photosensitizers derived from chlorophyll-a and bacteriochlorophyll-a. |
AID696422 | Ratio of drug uptake in tumor to heart of mouse Colon 26 cells xenografted BALB/c mouse at 150 uCi administered parenterally after 2 hrs by PET analysis | 2011 | Journal of medicinal chemistry, Oct-13, Volume: 54, Issue:19 ISSN: 1520-4804 | In vitro cellular uptake and dimerization of signal transducer and activator of transcription-3 (STAT3) identify the photosensitizing and imaging-potential of isomeric photosensitizers derived from chlorophyll-a and bacteriochlorophyll-a. |
AID554339 | Drug uptake in human HT-29 cells at 250 kBq after 20 mins by gamma-counting in presence of D-glucose | 2011 | Journal of medicinal chemistry, Jan-13, Volume: 54, Issue:1 ISSN: 1520-4804 | 4-[18F]fluoroglutamic acid (BAY 85-8050), a new amino acid radiotracer for PET imaging of tumors: synthesis and in vitro characterization. |
AID696414 | Ratio of drug uptake in tumor to blood of mouse Colon 26 cells xenografted BALB/c mouse at 150 uCi administered parenterally after 2 hrs by PET analysis | 2011 | Journal of medicinal chemistry, Oct-13, Volume: 54, Issue:19 ISSN: 1520-4804 | In vitro cellular uptake and dimerization of signal transducer and activator of transcription-3 (STAT3) identify the photosensitizing and imaging-potential of isomeric photosensitizers derived from chlorophyll-a and bacteriochlorophyll-a. |
AID476241 | Ratio of drug uptake in tumor to blood of mouse S180 cells xenografted Kunming mouse at 10 to 20 uCi, iv after 30 mins by gamma counting | 2010 | Bioorganic & medicinal chemistry, Apr-01, Volume: 18, Issue:7 ISSN: 1464-3391 | (18)F Labeled benzimidazole derivatives as potential radiotracer for positron emission tomography (PET) tumor imaging. |
AID434407 | Biodistribution in S180 tumor-bearing KM mouse heart assessed per gram of tissue weight at 240 to 370 kBq, iv after 60 mins | 2009 | Bioorganic & medicinal chemistry letters, Aug-15, Volume: 19, Issue:16 ISSN: 1464-3405 | Synthesis and evaluation of novel F-18 labeled fluoroarylvaline derivatives: potential PET imaging agents for tumor detection. |
AID696417 | Ratio of drug uptake in tumor to kidney of mouse Colon 26 cells xenografted BALB/c mouse at 150 uCi administered parenterally after 2 hrs by PET analysis | 2011 | Journal of medicinal chemistry, Oct-13, Volume: 54, Issue:19 ISSN: 1520-4804 | In vitro cellular uptake and dimerization of signal transducer and activator of transcription-3 (STAT3) identify the photosensitizing and imaging-potential of isomeric photosensitizers derived from chlorophyll-a and bacteriochlorophyll-a. |
AID434404 | Biodistribution in S180 tumor-bearing KM mouse liver assessed per gram of tissue weight at 240 to 370 kBq, iv after 15 mins | 2009 | Bioorganic & medicinal chemistry letters, Aug-15, Volume: 19, Issue:16 ISSN: 1464-3405 | Synthesis and evaluation of novel F-18 labeled fluoroarylvaline derivatives: potential PET imaging agents for tumor detection. |
AID476222 | Biodistribution in mouse S180 cells xenografted Kunming mouse kidney at 10 to 20 uCi, iv after 15 mins by gamma counting | 2010 | Bioorganic & medicinal chemistry, Apr-01, Volume: 18, Issue:7 ISSN: 1464-3391 | (18)F Labeled benzimidazole derivatives as potential radiotracer for positron emission tomography (PET) tumor imaging. |
AID434429 | Ratio of drug level in S180 tumor to blood in KM mouse at 240 to 370 kBq, iv after 120 mins | 2009 | Bioorganic & medicinal chemistry letters, Aug-15, Volume: 19, Issue:16 ISSN: 1464-3405 | Synthesis and evaluation of novel F-18 labeled fluoroarylvaline derivatives: potential PET imaging agents for tumor detection. |
