A member of the class of benzamides obtained from formal condensation between the carboxy group of 2-methoxy-5-sulfamoylbenzoic acid and the primary amino group of (1-ethylpyrrolidin-2-yl)methylamine.
ChEBI ID: 32168
Member | Definition | Role |
---|---|---|
(R)-(+)-sulpiride | An optically active form of sulpiride having (R)-configuration. The active enantiomer of the racemic drug sulpiride. | (R)-(+)-sulpiride |
levosulpiride | An optically active form of sulpiride having (S)-configuration. The active enantiomer of the racemic drug sulpiride. Selective D2-like dopamine antagonist (Ki values are ~ 0.015. ~ 0.013, 1, ~ 45 and ~ 77 muM at D2, D3, D4, D1 and D5 receptors respectively). | (S)-(-)-sulpiride |
Timeframe | Studies, Drugs in This Class (%) | All Drugs % |
---|---|---|
pre-1990 | 4 (3.92) | 18.7374 |
1990's | 24 (23.53) | 18.2507 |
2000's | 22 (21.57) | 29.6817 |
2010's | 39 (38.24) | 24.3611 |
2020's | 13 (12.75) | 2.80 |
Publication Type | Studies, Drugs in This Class (%) | All Drugs (%) |
---|---|---|
Trials | 21 (17.80%) | 5.53% |
Reviews | 10 (8.47%) | 6.00% |
Case Studies | 13 (11.02%) | 4.05% |
Observational | 0 (0.00%) | 0.25% |
Other | 74 (62.71%) | 84.16% |