AID434437 | Ratio of drug level in S180 tumor to muscleKM mouse at 240 to 370 kBq, iv after 30 mins | 2009 | Bioorganic & medicinal chemistry letters, Aug-15, Volume: 19, Issue:16 ISSN: 1464-3405 | Synthesis and evaluation of novel F-18 labeled fluoroarylvaline derivatives: potential PET imaging agents for tumor detection. |
AID434397 | Biodistribution in S180 tumor-bearing KM mouse lung assessed per gram of tissue at 240 to 370 kBq, iv after 60 mins | 2009 | Bioorganic & medicinal chemistry letters, Aug-15, Volume: 19, Issue:16 ISSN: 1464-3405 | Synthesis and evaluation of novel F-18 labeled fluoroarylvaline derivatives: potential PET imaging agents for tumor detection. |
AID463664 | Ratio of drug level from tumor to brain of Fischer 344 rat bearing rat 9L cells at 20 uCi, iv after 15 mins | 2010 | Journal of medicinal chemistry, Jan-28, Volume: 53, Issue:2 ISSN: 1520-4804 | Synthesis, radiolabeling, and biological evaluation of (R)- and (S)-2-amino-3-[(18)F]fluoro-2-methylpropanoic acid (FAMP) and (R)- and (S)-3-[(18)F]fluoro-2-methyl-2-N-(methylamino)propanoic acid (NMeFAMP) as potential PET radioligands for imaging brain t |
AID434401 | Biodistribution in S180 tumor-bearing KM mouse liver assessed per gram of tissue at 240 to 370 kBq, iv after 120 mins | 2009 | Bioorganic & medicinal chemistry letters, Aug-15, Volume: 19, Issue:16 ISSN: 1464-3405 | Synthesis and evaluation of novel F-18 labeled fluoroarylvaline derivatives: potential PET imaging agents for tumor detection. |
AID476254 | Ratio of drug uptake in tumor to blood of mouse S180 cells xenografted Kunming mouse at 10 to 20 uCi, iv after 60 mins by gamma counting | 2010 | Bioorganic & medicinal chemistry, Apr-01, Volume: 18, Issue:7 ISSN: 1464-3391 | (18)F Labeled benzimidazole derivatives as potential radiotracer for positron emission tomography (PET) tumor imaging. |
AID434427 | Ratio of drug level in S180 tumor to blood in KM mouse at 240 to 370 kBq, iv after 30mins | 2009 | Bioorganic & medicinal chemistry letters, Aug-15, Volume: 19, Issue:16 ISSN: 1464-3405 | Synthesis and evaluation of novel F-18 labeled fluoroarylvaline derivatives: potential PET imaging agents for tumor detection. |
AID476251 | Biodistribution in mouse S180 cells xenografted Kunming mouse blood at 10 to 20 uCi, iv after 60 mins by gamma counting | 2010 | Bioorganic & medicinal chemistry, Apr-01, Volume: 18, Issue:7 ISSN: 1464-3391 | (18)F Labeled benzimidazole derivatives as potential radiotracer for positron emission tomography (PET) tumor imaging. |
AID696419 | Ratio of drug uptake in tumor to stomach of mouse Colon 26 cells xenografted BALB/c mouse at 150 uCi administered parenterally after 2 hrs by PET analysis | 2011 | Journal of medicinal chemistry, Oct-13, Volume: 54, Issue:19 ISSN: 1520-4804 | In vitro cellular uptake and dimerization of signal transducer and activator of transcription-3 (STAT3) identify the photosensitizing and imaging-potential of isomeric photosensitizers derived from chlorophyll-a and bacteriochlorophyll-a. |
AID476226 | Biodistribution in mouse S180 cells xenografted Kunming mouse brain at 10 to 20 uCi, iv after 15 mins by gamma counting | 2010 | Bioorganic & medicinal chemistry, Apr-01, Volume: 18, Issue:7 ISSN: 1464-3391 | (18)F Labeled benzimidazole derivatives as potential radiotracer for positron emission tomography (PET) tumor imaging. |
AID434375 | Biodistribution in S180 tumor-bearing KM mouse brain assessed per gram of tissue at 240 to 370 kBq, iv after 5 mins | 2009 | Bioorganic & medicinal chemistry letters, Aug-15, Volume: 19, Issue:16 ISSN: 1464-3405 | Synthesis and evaluation of novel F-18 labeled fluoroarylvaline derivatives: potential PET imaging agents for tumor detection. |
AID476233 | Biodistribution in mouse S180 cells xenografted Kunming mouse pancreas at 10 to 20 uCi, iv after 30 mins by gamma counting | 2010 | Bioorganic & medicinal chemistry, Apr-01, Volume: 18, Issue:7 ISSN: 1464-3391 | (18)F Labeled benzimidazole derivatives as potential radiotracer for positron emission tomography (PET) tumor imaging. |
AID434382 | Biodistribution in S180 tumor-bearing KM mouse muscle assessed per gram of tissue at 240 to 370 kBq, iv after 60 mins | 2009 | Bioorganic & medicinal chemistry letters, Aug-15, Volume: 19, Issue:16 ISSN: 1464-3405 | Synthesis and evaluation of novel F-18 labeled fluoroarylvaline derivatives: potential PET imaging agents for tumor detection. |
AID696413 | Drug uptake in BALB/c mouse tumor xenografted with mouse Colon 26 cells at 150 uCi administered parenterally after 2 hrs by PET analysis | 2011 | Journal of medicinal chemistry, Oct-13, Volume: 54, Issue:19 ISSN: 1520-4804 | In vitro cellular uptake and dimerization of signal transducer and activator of transcription-3 (STAT3) identify the photosensitizing and imaging-potential of isomeric photosensitizers derived from chlorophyll-a and bacteriochlorophyll-a. |
AID434391 | Biodistribution in S180 tumor-bearing KM mouse kidney assessed per gram of tissue at 240 to 370 kBq, iv after 120 mins | 2009 | Bioorganic & medicinal chemistry letters, Aug-15, Volume: 19, Issue:16 ISSN: 1464-3405 | Synthesis and evaluation of novel F-18 labeled fluoroarylvaline derivatives: potential PET imaging agents for tumor detection. |
AID476258 | Biodistribution in mouse S180 cells xenografted Kunming mouse liver at 10 to 20 uCi, iv after 120 mins by gamma counting | 2010 | Bioorganic & medicinal chemistry, Apr-01, Volume: 18, Issue:7 ISSN: 1464-3391 | (18)F Labeled benzimidazole derivatives as potential radiotracer for positron emission tomography (PET) tumor imaging. |
AID434406 | Biodistribution in S180 tumor-bearing KM mouse heart assessed per gram of tissue weight at 240 to 370 kBq, iv after 120 mins | 2009 | Bioorganic & medicinal chemistry letters, Aug-15, Volume: 19, Issue:16 ISSN: 1464-3405 | Synthesis and evaluation of novel F-18 labeled fluoroarylvaline derivatives: potential PET imaging agents for tumor detection. |
AID476260 | Biodistribution in mouse S180 cells xenografted Kunming mouse lung at 10 to 20 uCi, iv after 120 mins by gamma counting | 2010 | Bioorganic & medicinal chemistry, Apr-01, Volume: 18, Issue:7 ISSN: 1464-3391 | (18)F Labeled benzimidazole derivatives as potential radiotracer for positron emission tomography (PET) tumor imaging. |
AID476209 | Biodistribution in mouse S180 cells xenografted Kunming mouse kidney at 10 to 20 uCi, iv after 5 mins by gamma counting | 2010 | Bioorganic & medicinal chemistry, Apr-01, Volume: 18, Issue:7 ISSN: 1464-3391 | (18)F Labeled benzimidazole derivatives as potential radiotracer for positron emission tomography (PET) tumor imaging. |
AID434431 | Ratio of drug level in S180 tumor to brain KM mouse at 240 to 370 kBq, iv after 15 mins | 2009 | Bioorganic & medicinal chemistry letters, Aug-15, Volume: 19, Issue:16 ISSN: 1464-3405 | Synthesis and evaluation of novel F-18 labeled fluoroarylvaline derivatives: potential PET imaging agents for tumor detection. |
AID434418 | Biodistribution in S180 tumor-bearing KM mouse brain assessed per gram of tissue at 240 to 370 kBq, iv after 60 mins | 2009 | Bioorganic & medicinal chemistry letters, Aug-15, Volume: 19, Issue:16 ISSN: 1464-3405 | Synthesis and evaluation of novel F-18 labeled fluoroarylvaline derivatives: potential PET imaging agents for tumor detection. |
AID434394 | Biodistribution in S180 tumor-bearing KM mouse kidney assessed per gram of tissue at 240 to 370 kBq, iv after 15 mins | 2009 | Bioorganic & medicinal chemistry letters, Aug-15, Volume: 19, Issue:16 ISSN: 1464-3405 | Synthesis and evaluation of novel F-18 labeled fluoroarylvaline derivatives: potential PET imaging agents for tumor detection. |
AID434383 | Biodistribution in S180 tumor-bearing KM mouse muscle assessed per gram of tissue at 240 to 370 kBq, iv after 30 mins | 2009 | Bioorganic & medicinal chemistry letters, Aug-15, Volume: 19, Issue:16 ISSN: 1464-3405 | Synthesis and evaluation of novel F-18 labeled fluoroarylvaline derivatives: potential PET imaging agents for tumor detection. |
AID434415 | Biodistribution in S180 tumor-bearing KM mouse blood assessed per gram of tissue weight at 240 to 370 kBq, iv after 5 mins | 2009 | Bioorganic & medicinal chemistry letters, Aug-15, Volume: 19, Issue:16 ISSN: 1464-3405 | Synthesis and evaluation of novel F-18 labeled fluoroarylvaline derivatives: potential PET imaging agents for tumor detection. |
AID434379 | Biodistribution in S180 tumor-bearing KM mouse spleen assessed per gram of tissue at 240 to 370 kBq, iv after 15 mins | 2009 | Bioorganic & medicinal chemistry letters, Aug-15, Volume: 19, Issue:16 ISSN: 1464-3405 | Synthesis and evaluation of novel F-18 labeled fluoroarylvaline derivatives: potential PET imaging agents for tumor detection. |
AID476224 | Biodistribution in mouse S180 cells xenografted Kunming mouse muscle at 10 to 20 uCi, iv after 15 mins by gamma counting | 2010 | Bioorganic & medicinal chemistry, Apr-01, Volume: 18, Issue:7 ISSN: 1464-3391 | (18)F Labeled benzimidazole derivatives as potential radiotracer for positron emission tomography (PET) tumor imaging. |
AID434398 | Biodistribution in S180 tumor-bearing KM mouse lung assessed per gram of tissue at 240 to 370 kBq, iv after 30 mins | 2009 | Bioorganic & medicinal chemistry letters, Aug-15, Volume: 19, Issue:16 ISSN: 1464-3405 | Synthesis and evaluation of novel F-18 labeled fluoroarylvaline derivatives: potential PET imaging agents for tumor detection. |
AID696411 | Drug uptake in BALB/c mouse muscle xenografted with mouse Colon 26 cells at 150 uCi administered parenterally after 2 hrs by PET analysis | 2011 | Journal of medicinal chemistry, Oct-13, Volume: 54, Issue:19 ISSN: 1520-4804 | In vitro cellular uptake and dimerization of signal transducer and activator of transcription-3 (STAT3) identify the photosensitizing and imaging-potential of isomeric photosensitizers derived from chlorophyll-a and bacteriochlorophyll-a. |
AID476256 | Ratio of drug uptake in tumor to brain of mouse S180 cells xenografted Kunming mouse at 10 to 20 uCi, iv after 60 mins by gamma counting | 2010 | Bioorganic & medicinal chemistry, Apr-01, Volume: 18, Issue:7 ISSN: 1464-3391 | (18)F Labeled benzimidazole derivatives as potential radiotracer for positron emission tomography (PET) tumor imaging. |
AID476259 | Biodistribution in mouse S180 cells xenografted Kunming mouse pancreas at 10 to 20 uCi, iv after 120 mins by gamma counting | 2010 | Bioorganic & medicinal chemistry, Apr-01, Volume: 18, Issue:7 ISSN: 1464-3391 | (18)F Labeled benzimidazole derivatives as potential radiotracer for positron emission tomography (PET) tumor imaging. |
AID434424 | Biodistribution in S180 tumor present in KM mouse assessed per gram of tissue at 240 to 370 kBq, iv after 120 mins | 2009 | Bioorganic & medicinal chemistry letters, Aug-15, Volume: 19, Issue:16 ISSN: 1464-3405 | Synthesis and evaluation of novel F-18 labeled fluoroarylvaline derivatives: potential PET imaging agents for tumor detection. |
AID434410 | Biodistribution in S180 tumor-bearing KM mouse heart assessed per gram of tissue weight at 240 to 370 kBq, iv after 5 mins | 2009 | Bioorganic & medicinal chemistry letters, Aug-15, Volume: 19, Issue:16 ISSN: 1464-3405 | Synthesis and evaluation of novel F-18 labeled fluoroarylvaline derivatives: potential PET imaging agents for tumor detection. |
AID434425 | Ratio of drug level in S180 tumor to blood in KM mouse at 240 to 370 kBq, iv after 5mins | 2009 | Bioorganic & medicinal chemistry letters, Aug-15, Volume: 19, Issue:16 ISSN: 1464-3405 | Synthesis and evaluation of novel F-18 labeled fluoroarylvaline derivatives: potential PET imaging agents for tumor detection. |
AID434377 | Biodistribution in S180 tumor-bearing KM mouse spleen assessed per gram of tissue at 240 to 370 kBq, iv after 60 mins | 2009 | Bioorganic & medicinal chemistry letters, Aug-15, Volume: 19, Issue:16 ISSN: 1464-3405 | Synthesis and evaluation of novel F-18 labeled fluoroarylvaline derivatives: potential PET imaging agents for tumor detection. |
AID476238 | Biodistribution in mouse S180 cells xenografted Kunming mouse blood at 10 to 20 uCi, iv after 30 mins by gamma counting | 2010 | Bioorganic & medicinal chemistry, Apr-01, Volume: 18, Issue:7 ISSN: 1464-3391 | (18)F Labeled benzimidazole derivatives as potential radiotracer for positron emission tomography (PET) tumor imaging. |
AID696415 | Ratio of drug uptake in tumor to muscle of mouse Colon 26 cells xenografted BALB/c mouse at 150 uCi administered parenterally after 2 hrs by PET analysis | 2011 | Journal of medicinal chemistry, Oct-13, Volume: 54, Issue:19 ISSN: 1520-4804 | In vitro cellular uptake and dimerization of signal transducer and activator of transcription-3 (STAT3) identify the photosensitizing and imaging-potential of isomeric photosensitizers derived from chlorophyll-a and bacteriochlorophyll-a. |
AID476253 | Biodistribution in mouse S180 cells xenografted Kunming mouse tumor at 10 to 20 uCi, iv after 60 mins by gamma counting | 2010 | Bioorganic & medicinal chemistry, Apr-01, Volume: 18, Issue:7 ISSN: 1464-3391 | (18)F Labeled benzimidazole derivatives as potential radiotracer for positron emission tomography (PET) tumor imaging. |
AID434376 | Biodistribution in S180 tumor-bearing KM mouse spleen assessed per gram of tissue at 240 to 370 kBq, iv after 120 mins | 2009 | Bioorganic & medicinal chemistry letters, Aug-15, Volume: 19, Issue:16 ISSN: 1464-3405 | Synthesis and evaluation of novel F-18 labeled fluoroarylvaline derivatives: potential PET imaging agents for tumor detection. |
AID434400 | Biodistribution in S180 tumor-bearing KM mouse lung assessed per gram of tissue at 240 to 370 kBq, iv after 5 mins | 2009 | Bioorganic & medicinal chemistry letters, Aug-15, Volume: 19, Issue:16 ISSN: 1464-3405 | Synthesis and evaluation of novel F-18 labeled fluoroarylvaline derivatives: potential PET imaging agents for tumor detection. |
AID476421 | Ratio of drug uptake in tumor to brain of mouse S180 cells xenografted Kunming mouse at 10 to 20 uCi, iv after 120 mins by gamma counting | 2010 | Bioorganic & medicinal chemistry, Apr-01, Volume: 18, Issue:7 ISSN: 1464-3391 | (18)F Labeled benzimidazole derivatives as potential radiotracer for positron emission tomography (PET) tumor imaging. |
AID663137 | Ratio of drug level in tumor to liver in rat TAA-induced cholangiocarcinoma model | 2012 | Bioorganic & medicinal chemistry letters, Jun-15, Volume: 22, Issue:12 ISSN: 1464-3405 | Synthesis and evaluation of [18F]Fluorobutyl ethacrynic amide: a potential PET tracer for studying glutathione transferase. |
AID434417 | Biodistribution in S180 tumor-bearing KM mouse brain assessed per gram of tissue at 240 to 370 kBq, iv after 30 mins | 2009 | Bioorganic & medicinal chemistry letters, Aug-15, Volume: 19, Issue:16 ISSN: 1464-3405 | Synthesis and evaluation of novel F-18 labeled fluoroarylvaline derivatives: potential PET imaging agents for tumor detection. |
AID434409 | Biodistribution in S180 tumor-bearing KM mouse heart assessed per gram of tissue weight at 240 to 370 kBq, iv after 15 mins | 2009 | Bioorganic & medicinal chemistry letters, Aug-15, Volume: 19, Issue:16 ISSN: 1464-3405 | Synthesis and evaluation of novel F-18 labeled fluoroarylvaline derivatives: potential PET imaging agents for tumor detection. |
AID476218 | Biodistribution in mouse S180 cells xenografted Kunming mouse heart at 10 to 20 uCi, iv after 15 mins by gamma counting | 2010 | Bioorganic & medicinal chemistry, Apr-01, Volume: 18, Issue:7 ISSN: 1464-3391 | (18)F Labeled benzimidazole derivatives as potential radiotracer for positron emission tomography (PET) tumor imaging. |
AID476235 | Biodistribution in mouse S180 cells xenografted Kunming mouse kidney at 10 to 20 uCi, iv after 30 mins by gamma counting | 2010 | Bioorganic & medicinal chemistry, Apr-01, Volume: 18, Issue:7 ISSN: 1464-3391 | (18)F Labeled benzimidazole derivatives as potential radiotracer for positron emission tomography (PET) tumor imaging. |
AID476217 | Ratio of drug uptake in tumor to brain of mouse S180 cells xenografted Kunming mouse at 10 to 20 uCi, iv after 5 mins by gamma counting | 2010 | Bioorganic & medicinal chemistry, Apr-01, Volume: 18, Issue:7 ISSN: 1464-3391 | (18)F Labeled benzimidazole derivatives as potential radiotracer for positron emission tomography (PET) tumor imaging. |
AID476214 | Biodistribution in mouse S180 cells xenografted Kunming mouse tumor at 10 to 20 uCi, iv after 5 mins by gamma counting | 2010 | Bioorganic & medicinal chemistry, Apr-01, Volume: 18, Issue:7 ISSN: 1464-3391 | (18)F Labeled benzimidazole derivatives as potential radiotracer for positron emission tomography (PET) tumor imaging. |
AID434385 | Biodistribution in S180 tumor-bearing KM mouse muscle assessed per gram of tissue at 240 to 370 kBq, iv after 5 mins | 2009 | Bioorganic & medicinal chemistry letters, Aug-15, Volume: 19, Issue:16 ISSN: 1464-3405 | Synthesis and evaluation of novel F-18 labeled fluoroarylvaline derivatives: potential PET imaging agents for tumor detection. |
AID476265 | Biodistribution in mouse S180 cells xenografted Kunming mouse brain at 10 to 20 uCi, iv after 120 mins by gamma counting | 2010 | Bioorganic & medicinal chemistry, Apr-01, Volume: 18, Issue:7 ISSN: 1464-3391 | (18)F Labeled benzimidazole derivatives as potential radiotracer for positron emission tomography (PET) tumor imaging. |
AID476205 | Biodistribution in mouse S180 cells xenografted Kunming mouse heart at 10 to 20 uCi, iv after 5 mins by gamma counting | 2010 | Bioorganic & medicinal chemistry, Apr-01, Volume: 18, Issue:7 ISSN: 1464-3391 | (18)F Labeled benzimidazole derivatives as potential radiotracer for positron emission tomography (PET) tumor imaging. |
AID434378 | Biodistribution in S180 tumor-bearing KM mouse spleen assessed per gram of tissue at 240 to 370 kBq, iv after 30 mins | 2009 | Bioorganic & medicinal chemistry letters, Aug-15, Volume: 19, Issue:16 ISSN: 1464-3405 | Synthesis and evaluation of novel F-18 labeled fluoroarylvaline derivatives: potential PET imaging agents for tumor detection. |
AID554338 | Drug uptake in human A549 cells at 250 kBq after 30 mins by gamma-counting in presence of D-glucose | 2011 | Journal of medicinal chemistry, Jan-13, Volume: 54, Issue:1 ISSN: 1520-4804 | 4-[18F]fluoroglutamic acid (BAY 85-8050), a new amino acid radiotracer for PET imaging of tumors: synthesis and in vitro characterization. |
AID476240 | Biodistribution in mouse S180 cells xenografted Kunming mouse tumor at 10 to 20 uCi, iv after 30 mins by gamma counting | 2010 | Bioorganic & medicinal chemistry, Apr-01, Volume: 18, Issue:7 ISSN: 1464-3391 | (18)F Labeled benzimidazole derivatives as potential radiotracer for positron emission tomography (PET) tumor imaging. |
AID434432 | Ratio of drug level in S180 tumor to brain KM mouse at 240 to 370 kBq, iv after 30 mins | 2009 | Bioorganic & medicinal chemistry letters, Aug-15, Volume: 19, Issue:16 ISSN: 1464-3405 | Synthesis and evaluation of novel F-18 labeled fluoroarylvaline derivatives: potential PET imaging agents for tumor detection. |
AID410814 | Biodistribution in tumor of iv dosed BALB/c mouse bearing mouse Colon-26 cells assessed as relative uptake value after 48 hrs by PET imaging | 2009 | Journal of medicinal chemistry, Jan-22, Volume: 52, Issue:2 ISSN: 1520-4804 | Comparative positron-emission tomography (PET) imaging and phototherapeutic potential of 124I- labeled methyl- 3-(1'-iodobenzyloxyethyl)pyropheophorbide-a vs the corresponding glucose and galactose conjugates. |
AID476219 | Biodistribution in mouse S180 cells xenografted Kunming mouse liver at 10 to 20 uCi, iv after 15 mins by gamma counting | 2010 | Bioorganic & medicinal chemistry, Apr-01, Volume: 18, Issue:7 ISSN: 1464-3391 | (18)F Labeled benzimidazole derivatives as potential radiotracer for positron emission tomography (PET) tumor imaging. |
AID696420 | Ratio of drug uptake in tumor to gut of mouse Colon 26 cells xenografted BALB/c mouse at 150 uCi administered parenterally after 2 hrs by PET analysis | 2011 | Journal of medicinal chemistry, Oct-13, Volume: 54, Issue:19 ISSN: 1520-4804 | In vitro cellular uptake and dimerization of signal transducer and activator of transcription-3 (STAT3) identify the photosensitizing and imaging-potential of isomeric photosensitizers derived from chlorophyll-a and bacteriochlorophyll-a. |
AID476257 | Biodistribution in mouse S180 cells xenografted Kunming mouse heart at 10 to 20 uCi, iv after 120 mins by gamma counting | 2010 | Bioorganic & medicinal chemistry, Apr-01, Volume: 18, Issue:7 ISSN: 1464-3391 | (18)F Labeled benzimidazole derivatives as potential radiotracer for positron emission tomography (PET) tumor imaging. |
AID434433 | Ratio of drug level in S180 tumor to brain KM mouse at 240 to 370 kBq, iv after 60 mins | 2009 | Bioorganic & medicinal chemistry letters, Aug-15, Volume: 19, Issue:16 ISSN: 1464-3405 | Synthesis and evaluation of novel F-18 labeled fluoroarylvaline derivatives: potential PET imaging agents for tumor detection. |
AID476250 | Biodistribution in mouse S180 cells xenografted Kunming mouse muscle at 10 to 20 uCi, iv after 60 mins by gamma counting | 2010 | Bioorganic & medicinal chemistry, Apr-01, Volume: 18, Issue:7 ISSN: 1464-3391 | (18)F Labeled benzimidazole derivatives as potential radiotracer for positron emission tomography (PET) tumor imaging. |
AID476244 | Biodistribution in mouse S180 cells xenografted Kunming mouse heart at 10 to 20 uCi, iv after 60 mins by gamma counting | 2010 | Bioorganic & medicinal chemistry, Apr-01, Volume: 18, Issue:7 ISSN: 1464-3391 | (18)F Labeled benzimidazole derivatives as potential radiotracer for positron emission tomography (PET) tumor imaging. |
AID434414 | Biodistribution in S180 tumor-bearing KM mouse blood assessed per gram of tissue weight at 240 to 370 kBq, iv after 15 mins | 2009 | Bioorganic & medicinal chemistry letters, Aug-15, Volume: 19, Issue:16 ISSN: 1464-3405 | Synthesis and evaluation of novel F-18 labeled fluoroarylvaline derivatives: potential PET imaging agents for tumor detection. |
AID696421 | Ratio of drug uptake in tumor to liver of mouse Colon 26 cells xenografted BALB/c mouse at 150 uCi administered parenterally after 2 hrs by PET analysis | 2011 | Journal of medicinal chemistry, Oct-13, Volume: 54, Issue:19 ISSN: 1520-4804 | In vitro cellular uptake and dimerization of signal transducer and activator of transcription-3 (STAT3) identify the photosensitizing and imaging-potential of isomeric photosensitizers derived from chlorophyll-a and bacteriochlorophyll-a. |
AID434438 | Ratio of drug level in S180 tumor to muscleKM mouse at 240 to 370 kBq, iv after 60 mins | 2009 | Bioorganic & medicinal chemistry letters, Aug-15, Volume: 19, Issue:16 ISSN: 1464-3405 | Synthesis and evaluation of novel F-18 labeled fluoroarylvaline derivatives: potential PET imaging agents for tumor detection. |
AID476234 | Biodistribution in mouse S180 cells xenografted Kunming mouse lung at 10 to 20 uCi, iv after 30 mins by gamma counting | 2010 | Bioorganic & medicinal chemistry, Apr-01, Volume: 18, Issue:7 ISSN: 1464-3391 | (18)F Labeled benzimidazole derivatives as potential radiotracer for positron emission tomography (PET) tumor imaging. |
AID476212 | Biodistribution in mouse S180 cells xenografted Kunming mouse blood at 10 to 20 uCi, iv after 5 mins by gamma counting | 2010 | Bioorganic & medicinal chemistry, Apr-01, Volume: 18, Issue:7 ISSN: 1464-3391 | (18)F Labeled benzimidazole derivatives as potential radiotracer for positron emission tomography (PET) tumor imaging. |
AID476229 | Ratio of drug uptake in tumor to muscle of mouse S180 cells xenografted Kunming mouse at 10 to 20 uCi, iv after 15 mins by gamma counting | 2010 | Bioorganic & medicinal chemistry, Apr-01, Volume: 18, Issue:7 ISSN: 1464-3391 | (18)F Labeled benzimidazole derivatives as potential radiotracer for positron emission tomography (PET) tumor imaging. |
AID476245 | Biodistribution in mouse S180 cells xenografted Kunming mouse liver at 10 to 20 uCi, iv after 60 mins by gamma counting | 2010 | Bioorganic & medicinal chemistry, Apr-01, Volume: 18, Issue:7 ISSN: 1464-3391 | (18)F Labeled benzimidazole derivatives as potential radiotracer for positron emission tomography (PET) tumor imaging. |
Timeframe | Studies, This Drug (%) | All Drugs % |
---|---|---|
pre-1990 | 0 (0.00) | 18.7374 |
1990's | 0 (0.00) | 18.2507 |
2000's | 2 (22.22) | 29.6817 |
2010's | 7 (77.78) | 24.3611 |
2020's | 0 (0.00) | 2.80 |
Publication Type | This drug (%) | All Drugs (%) |
---|---|---|
Trials | 0 (0.00%) | 5.53% |
Reviews | 0 (0.00%) | 6.00% |
Case Studies | 0 (0.00%) | 4.05% |
Observational | 0 (0.00%) | 0.25% |
Other | 9 (100.00%) | 84.16% |
Substance | Studies | Classes | Roles | First Year | Last Year | Average Age | Relationship Strength | Trials | pre-1990 | 1990's | 2000's | 2010's | post-2020 |
---|---|---|---|---|---|---|---|---|---|---|---|---|---|
ethacrynic acid | aromatic ether; aromatic ketone; dichlorobenzene; monocarboxylic acid | EC 2.5.1.18 (glutathione transferase) inhibitor; ion transport inhibitor; loop diuretic | 2012 | 2012 | 12.0 | high | 0 | 0 | 0 | 0 | 1 | 0 | |
imatinib | aromatic amine; benzamides; N-methylpiperazine; pyridines; pyrimidines | antineoplastic agent; apoptosis inducer; tyrosine kinase inhibitor | 2014 | 2014 | 10.0 | high | 0 | 0 | 0 | 0 | 1 | 0 | |
fluciclovine f-18 | 2010 | 2010 | 14.0 | high | 0 | 0 | 0 | 1 | 0 | 0 | |||
18f-fluoroethyl-l-tyrosine | 2010 | 2010 | 14.0 | high | 0 | 0 | 0 | 1 | 0 | 0 |
Condition | Indicated | Studies | First Year | Last Year | Average Age | Relationship Strength | Trials | pre-1990 | 1990's | 2000's | 2010's | post-2020 |
---|---|---|---|---|---|---|---|---|---|---|---|---|
Benign Neoplasms | 0 | 2009 | 2011 | 14.0 | medium | 0 | 0 | 0 | 2 | 1 | 0 | |
Benign Neoplasms, Brain | 0 | 2010 | 2010 | 14.0 | low | 0 | 0 | 0 | 1 | 0 | 0 | |
Bile Duct Cancer | 0 | 2012 | 2012 | 12.0 | low | 0 | 0 | 0 | 0 | 1 | 0 | |
Bile Duct Neoplasms | 0 | 2012 | 2012 | 12.0 | low | 0 | 0 | 0 | 0 | 1 | 0 | |
Brain Neoplasms | 0 | 2010 | 2010 | 14.0 | low | 0 | 0 | 0 | 1 | 0 | 0 | |
Cholangiocarcinoma | 0 | 2012 | 2012 | 12.0 | low | 0 | 0 | 0 | 0 | 1 | 0 | |
Cholangiocellular Carcinoma | 0 | 2012 | 2012 | 12.0 | low | 0 | 0 | 0 | 0 | 1 | 0 | |
Disease Models, Animal | 0 | 2011 | 2014 | 11.5 | medium | 0 | 0 | 0 | 0 | 2 | 0 | |
Experimental Neoplasms | 0 | 2011 | 2011 | 13.0 | low | 0 | 0 | 0 | 0 | 1 | 0 | |
Neoplasms | 0 | 2009 | 2011 | 14.0 | medium | 0 | 0 | 0 | 2 | 1 | 0 | |
Sarcoma 180 | 0 | 2010 | 2010 | 14.0 | low | 0 | 0 | 0 | 1 | 0 | 0 |